(R)-Rolipram | cAMP-specific 3',5'-cyclic phosphodiesterase 4B | Protein | Humans | Unknown | Inhibitor | Details |
(S)-Rolipram | cAMP-specific 3',5'-cyclic phosphodiesterase 4B | Protein | Humans | Unknown | Inhibitor | Details |
1-Guanidinium-7-Aminoheptane | Deoxyhypusine synthase | Protein | Humans | Unknown | Inhibitor | Details |
3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Fibroblast growth factor receptor 2 | Protein | Humans | Unknown | Not Available | Details |
3-Methylthiofentanyl | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Abatacept | T-lymphocyte activation antigen CD80 | Protein | Humans | Yes | Antagonist | Details |
Abatacept | T-lymphocyte activation antigen CD86 | Protein | Humans | Yes | Antagonist | Details |
Abciximab | Integrin beta-3 | Protein | Humans | Yes | Antagonist | Details |
Acebutolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Partial agonist | Details |
Acenocoumarol | Vitamin K epoxide reductase complex subunit 1 | Protein | Humans | Yes | Inhibitor | Details |
Acepromazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Aceprometazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Acetaminophen | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Acetaminophen | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Acetohydroxamic acid | Urease subunit alpha | Protein | Enterobacter aerogenes | Yes | Inhibitor | Details |
Acetophenazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Adenosine | Adenosine receptor A3 | Protein | Humans | Yes | Agonist | Details |
Adenosine phosphate | Adenylate cyclase type 1 | Protein | Humans | Unknown | Product of | Details |
Alanine | 4-aminobutyrate aminotransferase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Aldesleukin | Interleukin-2 receptor subunit alpha | Protein | Humans | Yes | Agonist Modulator | Details |
Aldesleukin | Interleukin-2 receptor subunit beta | Protein | Humans | Yes | Agonist Modulator | Details |
Alefacept | T-cell surface antigen CD2 | Protein | Humans | Yes | Inhibitor Antibody Regulator | Details |
Alemtuzumab | CAMPATH-1 antigen | Protein | Humans | Yes | Antibody | Details |
Alendronic acid | Farnesyl pyrophosphate synthase | Protein | Humans | Yes | Inhibitor | Details |
Alendronic acid | Receptor-type tyrosine-protein phosphatase S | Protein | Humans | Unknown | Inhibitor | Details |
Alfacalcidol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Alfentanil | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Alimemazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Alitretinoin | Retinoic acid receptor alpha | Protein | Humans | Yes | Agonist | Details |
Allopurinol | Xanthine dehydrogenase/oxidase | Protein | Humans | Yes | Inhibitor | Details |
Almitrine | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Yes | Binder | Details |
Almotriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Unknown | Agonist | Details |
Almotriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Unknown | Agonist | Details |
Alosetron | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Alpha-1-proteinase inhibitor | Neutrophil elastase | Protein | Humans | Yes | Inhibitor | Details |
Alprenolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Alsterpaullone | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Alsterpaullone | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Not Available | Details |
Aluminium | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Unknown | Binder | Details |
Aluminium monostearate | Troponin C, slow skeletal and cardiac muscles | Protein | Humans | Unknown | Stimulator | Details |
Aluminium phosphate | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Unknown | Not Available | Details |
Aluminum acetate | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Unknown | Not Available | Details |
Alvimopan | Mu-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Alvocidib | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Alvocidib | Cyclin-dependent kinase 4 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 6 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 7 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 8 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Cyclin-dependent kinase 9 | Protein | Humans | Unknown | Not Available | Details |
Alvocidib | Epidermal growth factor receptor | Protein | Humans | Unknown | Not Available | Details |
Ambenonium | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Amiloride | Amiloride-sensitive sodium channel subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Amiloride | Urokinase-type plasminogen activator | Protein | Humans | Unknown | Inhibitor | Details |
Aminocaproic acid | Plasminogen | Protein | Humans | Yes | Inhibitor | Details |
Aminoglutethimide | Cholesterol side-chain cleavage enzyme, mitochondrial | Protein | Humans | Yes | Inhibitor | Details |
Aminoglutethimide | Cytochrome P450 19A1 | Protein | Humans | Yes | Inhibitor | Details |
Aminolevulinic acid | Delta-aminolevulinic acid dehydratase | Protein | Humans | Yes | Inducer | Details |
Aminophylline | cGMP-inhibited 3',5'-cyclic phosphodiesterase A | Protein | Humans | Yes | Inhibitor | Details |
Amobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Amodiaquine | Histamine N-methyltransferase | Protein | Humans | Unknown | Inhibitor | Details |
Amrinone | cGMP-inhibited 3',5'-cyclic phosphodiesterase A | Protein | Humans | Yes | Inhibitor | Details |
Amsacrine | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Anakinra | Interleukin-1 receptor type 1 | Protein | Humans | Yes | Antagonist | Details |
Anileridine | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Anisindione | Vitamin K-dependent gamma-carboxylase | Protein | Humans | Yes | Inhibitor | Details |
Anistreplase | Plasminogen | Protein | Humans | Yes | Activator | Details |
Antithymocyte immunoglobulin (rabbit) | T-cell surface glycoprotein CD1a | Protein | Humans | Unknown | Inhibitor | Details |
Antrafenine | Prostaglandin G/H synthase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Apomorphine | Dopamine D1 receptor | Protein | Humans | Unknown | Agonist | Details |
Apomorphine | Dopamine D2 receptor | Protein | Humans | Yes | Agonist | Details |
Apomorphine | Dopamine D3 receptor | Protein | Humans | Yes | Agonist | Details |
Apomorphine | Dopamine D4 receptor | Protein | Humans | Yes | Agonist | Details |
Apomorphine | Dopamine D5 receptor | Protein | Humans | Unknown | Agonist | Details |
Aprepitant | Neurokinin 1 receptor | Protein | Humans | Yes | Antagonist | Details |
Arbaclofen | Gamma-aminobutyric acid type B receptor subunit 1 | Protein | Humans | Yes | Agonist | Details |
Arbaclofen Placarbil | Gamma-aminobutyric acid type B receptor subunit 1 | Protein | Humans | Yes | Agonist | Details |
Ardeparin | Heparin cofactor 2 | Protein | Humans | Yes | Agonist | Details |
Arformoterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Argatroban | Prothrombin | Protein | Humans | Yes | Inhibitor | Details |
Aripiprazole | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist Partial agonist | Details |
Aripiprazole lauroxil | Dopamine D2 receptor | Protein | Humans | Yes | Partial agonist | Details |
Arsenic trioxide | Inhibitor of nuclear factor kappa-B kinase subunit beta | Protein | Humans | Yes | Inducer | Details |
Ascorbic acid | Procollagen-lysine,2-oxoglutarate 5-dioxygenase 1 | Protein | Humans | Unknown | Cofactor | Details |
Astemizole | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Atazanavir | Human immunodeficiency virus type 1 protease | Protein | Human immunodeficiency virus 1 | Yes | Inhibitor | Details |
Atenolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Atorvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Atovaquone | Dihydroorotate dehydrogenase (quinone), mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Atovaquone | Dihydroorotate dehydrogenase (quinone), mitochondrial | Protein | Plasmodium falciparum (isolate 3D7) | Yes | Inhibitor | Details |
ATP | Tyrosine-protein kinase ABL1 | Protein | Humans | Unknown | Inhibitor | Details |
ATP | Tyrosine-protein kinase ABL2 | Protein | Humans | Unknown | Inhibitor | Details |
Auranofin | Peroxiredoxin-5, mitochondrial | Protein | Humans | Yes | Inhibitor | Details |
Azacitidine | DNA (cytosine-5)-methyltransferase 1 | Protein | Humans | Yes | Inhibitor | Details |
Azatadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Azilsartan medoxomil | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Bacitracin | Insulin-degrading enzyme | Protein | Humans | Yes | Inhibitor | Details |
Balsalazide | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Bambuterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Basiliximab | Interleukin-2 receptor subunit alpha | Protein | Humans | Yes | Antibody | Details |
Basiliximab | Interleukin-2 receptor subunit beta | Protein | Humans | Unknown | Antibody | Details |
Bb-3497 | Peptide deformylase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Benazepril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Bendroflumethiazide | Solute carrier family 12 member 3 | Protein | Humans | Yes | Inhibitor | Details |
Benzatropine | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Benzthiazide | Carbonic anhydrase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Benzylpenicilloyl polylysine | High affinity immunoglobulin epsilon receptor subunit alpha | Protein | Humans | Yes | Agonist | Details |
Benzylpenicilloyl polylysine | High affinity immunoglobulin epsilon receptor subunit gamma | Protein | Humans | Yes | Agonist | Details |
Bepotastine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Betaxolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Betazole | Histamine H2 receptor | Protein | Humans | Yes | Agonist | Details |
Bethanidine | Beta adrenergic receptor (Protein Group) | Protein group | Humans | Unknown | Antagonist | Details |
Bevacizumab | Vascular endothelial growth factor A | Protein | Humans | Yes | Not Available | Details |
Bezafibrate | Peroxisome proliferator-activated receptor alpha | Protein | Humans | Yes | Agonist | Details |
Bicalutamide | Androgen receptor | Protein | Humans | Yes | Antagonist | Details |
Biperiden | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Bisoprolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Bivalirudin | Prothrombin | Protein | Humans | Yes | Inhibitor | Details |
Bopindolol | 5-hydroxytryptamine receptor 1A | Protein | Humans | Unknown | Not Available | Details |
Bopindolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist Partial agonist | Details |
Bopindolol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Antagonist Partial agonist | Details |
Bopindolol | Beta-3 adrenergic receptor | Protein | Humans | Unknown | Not Available | Details |
Bosentan | Endothelin B receptor | Protein | Humans | Yes | Antagonist | Details |
Bosentan | Endothelin-1 receptor | Protein | Humans | Yes | Antagonist | Details |
Botulinum toxin type B | Vesicle-associated membrane protein 1 | Protein | Humans | Yes | Binder | Details |
Botulinum toxin type B | Vesicle-associated membrane protein 2 | Protein | Humans | Yes | Binder | Details |
Brimonidine | Alpha-2A adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Bromfenac | Prostaglandin G/H synthase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Bromocriptine | Dopamine D2 receptor | Protein | Humans | Yes | Agonist | Details |
Bromodiphenhydramine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Brompheniramine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Buclizine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Budesonide | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Bumetanide | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Buprenorphine | Mu-type opioid receptor | Protein | Humans | Yes | Partial agonist | Details |
Bupropion | Sodium-dependent dopamine transporter | Protein | Humans | Yes | Inhibitor | Details |
Bupropion | Sodium-dependent noradrenaline transporter | Protein | Humans | Yes | Inhibitor | Details |
Buspirone | 5-hydroxytryptamine receptor 1A | Protein | Humans | Yes | Partial agonist | Details |
Butalbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Butenafine | Squalene monooxygenase | Protein | Humans | Yes | Inhibitor | Details |
Butobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Butorphanol | Delta-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Cabergoline | Dopamine D2 receptor | Protein | Humans | Yes | Agonist | Details |
Caffeine | Adenosine receptor A2a | Protein | Humans | Yes | Antagonist | Details |
Calcifediol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Calcipotriol | Vitamin D3 receptor | Protein | Humans | Unknown | Antagonist | Details |
Calcitriol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Camptothecin | DNA topoisomerase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Canaline | Ornithine aminotransferase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Candesartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Candesartan cilexetil | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Candoxatril | Neprilysin | Protein | Humans | Yes | Inhibitor | Details |
Capecitabine | Thymidylate synthase | Protein | Humans | Yes | Inhibitor | Details |
Capromab pendetide | Glutamate carboxypeptidase 2 | Protein | Humans | Yes | Other/unknown | Details |
Captopril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Carbamoylcholine | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Agonist | Details |
Carbenoxolone | Corticosteroid 11-beta-dehydrogenase isozyme 1 | Protein | Humans | Unknown | Inhibitor | Details |
Carbetocin | Oxytocin receptor | Protein | Humans | Yes | Agonist | Details |
Carbidopa | Aromatic-L-amino-acid decarboxylase | Protein | Humans | Yes | Inhibitor | Details |
Carbimazole | Thyroid peroxidase | Protein | Humans | Yes | Inhibitor | Details |
Carbinoxamine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Carphenazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Carprofen | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Carteolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist Partial agonist | Details |
Carteolol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Cerivastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Cerulenin | Fatty acid synthase | Protein | Humans | Yes | Inhibitor | Details |
Cetrorelix | Gonadotropin-releasing hormone receptor | Protein | Humans | Yes | Antagonist | Details |
Cetuximab | Epidermal growth factor receptor | Protein | Humans | Yes | Binder | Details |
Cevimeline | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Agonist | Details |
Chlormerodrin | Succinate-semialdehyde dehydrogenase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Chlormezanone | Translocator protein | Protein | Humans | Yes | Agonist | Details |
Chloroquine | Glutathione S-transferase A2 | Protein | Humans | Unknown | Inhibitor | Details |
Chlorothiazide | Carbonic anhydrase 2 | Protein | Humans | Yes | Inhibitor | Details |
Chlorotrianisene | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Chlorpheniramine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Chlorpromazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Chlorprothixene | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Chlorthalidone | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Cholecalciferol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Choriogonadotropin alfa | Follicle-stimulating hormone receptor | Protein | Humans | Yes | Binder | Details |
Cilastatin | Dipeptidase 1 | Protein | Humans | Yes | Inhibitor | Details |
Cilazapril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Cilazaprilat | Angiotensin-converting enzyme | Protein | Humans | Yes | Not Available | Details |
Cilostazol | cGMP-inhibited 3',5'-cyclic phosphodiesterase A | Protein | Humans | Yes | Inhibitor | Details |
Cimetidine | Histamine H2 receptor | Protein | Humans | Yes | Antagonist | Details |
Cinacalcet | Extracellular calcium-sensing receptor | Protein | Humans | Yes | Agonist | Details |
Cinalukast | Cysteinyl leukotriene receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Cinchocaine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Cinnarizine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Ciprofloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Cisapride | 5-hydroxytryptamine receptor 4 | Protein | Humans | Yes | Agonist | Details |
Clemastine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Clenbuterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Clidinium | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Clodronic acid | ADP/ATP translocase 1 | Protein | Humans | Yes | Inhibitor | Details |
Clofedanol | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Clomifene | Estrogen receptor alpha | Protein | Humans | Yes | Antagonist Agonist | Details |
Clozapine | Dopamine D1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Clozapine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Clozapine | Dopamine D4 receptor | Protein | Humans | Unknown | Antagonist | Details |
Clozapine | Histamine H1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Clozapine | Histamine H4 receptor | Protein | Humans | No | Antagonist | Details |
Clozapine | Neuron-specific vesicular protein calcyon | Protein | Humans | Unknown | Unknown | Details |
Coagulation Factor IX (Recombinant) | Coagulation factor X | Protein | Humans | Yes | Activator | Details |
Coagulation Factor IX Human | Coagulation factor X | Protein | Humans | Yes | Activator | Details |
Conivaptan | Vasopressin V1a receptor | Protein | Humans | Yes | Antagonist | Details |
Conivaptan | Vasopressin V2 receptor | Protein | Humans | Yes | Antagonist | Details |
Cyclizine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Cycloserine | D-alanine--D-alanine ligase A | Protein | Escherichia coli (strain K12) | Yes | Inhibitor | Details |
Cyclothiazide | Carbonic anhydrase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Cycrimine | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Cyproheptadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
D-Serine | Glycine receptor subunit alpha-1 | Protein | Humans | Unknown | Not Available | Details |
Daclizumab | Interleukin-2 receptor subunit alpha | Protein | Humans | Yes | Antibody | Details |
Daclizumab | Interleukin-2 receptor subunit beta | Protein | Humans | Yes | Antibody | Details |
Danazol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Dantrolene | Ryanodine receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Darbepoetin alfa | Erythropoietin receptor | Protein | Humans | Yes | Agonist | Details |
Darifenacin | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Dazoxiben | Thromboxane-A synthase | Protein | Humans | Unknown | Inhibitor | Details |
Decamethonium | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Partial agonist | Details |
Decitabine | DNA (cytosine-5)-methyltransferase 1 | Protein | Humans | Yes | Inhibitor | Details |
Demecarium | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Denileukin diftitox | Interleukin-2 receptor subunit beta | Protein | Humans | Yes | Agonist | Details |
Desipramine | Sodium-dependent noradrenaline transporter | Protein | Humans | Yes | Inhibitor | Details |
Deslanoside | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Yes | Inhibitor | Details |
Desloratadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Desmopressin | Vasopressin V2 receptor | Protein | Humans | Yes | Agonist | Details |
Desogestrel | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Desoxycorticosterone pivalate | Mineralocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Dexamethasone | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Dexamethasone | Nitric oxide synthase, inducible | Protein | Humans | Unknown | Negative modulator | Details |
Dexbrompheniramine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Dexmethylphenidate | Sodium-dependent dopamine transporter | Protein | Humans | Yes | Inhibitor | Details |
Dexrazoxane | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Dextroamphetamine | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Dextromethorphan | Sigma non-opioid intracellular receptor 1 | Protein | Humans | Yes | Agonist | Details |
Dextropropoxyphene | Kappa-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Dextropropoxyphene | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Dezocine | Kappa-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Diamorphine | Delta-type opioid receptor | Protein | Humans | Unknown | Agonist | Details |
Diclofenac | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Dicoumarol | Vitamin K epoxide reductase complex subunit 1 | Protein | Humans | Yes | Inhibitor | Details |
Dicyclomine | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Dienestrol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Diethylcarbamazine | Arachidonate 5-lipoxygenase | Protein | Humans | Yes | Inhibitor | Details |
Diethylstilbestrol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Diflunisal | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Dihomo-gamma-linolenic acid | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Dihydroergotamine | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Dihydroergotamine | 5-hydroxytryptamine receptor 2B | Protein | Humans | Unknown | Agonist | Details |
Dihydrotachysterol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Dimenhydrinate | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Dinoprost tromethamine | Prostacyclin receptor | Protein | Humans | Unknown | Antagonist | Details |
Dinoprostone | Prostaglandin E2 receptor EP2 subtype | Protein | Humans | Yes | Agonist | Details |
Diphemanil | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Diphenhydramine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Diphenoxylate | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Diphenylpyraline | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Dipivefrin | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Dipyridamole | Adenosine deaminase | Protein | Humans | Yes | Inhibitor | Details |
Dipyridamole | cAMP-specific 3',5'-cyclic phosphodiesterase 4A | Protein | Humans | Yes | Inhibitor | Details |
Dipyridamole | cGMP-specific 3',5'-cyclic phosphodiesterase | Protein | Humans | Yes | Inhibitor | Details |
Disopyramide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Dobutamine | Beta-1 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Dofetilide | Potassium voltage-gated channel subfamily H member 2 | Protein | Humans | Yes | Inhibitor | Details |
Dolasetron | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Domperidone | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Donepezil | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Dopamine | Dopamine D2 receptor | Protein | Humans | Yes | Agonist | Details |
Dorzolamide | Carbonic anhydrase 2 | Protein | Humans | Yes | Inhibitor | Details |
Doxacurium | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Doxepin | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Doxorubicin | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Doxylamine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Dronabinol | Cannabinoid receptor 1 | Protein | Humans | Yes | Agonist | Details |
Drostanolone | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Drotrecogin alfa | Coagulation factor V | Protein | Humans | Yes | Inhibitor | Details |
Drotrecogin alfa | Coagulation factor VIII | Protein | Humans | Yes | Inhibitor | Details |
Duloxetine | Sodium-dependent noradrenaline transporter | Protein | Humans | Yes | Inhibitor | Details |
Dutasteride | 3-oxo-5-alpha-steroid 4-dehydrogenase 1 | Protein | Humans | Yes | Inhibitor | Details |
Dutasteride | 3-oxo-5-alpha-steroid 4-dehydrogenase 2 | Protein | Humans | Yes | Inhibitor | Details |
Dydrogesterone | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Dyphylline | cAMP-specific 3',5'-cyclic phosphodiesterase 4A | Protein | Humans | Yes | Inhibitor | Details |
Echothiophate | Cholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Eculizumab | Complement C5 | Protein | Humans | Yes | Antibody | Details |
Edrophonium | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Efalizumab | Integrin alpha-L | Protein | Humans | Yes | Antibody | Details |
Eletriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Yes | Agonist | Details |
Eletriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Emedastine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Enalapril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Enalkiren | Renin | Protein | Humans | Unknown | Inhibitor | Details |
Encainide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Enoxacin | DNA topoisomerase 2-alpha | Protein | Humans | No | Inhibitor | Details |
Enprofylline | Adenosine receptor A2b | Protein | Humans | Yes | Antagonist | Details |
Enprofylline | cAMP-specific 3',5'-cyclic phosphodiesterase 4A | Protein | Humans | Yes | Inhibitor | Details |
Entacapone | Catechol O-methyltransferase | Protein | Humans | Yes | Inhibitor | Details |
Epinastine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Epinephrine | Beta-1 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Epinephrine | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Eplerenone | Mineralocorticoid receptor | Protein | Humans | Yes | Antagonist | Details |
Epoprostenol | Prostacyclin receptor | Protein | Humans | Yes | Agonist | Details |
Eprosartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Ergocalciferol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Ergotamine | 5-hydroxytryptamine receptor 2A | Protein | Humans | Yes | Agonist | Details |
Erlotinib | Epidermal growth factor receptor | Protein | Humans | Yes | Antagonist | Details |
Erythropoietin | Erythropoietin receptor | Protein | Humans | Yes | Agonist | Details |
Esmolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Esomeprazole | Potassium-transporting ATPase alpha chain 1 | Protein | Humans | Yes | Inhibitor | Details |
Estradiol acetate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estradiol benzoate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estradiol cypionate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estradiol dienanthate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estradiol valerate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estriol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estriol tripropionate | Estrogen receptor alpha | Protein | Humans | Yes | Not Available | Details |
Estrone | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Estrone sulfate | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Etacrynic acid | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Etanercept | Tumor necrosis factor | Protein | Humans | Yes | Inhibitor Antibody | Details |
Ethanol | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Agonist | Details |
Ethinamate | Carbonic anhydrase 2 | Protein | Humans | Yes | Inhibitor | Details |
Ethinylestradiol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Ethionamide | Enoyl-[acyl-carrier-protein] reductase [NADH] | Protein | Mycobacterium tuberculosis | Yes | Inhibitor | Details |
Ethosuximide | Voltage-dependent T-type calcium channel subunit alpha-1G | Protein | Humans | Yes | Inhibitor | Details |
Ethotoin | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Ethylmorphine | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Ethynodiol diacetate | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Etidronic acid | Receptor-type tyrosine-protein phosphatase S | Protein | Humans | Unknown | Inhibitor | Details |
Etodolac | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Etomidate | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Agonist | Details |
Etonogestrel | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Etoposide | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Etoricoxib | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Etorphine | Delta-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Etorphine | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Everolimus | Serine/threonine-protein kinase mTOR | Protein | Humans | Yes | Inhibitor | Details |
Exemestane | Cytochrome P450 19A1 | Protein | Humans | Yes | Inhibitor | Details |
Exenatide | Glucagon-like peptide 1 receptor | Protein | Humans | Yes | Agonist | Details |
Ezetimibe | Niemann-Pick C1-like protein 1 | Protein | Humans | Yes | Inhibitor | Details |
Famotidine | Histamine H2 receptor | Protein | Humans | Yes | Antagonist | Details |
Felbamate | Glutamate receptor ionotropic, NMDA 2A | Protein | Humans | Yes | Antagonist | Details |
Felbamate | Glutamate receptor ionotropic, NMDA 2B | Protein | Humans | Yes | Antagonist | Details |
Felodipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Felodipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Felodipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Felypressin | Vasopressin V1a receptor | Protein | Humans | Yes | Agonist | Details |
Fenofibrate | Peroxisome proliferator-activated receptor alpha | Protein | Humans | Yes | Agonist | Details |
Fenoldopam | Dopamine D1 receptor | Protein | Humans | Yes | Agonist | Details |
Fenoterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Fentanyl | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Fesoterodine | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Fidarestat | Aldose reductase | Protein | Humans | Unknown | Inhibitor | Details |
Flecainide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Fleroxacin | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Flunarizine | Voltage-dependent T-type calcium channel subunit alpha-1H | Protein | Humans | Yes | Inhibitor | Details |
Flunisolide | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Fluorouracil | Thymidylate synthase | Protein | Humans | Yes | Other/unknown | Details |
Fluoxetine | Sodium-dependent serotonin transporter | Protein | Humans | Yes | Inhibitor | Details |
Fluoxymesterone | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Flupentixol | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Fluphenazine | Dopamine D1 receptor | Protein | Humans | Yes | Antagonist | Details |
Fluphenazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Fluspirilene | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Flutamide | Androgen receptor | Protein | Humans | Yes | Antagonist | Details |
Fluticasone propionate | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Fluvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Folic acid | Folate receptor beta | Protein | Humans | Unknown | Binder | Details |
Folic acid | Folate receptor gamma | Protein | Humans | Unknown | Binder | Details |
Follitropin | Follicle-stimulating hormone receptor | Protein | Humans | Yes | Agonist | Details |
Forasartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Fosamprenavir | Human immunodeficiency virus type 1 protease | Protein | Human immunodeficiency virus 1 | Yes | Inhibitor | Details |
Fosinopril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Fosphenytoin | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Freselestat | Neutrophil elastase | Protein | Humans | Unknown | Inhibitor | Details |
Frovatriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Yes | Agonist | Details |
Frovatriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Fulvestrant | Estrogen receptor alpha | Protein | Humans | Yes | Antagonist | Details |
Fumagillin | Methionine aminopeptidase 2 | Protein | Humans | Unknown | Ligand | Details |
Furosemide | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Gallamine triethiodide | Muscarinic acetylcholine receptor M2 | Protein | Humans | Yes | Antagonist | Details |
Gefitinib | Epidermal growth factor receptor | Protein | Humans | Yes | Antagonist | Details |
Gemcitabine | Thymidylate synthase | Protein | Humans | Unknown | Inhibitor | Details |
Gemtuzumab ozogamicin | Myeloid cell surface antigen CD33 | Protein | Humans | Yes | Antibody Regulator | Details |
Glucagon | Glucagon receptor | Protein | Humans | Yes | Agonist | Details |
Glycine | Glutamate receptor ionotropic, NMDA 2A | Protein | Humans | Unknown | Antagonist | Details |
Glycopyrronium | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Glyphosate | 3-phosphoshikimate 1-carboxyvinyltransferase | Protein | Streptococcus pneumoniae serotype 4 (strain ATCC BAA-334 / TIGR4) | Unknown | Inhibitor | Details |
Gonadorelin | Gonadotropin-releasing hormone receptor | Protein | Humans | Yes | Agonist | Details |
Granisetron | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Guanine | GTP cyclohydrolase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Hadacidin | Adenylosuccinate synthetase | Protein | Plasmodium falciparum | Unknown | Inhibitor | Details |
Haloperidol | Dopamine D1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Haloperidol | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Haloperidol | Glutamate receptor ionotropic, NMDA 2B | Protein | Humans | Unknown | Antagonist | Details |
Heparin | Antithrombin-III | Protein | Humans | Yes | Potentiator | Details |
Hexafluronium | Cholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Hexobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Hexylcaine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Histamine | Histamine H2 receptor | Protein | Humans | Yes | Agonist | Details |
Homatropine methylbromide | Muscarinic acetylcholine receptor M5 | Protein | Humans | Yes | Antagonist | Details |
Hydralazine | Prolyl 4-hydroxylase subunit alpha-1 | Protein | Humans | Unknown | Inhibitor | Details |
Hydrochlorothiazide | Solute carrier family 12 member 3 | Protein | Humans | Yes | Inhibitor | Details |
Hydrocodone | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Hydroflumethiazide | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Hydromorphone | Delta-type opioid receptor | Protein | Humans | Yes | Partial agonist | Details |
Hydroxocobalamin | Methylmalonyl-CoA mutase, mitochondrial | Protein | Humans | Yes | Cofactor | Details |
Hydroxyfasudil | Rho-associated protein kinase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Hymenialdisine | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Not Available | Details |
Hymenialdisine | Cyclin-dependent kinase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Hymenialdisine | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Inhibitor | Details |
Hyperforin | Arachidonate 5-lipoxygenase | Protein | Humans | Unknown | Inhibitor | Details |
Hyperforin | Prostaglandin G/H synthase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Ibandronate | Farnesyl pyrophosphate synthase | Protein | Humans | Yes | Inhibitor | Details |
Ibritumomab tiuxetan | B-lymphocyte antigen CD20 | Protein | Humans | Yes | Antibody Regulator | Details |
Ibuprofen | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Ibuprofen | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Ibutilide | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Activator | Details |
Icatibant | B2 bradykinin receptor | Protein | Humans | Yes | Antagonist | Details |
Idarubicin | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Imiquimod | Toll-like receptor 7 | Protein | Humans | Yes | Agonist | Details |
Immucillin-G | Purine nucleoside phosphorylase | Protein | Humans | Unknown | Not Available | Details |
Indecainide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Indirubin-3'-monoxime | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Binder | Details |
Indirubin-3'-monoxime | Cyclin-dependent kinase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Indirubin-3'-monoxime | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Inhibitor | Details |
Infliximab | Tumor necrosis factor | Protein | Humans | Yes | Inhibitor | Details |
Insulin detemir | Insulin receptor | Protein | Humans | Yes | Agonist | Details |
Insulin glargine | Insulin receptor | Protein | Humans | Yes | Agonist | Details |
Insulin human | Insulin receptor | Protein | Humans | Yes | Agonist | Details |
Insulin lispro | Insulin receptor | Protein | Humans | Yes | Agonist | Details |
Insulin pork | Insulin receptor | Protein | Humans | Yes | Binder | Details |
Interferon alfa-2b | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Binder | Details |
Interferon alfa-2b | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Binder | Details |
Interferon alfa-n1 | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Agonist | Details |
Interferon alfa-n1 | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Agonist | Details |
Interferon alfa-n3 | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Agonist | Details |
Interferon alfa-n3 | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Agonist | Details |
Interferon alfacon-1 | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Binder | Details |
Interferon alfacon-1 | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Binder | Details |
Interferon beta-1b | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Agonist | Details |
Interferon beta-1b | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Agonist | Details |
Interferon gamma-1b | Interferon gamma receptor 1 | Protein | Humans | Yes | Binder | Details |
Interferon gamma-1b | Interferon gamma receptor 2 | Protein | Humans | Yes | Binder | Details |
Inulin | Cycloinulo-oligosaccharide fructanotransferase | Protein | Paenibacillus macerans | No | Binder | Details |
Irbesartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Irinotecan | DNA topoisomerase 1 | Protein | Humans | Yes | Inhibitor | Details |
Irinotecan | DNA topoisomerase I, mitochondrial | Protein | Humans | Yes | Inhibitor | Details |
Iron Dextran | Hemoglobin subunit alpha | Protein | Humans | Yes | Activator | Details |
Iron Dextran | Hemoglobin subunit beta | Protein | Humans | Yes | Activator | Details |
Isocarboxazid | Amine oxidase [flavin-containing] A | Protein | Humans | Yes | Inhibitor | Details |
Isoflurophate | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Isoniazid | Enoyl-[acyl-carrier-protein] reductase [NADH] | Protein | Mycobacterium tuberculosis | Yes | Adduct | Details |
Isoprenaline | Beta-1 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Isoprenaline | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist Binder | Details |
Isradipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Isradipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Itraconazole | Lanosterol 14-alpha demethylase | Protein | Humans | Yes | Inhibitor | Details |
Ketoprofen | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Labetalol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Labetalol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Lansoprazole | Potassium-transporting ATPase alpha chain 1 | Protein | Humans | Yes | Inhibitor | Details |
Lapatinib | Epidermal growth factor receptor | Protein | Humans | Yes | Antagonist | Details |
Lapatinib | Receptor tyrosine-protein kinase erbB-2 | Protein | Humans | Yes | Antagonist | Details |
Leflunomide | Dihydroorotate dehydrogenase (quinone), mitochondrial | Protein | Humans | Yes | Inhibitor | Details |
Letrozole | Cytochrome P450 19A1 | Protein | Humans | Yes | Antagonist | Details |
Levacetylmethadol | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Levobunolol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Levocabastine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Levocarnitine | Carnitine O-palmitoyltransferase 1, liver isoform | Protein | Humans | Unknown | Activator | Details |
Levomenthol | Transient receptor potential cation channel subfamily A member 1 | Protein | Humans | Yes | Inducer | Details |
Levomenthol | Transient receptor potential cation channel subfamily M member 8 | Protein | Humans | Yes | Inducer | Details |
Levosimendan | Troponin C, slow skeletal and cardiac muscles | Protein | Humans | Yes | Potentiator | Details |
Levothyroxine | Thyroid hormone receptor alpha | Protein | Humans | Yes | Agonist | Details |
Licofelone | Arachidonate 5-lipoxygenase | Protein | Humans | Unknown | Not Available | Details |
Liothyronine | Thyroid hormone receptor alpha | Protein | Humans | Yes | Agonist | Details |
Liotrix | Thyroid hormone receptor alpha | Protein | Humans | Yes | Agonist | Details |
Lisinopril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Lisuride | Dopamine D2 receptor | Protein | Humans | Yes | Agonist | Details |
Lomefloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Lonapegsomatropin | Growth hormone receptor | Protein | Humans | Yes | Ligand | Details |
Loperamide | Delta-type opioid receptor | Protein | Humans | Unknown | Agonist | Details |
Loperamide | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Lopinavir | Human immunodeficiency virus type 1 protease | Protein | Human immunodeficiency virus 1 | Yes | Inhibitor | Details |
Loratadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Losartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Loteprednol etabonate | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Lovastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Loxapine | Dopamine D1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Loxapine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Lubiprostone | Chloride channel protein 2 | Protein | Humans | Yes | Inducer | Details |
Lucanthone | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Lumiracoxib | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Lutropin alfa | Lutropin-choriogonadotropic hormone receptor | Protein | Humans | Yes | Agonist | Details |
Lypressin | Vasopressin V2 receptor | Protein | Humans | Yes | Not Available | Details |
Maraviroc | C-C chemokine receptor type 5 | Protein | Humans | Yes | Antagonist Inhibitor | Details |
Marimastat | 72 kDa type IV collagenase | Protein | Humans | Yes | Inhibitor | Details |
Marimastat | Interstitial collagenase | Protein | Humans | Yes | Inhibitor | Details |
Marimastat | Matrix metalloproteinase-9 | Protein | Humans | Yes | Inhibitor | Details |
Marimastat | Stromelysin-1 | Protein | Humans | Yes | Antagonist | Details |
Masoprocol | Arachidonate 5-lipoxygenase | Protein | Humans | Yes | Inhibitor | Details |
Mecamylamine | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Medroxyprogesterone acetate | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Medrysone | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Mefenamic acid | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Megestrol acetate | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Melatonin | Melatonin receptor type 1A | Protein | Humans | Yes | Agonist | Details |
Menotropins | Follicle-stimulating hormone receptor | Protein | Humans | Yes | Binder | Details |
Mephenytoin | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Meprobamate | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Agonist | Details |
Mequitazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Mercaptopurine | Inosine-5'-monophosphate dehydrogenase (Protein Group) | Protein group | Humans | Unknown | Inhibitor | Details |
Mesalazine | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Mesoridazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Mestranol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Metamizole | Prostaglandin G/H synthase 1 | Protein | Humans | Unknown | Not Available | Details |
Methadyl acetate | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Metharbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Methdilazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Methimazole | Thyroid peroxidase | Protein | Humans | Yes | Substrate Inhibitor | Details |
Methohexital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Antagonist | Details |
Methotrexate | Dihydrofolate reductase | Protein | Humans | Yes | Inhibitor | Details |
Methoxamine | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Agonist | Details |
Methoxyflurane | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Agonist | Details |
Methscopolamine bromide | Muscarinic acetylcholine receptor M2 | Protein | Humans | Yes | Antagonist | Details |
Methyclothiazide | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Methylergometrine | Dopamine D1 receptor | Protein | Humans | Yes | Antagonist | Details |
Methylphenidate | Sodium-dependent dopamine transporter | Protein | Humans | Yes | Inhibitor | Details |
Methylphenobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Methylprednisolone | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Methyltestosterone | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Methyprylon | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Agonist | Details |
Methysergide | 5-hydroxytryptamine receptor 2C | Protein | Humans | Yes | Antagonist | Details |
Metocurine | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Metocurine iodide | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Metolazone | Solute carrier family 12 member 3 | Protein | Humans | Yes | Inhibitor | Details |
Metoprolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Metyrapone | Cytochrome P450 11B1, mitochondrial | Protein | Humans | Yes | Inhibitor | Details |
Metyrosine | Tyrosine 3-monooxygenase | Protein | Humans | Yes | Binder | Details |
Mevastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Mexiletine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Mibefradil | Voltage-dependent T-type calcium channel subunit alpha-1G | Protein | Humans | Yes | Inhibitor | Details |
Mifepristone | Progesterone receptor | Protein | Humans | Yes | Antagonist | Details |
Miglitol | Maltase-glucoamylase, intestinal | Protein | Humans | Yes | Antagonist Inhibitor | Details |
Miglustat | Ceramide glucosyltransferase | Protein | Humans | Yes | Inhibitor | Details |
Milrinone | cGMP-inhibited 3',5'-cyclic phosphodiesterase A | Protein | Humans | Yes | Inhibitor | Details |
Minaprine | 5-hydroxytryptamine receptor 2B | Protein | Humans | Yes | Antagonist | Details |
Mipomersen | mRNA of ApoB-100 | Nucleotide | Humans | Yes | Binder | Details |
Mitoxantrone | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Mivacurium | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Moclobemide | Amine oxidase [flavin-containing] A | Protein | Humans | Yes | Antagonist Inhibitor | Details |
Moexipril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Molindone | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Mometasone | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Mometasone furoate | Glucocorticoid receptor | Protein | Humans | Yes | Not Available | Details |
Montelukast | Cysteinyl leukotriene receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Moricizine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Morphine | Delta-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Morphine | Mu-type opioid receptor | Protein | Humans | Yes | Agonist Regulator | Details |
Moxifloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Muromonab | T-cell surface glycoprotein CD3 epsilon chain | Protein | Humans | Yes | Binder | Details |
N-Acetylglucosamine | Alpha-N-acetylglucosaminidase | Protein | Humans | Unknown | Activator | Details |
Nabilone | Cannabinoid receptor 1 | Protein | Humans | Yes | Partial agonist | Details |
Nabumetone | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
NADH | NADH-ubiquinone oxidoreductase chain 1 | Protein | Humans | Unknown | Binder | Details |
NADH | NADH-ubiquinone oxidoreductase chain 2 | Protein | Humans | Unknown | Binder | Details |
NADH | NADH-ubiquinone oxidoreductase chain 3 | Protein | Humans | Unknown | Binder | Details |
Nadolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Nadolol | Beta-2 adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Nafarelin | Gonadotropin-releasing hormone receptor | Protein | Humans | Yes | Agonist | Details |
Naftifine | Squalene monooxygenase | Protein | Humans | Yes | Inhibitor | Details |
Nalbuphine | Delta-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Naloxone | Mu-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Naltrexone | Delta-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Naltrexone | Kappa-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Naltrexone | Mu-type opioid receptor | Protein | Humans | Yes | Antagonist | Details |
Nandrolone phenpropionate | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Naratriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Yes | Agonist | Details |
Naratriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Naratriptan | 5-hydroxytryptamine receptor 1F | Protein | Humans | Yes | Agonist | Details |
Natalizumab | Integrin alpha-4 | Protein | Humans | Yes | Antibody | Details |
Natalizumab | Intercellular adhesion molecule 1 | Protein | Humans | Unknown | Ligand | Details |
Nebivolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Nefazodone | 5-hydroxytryptamine receptor 2C | Protein | Humans | Yes | Antagonist | Details |
Nefazodone | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Other/unknown | Details |
Nelfinavir | HIV-1 protease | Protein | Human Immunodeficiency Virus | Yes | Inhibitor | Details |
Neostigmine | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Nesiritide | Atrial natriuretic peptide receptor 1 | Protein | Humans | Unknown | Binder | Details |
Nicardipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Nicardipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Nicardipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Nicotinamide | Poly [ADP-ribose] polymerase 1 | Protein | Humans | Unknown | Binder | Details |
Nifedipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Nifedipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Nilutamide | Androgen receptor | Protein | Humans | Yes | Antagonist | Details |
Nilvadipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Nimesulide | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Nimodipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Nimodipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Nisoldipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Nisoldipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Nisoldipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Nitisinone | 4-hydroxyphenylpyruvate dioxygenase | Protein | Humans | Yes | Inhibitor | Details |
Nitrendipine | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Protein | Humans | Yes | Inhibitor | Details |
Nitrendipine | Voltage-dependent L-type calcium channel subunit alpha-1C | Protein | Humans | Yes | Inhibitor | Details |
Nitrendipine | Voltage-dependent L-type calcium channel subunit beta-2 | Protein | Humans | Yes | Inhibitor | Details |
Nizatidine | Histamine H2 receptor | Protein | Humans | Yes | Antagonist | Details |
Norepinephrine | Beta-1 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Norfloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Norgestimate | Progesterone receptor | Protein | Humans | Yes | Agonist | Details |
Olanzapine | 5-hydroxytryptamine receptor 2A | Protein | Humans | Yes | Antagonist | Details |
Olanzapine | 5-hydroxytryptamine receptor 2C | Protein | Humans | Unknown | Antagonist | Details |
Olanzapine | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Olanzapine | Dopamine D1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Olanzapine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Olanzapine | Dopamine D3 receptor | Protein | Humans | Unknown | Antagonist | Details |
Olanzapine | Dopamine D4 receptor | Protein | Humans | Unknown | Antagonist | Details |
Olanzapine | Histamine H1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Olmesartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Olomoucine | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Binder | Details |
Olomoucine | Cyclin-dependent kinase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Olomoucine | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Inhibitor | Details |
Olopatadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Ondansetron | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Oprelvekin | Interleukin-11 receptor subunit alpha | Protein | Humans | Yes | Agonist | Details |
Orciprenaline | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Orotic acid | Dihydroorotase | Protein | Escherichia coli (strain K12) | Unknown | Inhibitor | Details |
Ouabain | Sodium/potassium-transporting ATPase subunit alpha-1 | Protein | Humans | Yes | Inhibitor | Details |
Oxandrolone | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Oxprenolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Oxycodone | Delta-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Oxymorphone | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Oxyphenonium | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Palifermin | Fibroblast growth factor receptor 2 | Protein | Humans | Yes | Agonist Binder | Details |
Paliperidone | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Palonosetron | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Pamidronic acid | Farnesyl pyrophosphate synthase | Protein | Humans | Yes | Inhibitor | Details |
Panitumumab | Epidermal growth factor receptor | Protein | Humans | Yes | Suppressor | Details |
Paricalcitol | Vitamin D3 receptor | Protein | Humans | Yes | Agonist | Details |
Pefloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Peginterferon alfa-2a | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Agonist | Details |
Peginterferon alfa-2a | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Agonist | Details |
Peginterferon alfa-2b | Interferon alpha/beta receptor 1 | Protein | Humans | Yes | Agonist | Details |
Peginterferon alfa-2b | Interferon alpha/beta receptor 2 | Protein | Humans | Yes | Agonist | Details |
Pegvisomant | Growth hormone receptor | Protein | Humans | Yes | Antagonist | Details |
Pemetrexed | Dihydrofolate reductase | Protein | Humans | Yes | Inhibitor | Details |
Pemetrexed | Thymidylate synthase | Protein | Humans | Yes | Inhibitor | Details |
Penciclovir | DNA polymerase catalytic subunit | Protein | HHV-1 | Yes | Inhibitor | Details |
Pentagastrin | Gastrin/cholecystokinin type B receptor | Protein | Humans | Yes | Agonist | Details |
Pentobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Pentostatin | Adenosine deaminase | Protein | Humans | Yes | Inhibitor | Details |
Perhexiline | Carnitine O-palmitoyltransferase 1, liver isoform | Protein | Humans | Yes | Inhibitor | Details |
Periciazine | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Perindopril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Perphenazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Phenacemide | Sodium channel protein type 1 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Phenacetin | Prostaglandin G/H synthase 1 | Protein | Humans | Unknown | Not Available | Details |
Phendimetrazine | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Agonist | Details |
Phenelzine | Amine oxidase [flavin-containing] A | Protein | Humans | Yes | Antagonist | Details |
Phenelzine | Amine oxidase [flavin-containing] B | Protein | Humans | Yes | Antagonist | Details |
Phenindamine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Phenindione | Vitamin K epoxide reductase complex subunit 1 | Protein | Humans | Yes | Inhibitor | Details |
Pheniramine | Histamine H1 receptor | Protein | Humans | Yes | Inverse agonist | Details |
Phenprocoumon | Vitamin K epoxide reductase complex subunit 1 | Protein | Humans | Yes | Inhibitor | Details |
Phenylalanine | Tyrosine 3-monooxygenase | Protein | Humans | Unknown | Binder | Details |
Phenylbutazone | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Phenylephrine | Alpha-1B adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Phosphoramidon | Neprilysin | Protein | Humans | Unknown | Inhibitor | Details |
Phylloquinone | Vitamin K-dependent gamma-carboxylase | Protein | Humans | Yes | Substrate Inducer Cofactor | Details |
Physostigmine | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Picrotoxin | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Antagonist | Details |
Pimagedine | Nitric oxide synthase, inducible | Protein | Humans | Yes | Inhibitor Downregulator | Details |
Pimozide | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Pindolol | 5-hydroxytryptamine receptor 1A | Protein | Humans | Unknown | Antagonist Inhibitor Ligand | Details |
Pindolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Partial agonist | Details |
Pindolol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Partial agonist | Details |
Pipecuronium | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Pipotiazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Pirbuterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Pirenzepine | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Piretanide | Solute carrier family 12 member 1 | Protein | Humans | Unknown | Inhibitor | Details |
Piroxicam | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Podofilox | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Polythiazide | Solute carrier family 12 member 3 | Protein | Humans | Yes | Inhibitor | Details |
Potassium chloride | Solute carrier family 12 member 1 | Protein | Humans | Unknown | Binder | Details |
Practolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Pranlukast | Cysteinyl leukotriene receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Pravastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Prednisone | Glucocorticoid receptor | Protein | Humans | Yes | Agonist | Details |
Prilocaine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Primidone | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Probenecid | Solute carrier family 22 member 6 | Protein | Humans | Yes | Inhibitor | Details |
Procainamide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Unknown | Inhibitor | Details |
Procaine | 5-hydroxytryptamine receptor 3A | Protein | Humans | Yes | Antagonist | Details |
Procaterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Prochlorperazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Profenamine | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Progabide | Gamma-aminobutyric acid type B receptor subunit 1 | Protein | Humans | Yes | Agonist | Details |
Proguanil | Dihydrofolate reductase | Protein | Humans | Yes | Inhibitor | Details |
Proline | Peptidyl-prolyl cis-trans isomerase A | Protein | Humans | Unknown | Binder | Details |
Proline | Peptidyl-prolyl cis-trans isomerase B | Protein | Humans | Unknown | Binder | Details |
Promethazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Propafenone | Potassium voltage-gated channel subfamily H member 2 | Protein | Humans | Yes | Inhibitor | Details |
Propantheline | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Propiomazine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Propranolol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Propranolol | Beta-2 adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Propranolol | Beta-3 adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Propylthiouracil | Thyroid peroxidase | Protein | Humans | Yes | Inhibitor | Details |
Purvalanol | Cyclin-dependent kinase 4 | Protein | Humans | Unknown | Not Available | Details |
Purvalanol | Mitogen-activated protein kinase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Purvalanol | Mitogen-activated protein kinase 3 | Protein | Humans | Unknown | Inhibitor | Details |
Pyridostigmine | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Pyridoxal phosphate | 4-aminobutyrate aminotransferase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Pyridoxal phosphate | Aspartate aminotransferase, cytoplasmic | Protein | Humans | Unknown | Activator | Details |
Pyrimethamine | Dihydrofolate reductase | Protein | Humans | Yes | Inhibitor | Details |
Pyruvic acid | 4-aminobutyrate aminotransferase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Quinapril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Quinestrol | Estrogen receptor alpha | Protein | Humans | Yes | Agonist Modulator | Details |
Quinidine | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Quinidine barbiturate | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Quinidine barbiturate | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Quinine | Intermediate conductance calcium-activated potassium channel protein 4 | Protein | Humans | Unknown | Inhibitor | Details |
Rabeprazole | Potassium-transporting ATPase alpha chain 1 | Protein | Humans | Yes | Inhibitor | Details |
Raloxifene | Estrogen receptor alpha | Protein | Humans | Yes | Agonist | Details |
Raloxifene | Estrogen receptor beta | Protein | Humans | Yes | Agonist | Details |
Raltitrexed | Thymidylate synthase | Protein | Humans | Yes | Inhibitor | Details |
Ramelteon | Melatonin receptor type 1A | Protein | Humans | Yes | Multitarget | Details |
Ramelteon | Melatonin receptor type 1B | Protein | Humans | Yes | Multitarget | Details |
Ramipril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Rasagiline | Amine oxidase [flavin-containing] B | Protein | Humans | Yes | Inhibitor | Details |
Rauwolfia serpentina root | Synaptic vesicular amine transporter | Protein | Humans | Yes | Inhibitor | Details |
Remifentanil | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Remikiren | Renin | Protein | Humans | Yes | Inhibitor | Details |
Remoxipride | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Rescinnamine | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Reserpine | Synaptic vesicular amine transporter | Protein | Humans | Yes | Inhibitor | Details |
Resveratrol | Casein kinase II subunit alpha | Protein | Humans | Unknown | Not Available | Details |
Resveratrol | Prostaglandin G/H synthase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Resveratrol | Prostaglandin G/H synthase 2 | Protein | Humans | Unknown | Inhibitor | Details |
Reteplase | Plasminogen | Protein | Humans | Yes | Activator | Details |
Ribavirin | Inosine-5'-monophosphate dehydrogenase 1 | Protein | Humans | Yes | Inhibitor | Details |
Ridogrel | Thromboxane A2 receptor | Protein | Humans | Yes | Antagonist | Details |
Rifaximin | DNA-directed RNA polymerase subunit beta | Protein | Escherichia coli (strain K12) | Yes | Inhibitor | Details |
Rimonabant | Cannabinoid receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Risedronic acid | Farnesyl pyrophosphate synthase | Protein | Humans | Yes | Inhibitor | Details |
Ritodrine | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Rituximab | B-lymphocyte antigen CD20 | Protein | Humans | Yes | Antibody Regulator | Details |
Rivastigmine | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Rivastigmine | Cholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Rizatriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Yes | Agonist | Details |
Rizatriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Rizatriptan | 5-hydroxytryptamine receptor 1F | Protein | Humans | Unknown | Agonist | Details |
Rocuronium | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Rofecoxib | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Ropinirole | Dopamine D4 receptor | Protein | Humans | Unknown | Agonist | Details |
Rosiglitazone | Peroxisome proliferator-activated receptor gamma | Protein | Humans | Yes | Agonist | Details |
Rosoxacin | DNA gyrase subunit B | Protein | Escherichia coli (strain K12) | Yes | Inhibitor | Details |
Rosuvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Salbutamol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Salicylic acid | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Salmeterol | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Salmon calcitonin | Calcitonin receptor | Protein | Humans | Unknown | Agonist | Details |
Salsalate | Prostaglandin G/H synthase 1 | Protein | Humans | Yes | Inhibitor | Details |
Saprisartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Sapropterin | Tyrosine 3-monooxygenase | Protein | Humans | Yes | Cofactor | Details |
Sargramostim | Granulocyte-macrophage colony-stimulating factor receptor subunit alpha | Protein | Humans | Yes | Agonist | Details |
Scopolamine | Muscarinic acetylcholine receptor M2 | Protein | Humans | Yes | Antagonist | Details |
scyllo-inositol | CDP-diacylglycerol--inositol 3-phosphatidyltransferase | Protein | Humans | Unknown | Inhibitor | Details |
Secobarbital | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Selegiline | Amine oxidase [flavin-containing] B | Protein | Humans | Yes | Inhibitor | Details |
Sermorelin | Growth hormone-releasing hormone receptor | Protein | Humans | Yes | Agonist | Details |
Sertindole | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Sibutramine | Sodium-dependent noradrenaline transporter | Protein | Humans | Yes | Inhibitor | Details |
Sildenafil | cGMP-specific 3',5'-cyclic phosphodiesterase | Protein | Humans | Yes | Inhibitor | Details |
Simvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Protein | Humans | Yes | Inhibitor | Details |
Sirolimus | Serine/threonine-protein kinase mTOR | Protein | Humans | Yes | Inhibitor | Details |
Sitagliptin | Dipeptidyl peptidase 4 | Protein | Humans | Yes | Inhibitor | Details |
Sitaxentan | Endothelin B receptor | Protein | Humans | Unknown | Antagonist | Details |
Sitaxentan | Endothelin-1 receptor | Protein | Humans | Yes | Antagonist | Details |
Sodium tetradecyl sulfate | Vitamin K-dependent protein C | Protein | Humans | Yes | Inhibitor | Details |
Solifenacin | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Somatotropin | Growth hormone receptor | Protein | Humans | Yes | Ligand | Details |
Sorafenib | Serine/threonine-protein kinase B-raf | Protein | Humans | Yes | Inhibitor | Details |
Sorbinil | Aldose reductase | Protein | Humans | Unknown | Inhibitor | Details |
Sotalol | Beta-1 adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Sparfloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Spirapril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Spironolactone | Mineralocorticoid receptor | Protein | Humans | Yes | Antagonist | Details |
Streptokinase | Plasminogen | Protein | Humans | Yes | Activator | Details |
SU9516 | Cyclin-dependent kinase 1 | Protein | Humans | Unknown | Binder | Details |
SU9516 | Cyclin-dependent kinase 2 | Protein | Humans | Unknown | Inhibitor | Details |
SU9516 | Cyclin-dependent kinase 5 | Protein | Humans | Unknown | Inhibitor | Details |
Succinic acid | Succinate-semialdehyde dehydrogenase, mitochondrial | Protein | Humans | Unknown | Inhibitor | Details |
Sufentanil | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Sulfinpyrazone | Multidrug resistance-associated protein 1 | Protein | Humans | Yes | Inhibitor | Details |
Sulindac | Aldose reductase | Protein | Humans | Unknown | Inhibitor | Details |
Sulodexide | Antithrombin-III | Protein | Humans | Yes | Potentiator | Details |
Sulpiride | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Sumatriptan | 5-hydroxytryptamine receptor 1B | Protein | Humans | Yes | Agonist | Details |
Sumatriptan | 5-hydroxytryptamine receptor 1D | Protein | Humans | Yes | Agonist | Details |
Sumatriptan | 5-hydroxytryptamine receptor 1F | Protein | Humans | Yes | Agonist | Details |
Sunitinib | Mast/stem cell growth factor receptor Kit | Protein | Humans | Yes | Inhibitor | Details |
Sunitinib | Receptor-type tyrosine-protein kinase FLT3 | Protein | Humans | Yes | Inhibitor | Details |
Sunitinib | Vascular endothelial growth factor receptor 2 | Protein | Humans | Yes | Inhibitor | Details |
Tacrine | Acetylcholinesterase | Protein | Humans | Yes | Inhibitor | Details |
Talbutal | Gamma-aminobutyric acid receptor subunit alpha-1 | Protein | Humans | Yes | Potentiator | Details |
Tamibarotene | Retinoic acid receptor alpha | Protein | Humans | Yes | Agonist | Details |
Tamoxifen | Estrogen receptor alpha | Protein | Humans | Yes | Antagonist Agonist | Details |
Tamoxifen | Estrogen receptor beta | Protein | Humans | Yes | Antagonist Agonist | Details |
Tamsulosin | Alpha-1A adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Tamsulosin | Alpha-1B adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Tamsulosin | Alpha-1D adrenergic receptor | Protein | Humans | Unknown | Antagonist | Details |
Tasosartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Tazarotene | Retinoic acid receptor gamma | Protein | Humans | Yes | Agonist | Details |
Tegaserod | 5-hydroxytryptamine receptor 4 | Protein | Humans | Yes | Antagonist Partial agonist | Details |
Telmisartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Temsirolimus | Serine/threonine-protein kinase mTOR | Protein | Humans | Yes | Inhibitor | Details |
Tenecteplase | Plasminogen | Protein | Humans | Yes | Activator | Details |
Teniposide | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Tenoxicam | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Terazosin | Alpha-1A adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Terazosin | Alpha-1B adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Terazosin | Alpha-1D adrenergic receptor | Protein | Humans | Yes | Antagonist | Details |
Terbinafine | Squalene monooxygenase | Protein | Humans | No | Inhibitor | Details |
Terbutaline | Beta-2 adrenergic receptor | Protein | Humans | Yes | Agonist | Details |
Terfenadine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Terfenadine | Potassium voltage-gated channel subfamily H member 2 | Protein | Humans | Unknown | Inhibitor | Details |
Teriparatide | Parathyroid hormone/parathyroid hormone-related peptide receptor | Protein | Humans | Unknown | Ligand | Details |
Terlipressin | Vasopressin V1a receptor | Protein | Humans | Yes | Agonist | Details |
Testolactone | Cytochrome P450 19A1 | Protein | Humans | Yes | Inhibitor | Details |
Testosterone | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Testosterone cypionate | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Testosterone enanthate | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Testosterone undecanoate | Androgen receptor | Protein | Humans | Yes | Agonist | Details |
Tetrabenazine | Synaptic vesicular amine transporter | Protein | Humans | Yes | Inhibitor | Details |
Tetracosactide | Adrenocorticotropic hormone receptor | Protein | Humans | Yes | Agonist | Details |
Tetracycline | Major prion protein | Protein | Humans | Unknown | Inhibitor | Details |
Theophylline | Adenosine receptor A2b | Protein | Humans | Yes | Antagonist | Details |
Theophylline | cGMP-specific 3',5'-cyclic phosphodiesterase | Protein | Humans | Yes | Inhibitor | Details |
Thiabendazole | Fumarate reductase flavoprotein subunit | Protein | Escherichia coli (strain K12) | Yes | Inhibitor | Details |
Thiopental | Fatty-acid amide hydrolase 1 | Protein | Humans | Unknown | Inhibitor | Details |
Thioproperazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Thiorphan | Neprilysin | Protein | Humans | Unknown | Inhibitor | Details |
Thiothixene | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Thyrotropin alfa | Thyrotropin receptor | Protein | Humans | Yes | Agonist | Details |
Tiagabine | Sodium- and chloride-dependent GABA transporter 1 | Protein | Humans | Yes | Inhibitor | Details |
Tiaprofenic acid | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Ticlopidine | P2Y purinoceptor 12 | Protein | Humans | Yes | Antagonist | Details |
Tiotropium | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Tipranavir | Human immunodeficiency virus type 1 protease | Protein | Human immunodeficiency virus 1 | Yes | Inhibitor | Details |
Tirofiban | Integrin beta-3 | Protein | Humans | Yes | Antagonist | Details |
Tocainide | Sodium channel protein type 5 subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Tolcapone | Catechol O-methyltransferase | Protein | Humans | Yes | Inhibitor | Details |
Tolmetin | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Tolrestat | Aldose reductase | Protein | Humans | Unknown | Inhibitor | Details |
Tolterodine | Muscarinic acetylcholine receptor M3 | Protein | Humans | Yes | Antagonist | Details |
Topotecan | DNA topoisomerase 1 | Protein | Humans | Yes | Inhibitor | Details |
Torasemide | Solute carrier family 12 member 1 | Protein | Humans | Yes | Inhibitor | Details |
Torasemide | Solute carrier family 12 member 2 | Protein | Humans | Yes | Inhibitor | Details |
Toremifene | Estrogen receptor alpha | Protein | Humans | Yes | Modulator | Details |
Tositumomab | B-lymphocyte antigen CD20 | Protein | Humans | Yes | Antibody | Details |
Tramadol | Mu-type opioid receptor | Protein | Humans | Yes | Agonist | Details |
Tramadol | Sodium-dependent noradrenaline transporter | Protein | Humans | Yes | Inhibitor | Details |
Trandolapril | Angiotensin-converting enzyme | Protein | Humans | Yes | Inhibitor | Details |
Tranylcypromine | Amine oxidase [flavin-containing] A | Protein | Humans | Yes | Inhibitor | Details |
Tranylcypromine | Amine oxidase [flavin-containing] B | Protein | Humans | Yes | Inhibitor | Details |
Trastuzumab | Receptor tyrosine-protein kinase erbB-2 | Protein | Humans | Yes | Binder Antibody | Details |
Trastuzumab emtansine | Receptor tyrosine-protein kinase erbB-2 | Protein | Humans | Yes | Antibody | Details |
Treprostinil | Prostacyclin receptor | Protein | Humans | Yes | Agonist | Details |
Tretinoin | Retinoic acid receptor gamma | Protein | Humans | Yes | Agonist | Details |
Triamterene | Amiloride-sensitive sodium channel subunit alpha | Protein | Humans | Yes | Inhibitor | Details |
Trichlormethiazide | Solute carrier family 12 member 3 | Protein | Humans | Yes | Inhibitor | Details |
Trifluoperazine | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |
Trifluoperazine | Neuron-specific vesicular protein calcyon | Protein | Humans | Yes | Antagonist | Details |
Triflupromazine | 5-hydroxytryptamine receptor 2B | Protein | Humans | Yes | Antagonist | Details |
Trifluridine | Thymidylate synthase | Protein | Humans | Yes | Inhibitor | Details |
Trihexyphenidyl | Muscarinic acetylcholine receptor M1 | Protein | Humans | Yes | Antagonist | Details |
Trimethadione | Voltage-dependent T-type calcium channel subunit alpha-1G | Protein | Humans | Yes | Inhibitor | Details |
Trimipramine | 5-hydroxytryptamine receptor 2C | Protein | Humans | Unknown | Antagonist | Details |
Tripelennamine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Triprolidine | Histamine H1 receptor | Protein | Humans | Yes | Antagonist | Details |
Troglitazone | Peroxisome proliferator-activated receptor gamma | Protein | Humans | Yes | Agonist Regulator | Details |
Tropicamide | Muscarinic acetylcholine receptor M4 | Protein | Humans | Yes | Antagonist | Details |
Trovafloxacin | DNA topoisomerase 2-alpha | Protein | Humans | Unknown | Inhibitor | Details |
Tubocurarine | Neuronal acetylcholine receptor subunit alpha-2 | Protein | Humans | Yes | Antagonist | Details |
Tyrosine | Tyrosine 3-monooxygenase | Protein | Humans | Unknown | Binder | Details |
Udenafil | cGMP-specific 3',5'-cyclic phosphodiesterase | Protein | Humans | Yes | Inhibitor | Details |
Urofollitropin | Follicle-stimulating hormone receptor | Protein | Humans | Yes | Agonist | Details |
Urokinase | Plasminogen | Protein | Humans | Yes | Activator | Details |
Valdecoxib | Prostaglandin G/H synthase 2 | Protein | Humans | Yes | Inhibitor | Details |
Valrubicin | DNA topoisomerase 2-alpha | Protein | Humans | Yes | Inhibitor | Details |
Valsartan | Type-1 angiotensin II receptor | Protein | Humans | Yes | Antagonist | Details |
Vapreotide | Neurokinin 1 receptor | Protein | Humans | Unknown | Antagonist | Details |
Varenicline | Neuronal acetylcholine receptor subunit alpha-4 | Protein | Humans | Yes | Partial agonist | Details |
Vasopressin | Vasopressin V2 receptor | Protein | Humans | Yes | Agonist Regulator | Details |
Voglibose | Maltase-glucoamylase, intestinal | Protein | Humans | Yes | Inhibitor | Details |
Vorinostat | Histone deacetylase 1 | Protein | Humans | Yes | Inhibitor | Details |
Warfarin | Vitamin K epoxide reductase complex subunit 1 | Protein | Humans | Yes | Inhibitor | Details |
Ximelagatran | Prothrombin | Protein | Humans | Yes | Inhibitor | Details |
Zafirlukast | Cysteinyl leukotriene receptor 1 | Protein | Humans | Yes | Antagonist | Details |
Zanamivir | Neuraminidase | Protein | Influenza A virus (strain A/Bangkok/1/1979 H3N2) | Yes | Inhibitor | Details |
Zileuton | Arachidonate 5-lipoxygenase | Protein | Humans | Yes | Inhibitor | Details |
Zoledronic acid | Farnesyl pyrophosphate synthase | Protein | Humans | Yes | Inhibitor | Details |
Zuclopenthixol | Dopamine D2 receptor | Protein | Humans | Yes | Antagonist | Details |