| DB00353 | Methylergometrine | approved | yes | antagonist | Details |
| DB00508 | Triflupromazine | approved, vet_approved | yes | antagonist | Details |
| DB00589 | Lisuride | approved, investigational | unknown | antagonist | Details |
| DB00805 | Minaprine | approved | unknown | agonist | Details |
| DB00850 | Perphenazine | approved | yes | antagonist | Details |
| DB00988 | Dopamine | approved | yes | agonist | Details |
| DB01235 | Levodopa | approved | yes | agonist | Details |
| DB01239 | Chlorprothixene | approved, experimental, investigational, withdrawn | yes | antagonist | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | antagonist | Details |
| DB00679 | Thioridazine | approved, withdrawn | yes | antagonist | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | agonist | Details |
| DB00800 | Fenoldopam | approved | yes | agonist | Details |
| DB00875 | Flupentixol | approved, investigational, withdrawn | yes | antagonist | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01624 | Zuclopenthixol | approved, investigational | yes | antagonist | Details |
| DB00363 | Clozapine | approved | unknown | antagonist | Details |
| DB00623 | Fluphenazine | approved | yes | antagonist | Details |
| DB00502 | Haloperidol | approved | unknown | antagonist | Details |
| DB00408 | Loxapine | approved | unknown | antagonist | Details |
| DB01038 | Carphenazine | withdrawn | yes | antagonist | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | agonist | Details |
| DB00248 | Cabergoline | approved | unknown | agonist | Details |
| DB05271 | Rotigotine | approved | unknown | agonist | Details |
| DB01267 | Paliperidone | approved | unknown | antagonist | Details |
| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | antagonistpartial agonistligand | Details |
| DB01224 | Quetiapine | approved | unknown | antagonist | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | antagonist | Details |
| DB01608 | Periciazine | approved, investigational | yes | antagonist | Details |
| DB00397 | Phenylpropanolamine | approved, vet_approved, withdrawn | unknown | partial agonist | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | yes | antagonist | Details |
| DB01614 | Acepromazine | experimental, vet_approved | yes | antagonist | Details |
| DB01621 | Pipotiazine | approved, investigational | yes | antagonist | Details |
| DB01622 | Thioproperazine | experimental | unknown | antagonist | Details |
| DB01623 | Thiothixene | approved | yes | antagonist | Details |
| DB04946 | Iloperidone | approved | unknown | antagonist | Details |
| DB12890 | Dihydrexidine | investigational | unknown | | Details |
| DB12093 | Tetrahydropalmatine | investigational | unknown | antagonist | Details |
| DB09286 | Pipamperone | investigational | unknown | antagonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | | Details |
| DB06077 | Lumateperone | approved, investigational | unknown | | Details |
| DB00734 | Risperidone | approved, investigational | unknown | antagonist | Details |