The human T-type amino acid transporter-1: characterization, gene organization, and chromosomal location.

Article Details

Citation

Kim DK, Kanai Y, Matsuo H, Kim JY, Chairoungdua A, Kobayashi Y, Enomoto A, Cha SH, Goya T, Endou H

The human T-type amino acid transporter-1: characterization, gene organization, and chromosomal location.

Genomics. 2002 Jan;79(1):95-103.

PubMed ID
11827462 [ View in PubMed
]
Abstract

System T is a Na+-independent transport system that selectively transports aromatic amino acids. Here, we determined the structure of the human T-type amino-acid transporter-1 (TAT1) cDNA and gene (SLC16A10). The human TAT1 cDNA encoded a 515-amino-acid protein with 12 putative membrane-spanning domains. Human SLC16A10 was localized on human chromosome 6, mapped to 6q21-q22. SLC16A10 contains six exons spanning 136 kb. In contrast to rat TAT1, which is mainly present in the intestine, human TAT1 was strongly expressed in human kidney as well as in human intestine. Expression of human TAT1 in Xenopus laevis oocytes demonstrated the Na+-independent transport of tryptophan, tyrosine, phenylalanine, and L-dopa, indicating that human TAT1 is a transporter subserving system T. Because human TAT1 is proposed to be crucial to the efficient absorption of aromatic amino acids from intestine and kidney, its defect could be involved in the disruption of aromatic amino-acid transport, such as in blue diaper syndrome.

DrugBank Data that Cites this Article

Drug Transporters
DrugTransporterKindOrganismPharmacological ActionActions
2-aminoisobutyric acidMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Details
beta-AlanineMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Details
D-PhenylalanineMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
Glutamic acidMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
GlycineMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
HistidineMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
Lactic acidMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
LeucineMonocarboxylate transporter 10ProteinHumans
Unknown
Inhibitor
Details
LysineMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
PhenylalanineMonocarboxylate transporter 10ProteinHumans
Unknown
Inhibitor
Details
Pyruvic acidMonocarboxylate transporter 10ProteinHumans
Unknown
Substrate
Inhibitor
Details
TryptophanMonocarboxylate transporter 10ProteinHumans
Unknown
Inhibitor
Details
TyrosineMonocarboxylate transporter 10ProteinHumans
Unknown
Inhibitor
Details
Polypeptides
NameUniProt ID
Monocarboxylate transporter 10Q8TF71Details