| DB00154 | Dihomo-gamma-linolenic acid | investigational, nutraceutical | yes | | Details |
| DB00159 | Icosapent | approved, nutraceutical | yes | inhibitor | Details |
| DB00480 | Lenalidomide | approved | unknown | negative modulator | Details |
| DB00482 | Celecoxib | approved, investigational | yes | inhibitor | Details |
| DB00533 | Rofecoxib | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB00580 | Valdecoxib | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB00605 | Sulindac | approved, investigational | yes | inhibitor | Details |
| DB00712 | Flurbiprofen | approved, investigational | yes | inhibitor | Details |
| DB00784 | Mefenamic acid | approved | yes | inhibitor | Details |
| DB00812 | Phenylbutazone | approved, vet_approved | yes | inhibitor | Details |
| DB00821 | Carprofen | approved, vet_approved, withdrawn | yes | inhibitor | Details |
| DB00991 | Oxaprozin | approved | yes | inhibitor | Details |
| DB00244 | Mesalazine | approved | yes | inhibitor | Details |
| DB00316 | Acetaminophen | approved | yes | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | yes | inhibitor | Details |
| DB00461 | Nabumetone | approved | yes | inhibitor | Details |
| DB00465 | Ketorolac | approved | yes | inhibitor | Details |
| DB00469 | Tenoxicam | approved | yes | inhibitor | Details |
| DB00500 | Tolmetin | approved | yes | inhibitor | Details |
| DB00573 | Fenoprofen | approved | yes | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | yes | inhibitor | Details |
| DB00749 | Etodolac | approved, investigational, vet_approved | yes | inhibitor | Details |
| DB00788 | Naproxen | approved, vet_approved | yes | inhibitor | Details |
| DB00814 | Meloxicam | approved, vet_approved | yes | inhibitor | Details |
| DB00861 | Diflunisal | approved, investigational | yes | inhibitor | Details |
| DB00870 | Suprofen | approved, withdrawn | yes | inhibitor | Details |
| DB00939 | Meclofenamic acid | approved, vet_approved | yes | inhibitor | Details |
| DB00945 | Acetylsalicylic acid | approved, vet_approved | yes | inhibitor | Details |
| DB00963 | Bromfenac | approved, withdrawn | yes | inhibitor | Details |
| DB01009 | Ketoprofen | approved, vet_approved | yes | inhibitor | Details |
| DB01014 | Balsalazide | approved, investigational | yes | inhibitor | Details |
| DB01050 | Ibuprofen | approved | yes | inhibitor | Details |
| DB01283 | Lumiracoxib | approved, investigational | yes | inhibitor | Details |
| DB01399 | Salsalate | approved | yes | inhibitor | Details |
| DB00936 | Salicylic acid | approved, investigational, vet_approved | yes | inhibitor | Details |
| DB01404 | Ginseng | investigational, nutraceutical | unknown | inhibitor | Details |
| DB01628 | Etoricoxib | approved, investigational | yes | inhibitor | Details |
| DB01600 | Tiaprofenic acid | approved | yes | inhibitor | Details |
| DB04743 | Nimesulide | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB02709 | Resveratrol | investigational | unknown | inhibitor | Details |
| DB04725 | Licofelone | investigational | unknown | | Details |
| DB05095 | Cimicoxib | investigational | unknown | | Details |
| DB02266 | Flufenamic acid | approved | unknown | | Details |
| DB00554 | Piroxicam | approved, investigational | yes | inhibitor | Details |
| DB01397 | Magnesium salicylate | experimental | yes | inhibitor | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrate | Details |
| DB06725 | Lornoxicam | approved, investigational | yes | inhibitor | Details |
| DB03866 | Prostaglandin G2 | experimental | unknown | | Details |
| DB03477 | 1-Phenylsulfonamide-3-Trifluoromethyl-5-Parabromophenylpyrazole | experimental | unknown | | Details |
| DB06802 | Nepafenac | approved, investigational | unknown | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | yes | inhibitor | Details |
| DB04552 | Niflumic acid | experimental | yes | inhibitor | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | inhibitor | Details |
| DB01419 | Antrafenine | approved | unknown | inhibitor | Details |
| DB01401 | Choline magnesium trisalicylate | approved | unknown | inhibitor | Details |
| DB00233 | Aminosalicylic acid | approved | unknown | inhibitor | Details |
| DB00963 | Bromfenac | approved, withdrawn | unknown | inhibitor | Details |
| DB00887 | Bumetanide | approved | unknown | inducer | Details |
| DB06774 | Capsaicin | approved | unknown | inhibitor | Details |
| DB00856 | Chlorphenesin | approved, experimental | unknown | inhibitor | Details |
| DB05095 | Cimicoxib | investigational | unknown | inhibitor | Details |
| DB00720 | Clodronic acid | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB06195 | Seliciclib | investigational | unknown | inhibitor | Details |
| DB00035 | Desmopressin | approved | unknown | inducer | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | inducer | Details |
| DB01395 | Drospirenone | approved | unknown | inhibitorinducer | Details |
| DB06804 | Nonoxynol-9 | approved, withdrawn | unknown | inducer | Details |
| DB00515 | Cisplatin | approved | unknown | inhibitor | Details |
| DB00884 | Risedronic acid | approved, investigational | unknown | inducer | Details |
| DB00360 | Sapropterin | approved, investigational | unknown | inducer | Details |
| DB06436 | Semaxanib | investigational | unknown | inducer | Details |
| DB05875 | Sar9, Met (O2)11-Substance P | investigational | unknown | inducer | Details |
| DB00041 | Aldesleukin | approved | unknown | inducer | Details |
| DB00620 | Triamcinolone | approved, vet_approved | unknown | inhibitor | Details |
| DB08819 | Tafluprost | approved | unknown | inducer | Details |
| DB08910 | Pomalidomide | approved | yes | inhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB08439 | Parecoxib | approved | yes | inhibitor | Details |
| DB09217 | Firocoxib | experimental, vet_approved | unknown | | Details |
| DB13167 | Alclofenac | approved, withdrawn | yes | antagonist | Details |
| DB09213 | Dexibuprofen | approved, investigational | yes | inhibitor | Details |
| DB11133 | Omega-3 fatty acids | approved, nutraceutical | unknown | substrate | Details |
| DB13168 | Omega-6 fatty acids | nutraceutical | unknown | substrate | Details |
| DB06736 | Aceclofenac | approved, investigational | yes | inhibitor | Details |
| DB13783 | Acemetacin | approved, investigational | yes | antagonist | Details |
| DB09215 | Droxicam | withdrawn | yes | inhibitor | Details |
| DB09212 | Loxoprofen | approved | yes | antagonist | Details |
| DB09216 | Tolfenamic acid | approved, investigational | yes | antagonist | Details |
| DB09214 | Dexketoprofen | approved, investigational | unknown | antagonist | Details |
| DB09214 | Dexketoprofen | approved, investigational | unknown | inhibitor | Details |
| DB09295 | Talniflumate | experimental | unknown | antagonist | Details |
| DB09295 | Talniflumate | experimental | unknown | inhibitor | Details |
| DB09285 | Morniflumate | experimental | unknown | | Details |
| DB09285 | Morniflumate | experimental | unknown | inhibitor | Details |
| DB09288 | Propacetamol | experimental | yes | antagonist | Details |
| DB11079 | Trolamine salicylate | approved | yes | inhibitor | Details |
| DB11071 | Phenyl salicylate | approved | unknown | antagonist | Details |
| DB13346 | Bufexamac | approved, withdrawn | yes | inhibitor | Details |
| DB11327 | Dipyrithione | approved | unknown | | Details |
| DB13961 | Fish oil | approved, nutraceutical | yes | inhibitor | Details |
| DB11323 | Glycol salicylate | approved | yes | antagonist | Details |
| DB11201 | Menthyl salicylate | approved | yes | antagonist | Details |
| DB13501 | Bendazac | approved, withdrawn | unknown | | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB11752 | Bryostatin 1 | investigational | unknown | inducer | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | inhibitor | Details |
| DB14060 | NS-398 | experimental | unknown | inhibitor | Details |