| DB00070 | Hyaluronidase (ovine) | approved, investigational | unknown | inhibitor | Details |
| DB00137 | Lutein | approved, investigational, nutraceutical | unknown | | Details |
| DB00459 | Acitretin | approved | unknown | | Details |
| DB00576 | Sulfamethizole | approved, investigational, vet_approved | unknown | | Details |
| DB00743 | Gadobenic acid | approved, investigational | no | binder | Details |
| DB00815 | Sodium lauryl sulfate | experimental | unknown | binder | Details |
| DB00936 | Salicylic acid | approved, investigational, vet_approved | no | other/unknown | Details |
| DB00946 | Phenprocoumon | approved, investigational | no | binderregulator | Details |
| DB00995 | Auranofin | approved, investigational | unknown | | Details |
| DB01120 | Gliclazide | approved | unknown | | Details |
| DB01328 | Cefonicid | approved, investigational | no | other/unknown | Details |
| DB01329 | Cefoperazone | approved, investigational | no | other/unknown | Details |
| DB01396 | Digitoxin | approved, investigational | no | | Details |
| DB03017 | Lauric acid | approved, experimental | unknown | | Details |
| DB03193 | Stearic acid | approved, experimental | unknown | | Details |
| DB03600 | Capric acid | experimental | no | | Details |
| DB03796 | Palmitic Acid | approved | unknown | | Details |
| DB04224 | Oleic Acid | approved, investigational, vet_approved | unknown | | Details |
| DB04557 | Arachidonic Acid | experimental | no | | Details |
| DB04711 | Iodipamide | approved | unknown | binder | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | | Details |
| DB01197 | Captopril | approved | no | other/unknown | Details |
| DB01050 | Ibuprofen | approved | no | binder | Details |
| DB00563 | Methotrexate | approved | no | binder | Details |
| DB00451 | Levothyroxine | approved | no | | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | | Details |
| DB00605 | Sulindac | approved, investigational | unknown | | Details |
| DB00749 | Etodolac | approved, investigational, vet_approved | unknown | | Details |
| DB00861 | Diflunisal | approved, investigational | unknown | | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | no | | Details |
| DB00655 | Estrone | approved | no | | Details |
| DB00624 | Testosterone | approved, investigational | no | binder | Details |
| DB01307 | Insulin detemir | approved | no | binder | Details |
| DB01418 | Acenocoumarol | approved, investigational | no | | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | no | | Details |
| DB00228 | Enflurane | approved, investigational, vet_approved | unknown | binder | Details |
| DB00753 | Isoflurane | approved, vet_approved | unknown | | Details |
| DB01189 | Desflurane | approved | unknown | binder | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | | Details |
| DB01236 | Sevoflurane | approved, vet_approved | unknown | binder | Details |
| DB00252 | Phenytoin | approved, vet_approved | unknown | | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | | Details |
| DB00540 | Nortriptyline | approved | no | binder | Details |
| DB00321 | Amitriptyline | approved | no | binder | Details |
| DB00903 | Etacrynic acid | approved, investigational | unknown | | Details |
| DB00695 | Furosemide | approved, vet_approved | no | binder | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | no | | Details |
| DB00682 | Warfarin | approved | no | binderregulator | Details |
| DB00554 | Piroxicam | approved, investigational | unknown | | Details |
| DB00573 | Fenoprofen | approved | unknown | | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | | Details |
| DB03585 | Oxyphenbutazone | approved, withdrawn | unknown | | Details |
| DB00544 | Fluorouracil | approved | no | | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | | Details |
| DB01032 | Probenecid | approved, investigational | no | | Details |
| DB01044 | Gatifloxacin | approved, investigational, withdrawn | unknown | other/unknown | Details |
| DB01068 | Clonazepam | approved, illicit | no | | Details |
| DB01147 | Cloxacillin | approved, investigational, vet_approved | no | binder | Details |
| DB01327 | Cefazolin | approved | unknown | other/unknown | Details |
| DB00931 | Metacycline | approved, investigational | no | | Details |
| DB01015 | Sulfamethoxazole | approved | no | substrate | Details |
| DB00415 | Ampicillin | approved, vet_approved | no | other/unknown | Details |
| DB00567 | Cephalexin | approved, investigational, vet_approved | no | binder | Details |
| DB00759 | Tetracycline | approved, vet_approved, withdrawn | no | | Details |
| DB01212 | Ceftriaxone | approved | no | other/unknown | Details |
| DB01330 | Cefotetan | approved | no | | Details |
| DB00274 | Cefmetazole | approved, investigational | no | | Details |
| DB00495 | Zidovudine | approved | no | | Details |
| DB01397 | Magnesium salicylate | experimental | no | | Details |
| DB00788 | Naproxen | approved, vet_approved | no | | Details |
| DB00334 | Olanzapine | approved, investigational | no | binder | Details |
| DB01056 | Tocainide | approved | no | other/unknown | Details |
| DB01320 | Fosphenytoin | approved, investigational | no | other/unknown | Details |
| DB00712 | Flurbiprofen | approved, investigational | no | other/unknown | Details |
| DB07402 | Azapropazone | withdrawn | unknown | | Details |
| DB07517 | 3-CARBOXY-4-METHYL-5-PROPYL-2-FURANPROPIONIC | experimental | unknown | | Details |
| DB07992 | Indoxyl sulfate | experimental | unknown | | Details |
| DB08231 | Myristic acid | experimental | unknown | | Details |
| DB08496 | (R)-warfarin | experimental | unknown | | Details |
| DB08735 | R,S-Warfarin alcohol | experimental | unknown | | Details |
| DB08736 | S,R-Warfarin alcohol | experimental | unknown | | Details |
| DB00430 | Cefpiramide | approved | unknown | | Details |
| DB01583 | Liotrix | approved | unknown | | Details |
| DB01294 | Bismuth subsalicylate | approved, vet_approved | no | binder | Details |
| DB00456 | Cefalotin | approved, investigational, vet_approved | unknown | binder | Details |
| DB01581 | Sulfamerazine | approved, vet_approved | unknown | | Details |
| DB01582 | Sulfamethazine | approved, investigational, vet_approved | unknown | | Details |
| DB01587 | Ketazolam | approved | unknown | | Details |
| DB01614 | Acepromazine | experimental, vet_approved | unknown | | Details |
| DB01621 | Pipotiazine | approved, investigational | unknown | | Details |
| DB04574 | Estrone sulfate | approved | unknown | | Details |
| DB06710 | Methyltestosterone | approved | unknown | | Details |
| DB01622 | Thioproperazine | experimental | unknown | | Details |
| DB01623 | Thiothixene | approved | unknown | | Details |
| DB06705 | Gadofosveset trisodium | approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | binder | Details |
| DB01016 | Glyburide | approved | unknown | binder | Details |
| DB00912 | Repaglinide | approved, investigational | unknown | | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | | Details |
| DB08867 | Ulipristal | approved | no | substrate | Details |
| DB05294 | Vandetanib | approved | unknown | binder | Details |
| DB05521 | Telaprevir | approved, withdrawn | no | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | binder | Details |
| DB08881 | Vemurafenib | approved | unknown | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | binder | Details |
| DB08893 | Mirabegron | approved | no | binder | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | substrate | Details |
| DB08899 | Enzalutamide | approved | no | binder | Details |
| DB08820 | Ivacaftor | approved | no | carrier | Details |
| DB00776 | Oxcarbazepine | approved | unknown | substrate | Details |
| DB06201 | Rufinamide | approved | unknown | substrate | Details |
| DB06716 | Fospropofol | approved, illicit, investigational | unknown | substrate | Details |
| DB04855 | Dronedarone | approved | no | binder | Details |
| DB06209 | Prasugrel | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | binder | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrate | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | binder | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00678 | Losartan | approved | unknown | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrate | Details |
| DB00864 | Tacrolimus | approved, investigational | unknown | substrate | Details |
| DB00717 | Norethisterone | approved | unknown | substrate | Details |
| DB08931 | Riociguat | approved | unknown | substrate | Details |
| DB08895 | Tofacitinib | approved, investigational | unknown | | Details |
| DB08932 | Macitentan | approved | no | binder | Details |
| DB06290 | Simeprevir | approved | no | binder | Details |
| DB00493 | Cefotaxime | approved | unknown | | Details |
| DB09280 | Lumacaftor | approved | no | carrier | Details |
| DB09130 | Copper | approved, investigational | no | binder | Details |
| DB11093 | Calcium citrate | approved, investigational | no | substrate | Details |
| DB11348 | Calcium Phosphate | approved | no | substrate | Details |
| DB11575 | Grazoprevir | approved | no | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | binder | Details |
| DB09093 | Chlortetracycline | approved, investigational, vet_approved | no | | Details |
| DB06796 | Mangafodipir | approved, investigational, withdrawn | unknown | binder | Details |
| DB09262 | Imidafenacin | investigational | no | substrate | Details |
| DB00276 | Amsacrine | approved, investigational | unknown | | Details |
| DB11359 | Guaiacol | approved | unknown | | Details |
| DB03255 | Phenol | approved, experimental | unknown | | Details |
| DB06728 | Aniline | experimental | unknown | | Details |
| DB06713 | Norelgestromin | approved, investigational | unknown | | Details |
| DB01370 | Aluminium | approved, investigational | unknown | | Details |
| DB13014 | Hypericin | investigational | unknown | | Details |
| DB01057 | Echothiophate | approved | unknown | | Details |
| DB11397 | Dichlorvos | vet_approved | unknown | | Details |
| DB00677 | Isoflurophate | approved, investigational, withdrawn | unknown | | Details |
| DB00943 | Zalcitabine | approved, investigational | unknown | | Details |
| DB01072 | Atazanavir | approved, investigational | no | binder | Details |
| DB00649 | Stavudine | approved, investigational | unknown | | Details |
| DB00900 | Didanosine | approved | unknown | | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | | Details |
| DB00879 | Emtricitabine | approved, investigational | unknown | binder | Details |
| DB00220 | Nelfinavir | approved | no | binder | Details |
| DB00238 | Nevirapine | approved | unknown | | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrate | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | | Details |
| DB04816 | Dantron | approved, investigational, withdrawn | unknown | | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | binder | Details |
| DB00515 | Cisplatin | approved | unknown | | Details |
| DB00162 | Vitamin A | approved, nutraceutical, vet_approved | unknown | binder | Details |
| DB04690 | Camptothecin | experimental | unknown | | Details |
| DB02709 | Resveratrol | investigational | unknown | | Details |
| DB00744 | Zileuton | approved, investigational, withdrawn | unknown | | Details |
| DB04539 | Glyphosate | experimental | unknown | | Details |
| DB11590 | Thimerosal | approved | unknown | | Details |
| DB05134 | Tanespimycin | investigational | unknown | | Details |
| DB01124 | Tolbutamide | approved, investigational | unknown | | Details |
| DB01276 | Exenatide | approved, investigational | unknown | | Details |
| DB00414 | Acetohexamide | approved, investigational, withdrawn | unknown | | Details |
| DB00458 | Imipramine | approved | unknown | | Details |
| DB00159 | Icosapent | approved, nutraceutical | no | binder | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | | Details |
| DB01104 | Sertraline | approved | unknown | binder | Details |
| DB09383 | Meprednisone | approved, investigational | unknown | | Details |
| DB00266 | Dicoumarol | approved | unknown | | Details |
| DB04828 | Zomepirac | withdrawn | unknown | | Details |
| DB00500 | Tolmetin | approved | unknown | | Details |
| DB11217 | Arbutin | approved | unknown | | Details |
| DB09526 | Hydroquinone | approved, investigational | unknown | | Details |
| DB00784 | Mefenamic acid | approved | unknown | | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | | Details |
| DB01169 | Arsenic trioxide | approved, investigational | no | substrate | Details |
| DB11828 | Neratinib | approved, investigational | no | substrate | Details |
| DB00607 | Nafcillin | approved, investigational | unknown | | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | substrate | Details |
| DB00512 | Vancomycin | approved | no | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | binder | Details |
| DB08864 | Rilpivirine | approved | no | binder | Details |
| DB13928 | Semaglutide | approved, investigational | no | substrate | Details |
| DB09087 | Potassium alum | approved | unknown | binder | Details |
| DB09223 | Blonanserin | investigational | no | substrate | Details |
| DB09236 | Lacidipine | approved, investigational | unknown | binder | Details |
| DB09124 | Medrogestone | approved, withdrawn | no | binder | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | binder | Details |
| DB09139 | Technetium Tc-99m oxidronate | approved | no | binder | Details |
| DB13943 | Testosterone cypionate | approved | no | other/unknown | Details |
| DB13944 | Testosterone enanthate | approved | no | other/unknown | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | no | binder | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | no | | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | no | | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | no | | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | no | | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | no | | Details |
| DB11638 | Artenimol | approved, experimental, investigational | unknown | ligand | Details |
| DB01420 | Testosterone propionate | approved, investigational, vet_approved, withdrawn | no | substrate | Details |
| DB09195 | Lorpiprazole | approved | no | substrate | Details |
| DB09204 | Arotinolol | investigational | no | substrate | Details |
| DB08814 | Triflusal | approved, investigational | no | substrate | Details |
| DB09229 | Aranidipine | experimental | no | binder | Details |
| DB09333 | Iopodic acid | approved, investigational, withdrawn | no | substrate | Details |
| DB09347 | Acetrizoic acid | withdrawn | no | binder | Details |
| DB09348 | Propiolactone | approved, withdrawn | no | binder | Details |
| DB11130 | Opium | approved, illicit | no | binder | Details |
| DB06778 | Cupric sulfate | approved | unknown | | Details |
| DB09053 | Ibrutinib | approved | no | substrate | Details |
| DB11182 | Rose bengal | approved, investigational | unknown | binder | Details |
| DB13967 | Patent Blue | approved | yes | binder | Details |
| DB13909 | Bismuth subgallate | approved | unknown | carrier | Details |
| DB09418 | Potassium perchlorate | approved, investigational | unknown | binder | Details |
| DB11641 | Vinflunine | approved, investigational | no | substrate | Details |
| DB13421 | Edoxudine | approved, investigational, withdrawn | no | binder | Details |
| DB11134 | Cupric oxide | approved | unknown | binder | Details |
| DB11148 | Butamben | approved, withdrawn | no | substrate | Details |
| DB11637 | Delamanid | approved, investigational | unknown | substrate | Details |
| DB13751 | Glycyrrhizic acid | approved, experimental | no | binder | Details |
| DB12965 | Silver | approved, investigational | unknown | binder | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | binder | Details |
| DB14481 | Calcium phosphate dihydrate | approved | no | | Details |
| DB14517 | Aluminium phosphate | approved, investigational | unknown | | Details |
| DB14518 | Aluminum acetate | approved, investigational | unknown | | Details |
| DB00432 | Trifluridine | approved, investigational | unknown | binder | Details |
| DB14582 | Patisiran | approved, investigational | unknown | ligand | Details |
| DB09213 | Dexibuprofen | approved, investigational | no | | Details |
| DB12455 | Omadacycline | approved, investigational | unknown | | Details |
| DB12836 | Grapiprant | investigational, vet_approved | no | substrate | Details |
| DB11753 | Rifamycin | approved, investigational | no | substrate | Details |
| DB11963 | Dacomitinib | approved, investigational | no | binder | Details |
| DB11855 | Revefenacin | approved, investigational | no | binder | Details |
| DB12141 | Gilteritinib | approved, investigational | no | binder | Details |
| DB06480 | Prucalopride | approved | unknown | binder | Details |
| DB11978 | Glasdegib | approved, investigational | no | binder | Details |
| DB00214 | Torasemide | approved | unknown | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | no | substrate | Details |
| DB09564 | Insulin degludec | approved | no | binder | Details |
| DB00245 | Benzatropine | approved | no | binder | Details |
| DB00264 | Metoprolol | approved, investigational | no | binder | Details |
| DB00286 | Conjugated estrogens | approved | no | binder | Details |
| DB00289 | Atomoxetine | approved | no | binder | Details |
| DB00294 | Etonogestrel | approved, investigational | no | binder | Details |
| DB00295 | Morphine | approved, investigational | no | binder | Details |
| DB00310 | Chlorthalidone | approved | no | | Details |
| DB00304 | Desogestrel | approved | no | binder | Details |
| DB00327 | Hydromorphone | approved, illicit | no | binder | Details |
| DB09073 | Palbociclib | approved, investigational | no | binder | Details |
| DB00332 | Ipratropium | approved, experimental | no | binder | Details |
| DB01142 | Doxepin | approved, investigational | no | binder | Details |
| DB01076 | Atorvastatin | approved | no | binder | Details |
| DB06655 | Liraglutide | approved | unknown | binder | Details |
| DB01235 | Levodopa | approved | unknown | binder | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | binder | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | binder | Details |
| DB00421 | Spironolactone | approved | unknown | binder | Details |
| DB00335 | Atenolol | approved | no | substrate | Details |
| DB01126 | Dutasteride | approved, investigational | no | binder | Details |
| DB09299 | Tenofovir alafenamide | approved | no | binder | Details |
| DB00343 | Diltiazem | approved, investigational | no | binder | Details |
| DB14126 | Tenofovir | experimental, investigational | no | binder | Details |
| DB00476 | Duloxetine | approved | unknown | ligand | Details |
| DB00497 | Oxycodone | approved, illicit, investigational | unknown | binder | Details |
| DB00481 | Raloxifene | approved, investigational | no | binder | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | binder | Details |
| DB00461 | Nabumetone | approved | unknown | | Details |
| DB00982 | Isotretinoin | approved | unknown | binder | Details |
| DB00584 | Enalapril | approved, vet_approved | no | binder | Details |
| DB01067 | Glipizide | approved, investigational | no | binder | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | binder | Details |
| DB00737 | Meclizine | approved | no | binder | Details |
| DB00768 | Olopatadine | approved | no | binder | Details |
| DB00571 | Propranolol | approved, investigational | unknown | | Details |
| DB00575 | Clonidine | approved | unknown | binder | Details |
| DB00787 | Acyclovir | approved | unknown | binder | Details |
| DB00490 | Buspirone | approved, investigational | unknown | binder | Details |
| DB01029 | Irbesartan | approved, investigational | unknown | binder | Details |
| DB06282 | Levocetirizine | approved | unknown | binder | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | ligand | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | binder | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | binder | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | binder | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | binder | Details |
| DB01045 | Rifampicin | approved | unknown | ligand | Details |
| DB01394 | Colchicine | approved | unknown | binder | Details |
| DB00333 | Methadone | approved | no | | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | binder | Details |
| DB00620 | Triamcinolone | approved, vet_approved | unknown | binder | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | substrate | Details |
| DB00881 | Quinapril | approved, investigational | unknown | binder | Details |
| DB09079 | Nintedanib | approved | unknown | substrate | Details |
| DB00999 | Hydrochlorothiazide | approved, vet_approved | unknown | binder | Details |
| DB01241 | Gemfibrozil | approved | unknown | binder | Details |
| DB01039 | Fenofibrate | approved | unknown | binder | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | binder | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | binder | Details |
| DB01275 | Hydralazine | approved | unknown | binder | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | binder | Details |
| DB00687 | Fludrocortisone | approved, investigational | unknown | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | binder | Details |
| DB00278 | Argatroban | approved, investigational | unknown | binder | Details |
| DB06216 | Asenapine | approved | unknown | binder | Details |
| DB15444 | Elexacaftor | approved, investigational | unknown | substrate | Details |
| DB00860 | Prednisolone | approved, vet_approved | unknown | binder | Details |
| DB15566 | Prednisolone acetate | approved, vet_approved | unknown | binder | Details |
| DB11703 | Acalabrutinib | approved, investigational | unknown | binder | Details |
| DB14513 | Magnesium | approved, experimental, investigational | unknown | | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | binder | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB00273 | Topiramate | approved | unknown | binder | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | binder | Details |
| DB01222 | Budesonide | approved | unknown | binder | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | binder | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | binder | Details |
| DB09237 | Levamlodipine | approved, investigational | unknown | binder | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | binder | Details |
| DB14879 | Cefiderocol | approved, investigational | no | ligand | Details |
| DB00852 | Pseudoephedrine | approved | unknown | binder | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB00993 | Azathioprine | approved | unknown | binder | Details |
| DB00557 | Hydroxyzine | approved | unknown | substrateregulator | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | binder | Details |
| DB01069 | Promethazine | approved, investigational | unknown | binder | Details |
| DB01115 | Nifedipine | approved | unknown | binder | Details |
| DB01132 | Pioglitazone | approved, investigational | unknown | substrate | Details |
| DB00814 | Meloxicam | approved, vet_approved | unknown | | Details |
| DB00938 | Salmeterol | approved | unknown | binder | Details |
| DB00878 | Chlorhexidine | approved, vet_approved, withdrawn | unknown | substrate | Details |
| DB01006 | Letrozole | approved, investigational | unknown | binder | Details |
| DB00246 | Ziprasidone | approved | unknown | | Details |
| DB01060 | Amoxicillin | approved, vet_approved | unknown | binder | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | substrate | Details |
| DB09100 | Thyroid, porcine | approved | unknown | binder | Details |
| DB01013 | Clobetasol propionate | approved | unknown | binder | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | binder | Details |
| DB00977 | Ethinylestradiol | approved | unknown | binder | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | substrate | Details |
| DB01264 | Darunavir | approved | unknown | substrate | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | binder | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | carrier | Details |
| DB01601 | Lopinavir | approved | unknown | substrate | Details |
| DB14999 | Human interferon beta | approved, investigational | unknown | binder | Details |
| DB00126 | Ascorbic acid | approved, nutraceutical | unknown | binder | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | | Details |
| DB05382 | Iodine | approved, investigational | unknown | binder | Details |
| DB11642 | Pitolisant | approved, investigational | no | binder | Details |
| DB00152 | Thiamine | approved, investigational, nutraceutical, vet_approved | unknown | binder | Details |
| DB00165 | Pyridoxine | approved, investigational, nutraceutical, vet_approved | unknown | binder | Details |
| DB00595 | Oxytetracycline | approved, investigational, vet_approved | unknown | binder | Details |
| DB00870 | Suprofen | approved, withdrawn | unknown | binder | Details |
| DB00774 | Hydroflumethiazide | approved, investigational, withdrawn | unknown | binder | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | binder | Details |
| DB15534 | Colchiceine | approved, experimental | unknown | substrate | Details |
| DB01053 | Benzylpenicillin | approved, vet_approved | unknown | binder | Details |
| DB01324 | Polythiazide | approved | unknown | binder | Details |
| DB07565 | Chloramphenicol succinate | approved | unknown | binder | Details |
| DB01914 | D-glucose | approved, investigational, vet_approved | unknown | binder | Details |
| DB14533 | Zinc chloride | approved, investigational | unknown | binder | Details |
| DB11689 | Selumetinib | approved, investigational | unknown | carrier | Details |
| DB04911 | Oritavancin | approved, investigational | unknown | binder | Details |
| DB14548 | Zinc sulfate, unspecified form | approved, experimental | unknown | binder | Details |
| DB00734 | Risperidone | approved, investigational | unknown | binder | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | binder | Details |
| DB01364 | Ephedrine | approved | unknown | binder | Details |
| DB00237 | Butabarbital | approved, illicit | unknown | binder | Details |
| DB01133 | Tiludronic acid | approved, investigational, vet_approved | unknown | binder | Details |
| DB14840 | Ripretinib | approved | unknown | binder | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | binder | Details |
| DB00842 | Oxazepam | approved | unknown | binder | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | binder | Details |
| DB09274 | Artesunate | approved, investigational | unknown | binder | Details |
| DB15690 | Fluoroestradiol F-18 | approved | unknown | binder | Details |
| DB00808 | Indapamide | approved | unknown | binder | Details |
| DB08816 | Ticagrelor | approved | unknown | binder | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | binder | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | binder | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | binder | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | binder | Details |
| DB00104 | Octreotide | approved, investigational | unknown | binder | Details |
| DB11677 | Triheptanoin | approved, investigational | unknown | binder | Details |
| DB12404 | Remimazolam | approved, investigational | unknown | binder | Details |
| DB11796 | Fostemsavir | approved, investigational | unknown | carrier | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | binder | Details |
| DB11820 | Nifurtimox | approved, investigational | unknown | binder | Details |
| DB00847 | Cysteamine | approved, investigational | unknown | binder | Details |
| DB15093 | Somapacitan | approved, investigational | unknown | binder | Details |
| DB00908 | Quinidine | approved, investigational | unknown | binder | Details |
| DB15935 | Lumasiran | approved, investigational | no | binder | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | binder | Details |
| DB11853 | Relugolix | approved, investigational | unknown | binder | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | binder | Details |
| DB15248 | Bulevirtide | approved, investigational | unknown | binder | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrate | Details |
| DB15456 | Vericiguat | approved, investigational | unknown | binder | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | binder | Details |
| DB15133 | Tepotinib | approved, investigational | unknown | binder | Details |
| DB06151 | Acetylcysteine | approved, investigational | unknown | binder | Details |
| DB00346 | Alfuzosin | approved, investigational | unknown | binder | Details |
| DB00376 | Trihexyphenidyl | approved | unknown | binder | Details |
| DB00391 | Sulpiride | approved, investigational | no | binder | Details |
| DB01083 | Orlistat | approved, investigational | unknown | binder | Details |
| DB08877 | Ruxolitinib | approved | unknown | binder | Details |
| DB00640 | Adenosine | approved, investigational | unknown | binder | Details |
| DB00853 | Temozolomide | approved, investigational | no | binder | Details |
| DB06237 | Avanafil | approved | unknown | binder | Details |
| DB04854 | Febuxostat | approved | unknown | binder | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | binder | Details |
| DB11800 | Tivozanib | approved, investigational | unknown | binder | Details |
| DB00080 | Daptomycin | approved, investigational | no | binder | Details |
| DB00434 | Cyproheptadine | approved | unknown | binder | Details |
| DB00083 | Botulinum toxin type A | approved, investigational | unknown | binder | Details |
| DB00968 | Methyldopa | approved | no | binder | Details |
| DB08995 | Diosmin | approved, investigational | unknown | binder | Details |
| DB08822 | Azilsartan medoxomil | approved, investigational | no | binder | Details |
| DB00438 | Ceftazidime | approved | no | binder | Details |
| DB09069 | Trimetazidine | approved, investigational | unknown | binder | Details |
| DB00601 | Linezolid | approved, investigational | no | binder | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | binder | Details |
| DB12235 | Estetrol | approved, investigational | unknown | binder | Details |
| DB01064 | Isoprenaline | approved, investigational | unknown | binder | Details |
| DB12471 | Ibrexafungerp | approved, investigational | unknown | binder | Details |
| DB06695 | Dabigatran etexilate | approved | unknown | binder | Details |
| DB16165 | Finerenone | approved, investigational | unknown | binder | Details |
| DB16703 | Belumosudil | approved, investigational | no | binder | Details |
| DB00877 | Sirolimus | approved, investigational | no | binder | Details |
| DB06234 | Maribavir | approved, investigational | no | binder | Details |
| DB14973 | Abrocitinib | approved, investigational | no | binder | Details |
| DB15575 | Padeliporfin | approved, experimental | unknown | binder | Details |
| DB09070 | Tibolone | approved, investigational | unknown | binder | Details |
| DB04847 | Roxadustat | approved, investigational | unknown | binder | Details |
| DB09074 | Olaparib | approved | unknown | binder | Details |
| DB15171 | Tirzepatide | approved, investigational | unknown | binder | Details |
| DB13959 | Medium-chain triglycerides | approved | unknown | binder | Details |
| DB06813 | Pralatrexate | approved, investigational | no | binder | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | binderregulator | Details |
| DB13514 | Pranoprofen | experimental, investigational | no | regulator | Details |
| DB00427 | Triprolidine | approved | unknown | binderregulator | Details |
| DB00485 | Dicloxacillin | approved, investigational, vet_approved | unknown | binderregulator | Details |
| DB01173 | Orphenadrine | approved | unknown | binderregulator | Details |
| DB01619 | Phenindamine | approved | unknown | binderregulator | Details |
| DB00792 | Tripelennamine | approved, vet_approved | unknown | binderregulator | Details |
| DB08912 | Dabrafenib | approved, investigational | no | binder | Details |
| DB16699 | Vutrisiran | approved, investigational | unknown | ligand | Details |
| DB06150 | Sulfadimethoxine | approved, vet_approved, withdrawn | unknown | substrate | Details |
| DB00254 | Doxycycline | approved, investigational, vet_approved | unknown | substratebinder | Details |
| DB08936 | Chlorcyclizine | approved | unknown | regulator | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | regulator | Details |
| DB01176 | Cyclizine | approved | unknown | regulator | Details |
| DB00366 | Doxylamine | approved, vet_approved | unknown | regulator | Details |
| DB00850 | Perphenazine | approved | unknown | regulator | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | binder | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | binder | Details |
| DB13310 | Ormeloxifene | experimental | unknown | binder | Details |
| DB00758 | Clopidogrel | approved | no | binder | Details |
| DB15149 | Futibatinib | approved, investigational | no | binder | Details |
| DB08930 | Dolutegravir | approved | no | binder | Details |
| DB17083 | Linzagolix | approved | no | binder | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | binder | Details |
| DB11793 | Niraparib | approved, investigational | unknown | binder | Details |
| DB00642 | Pemetrexed | approved, investigational | no | binder | Details |
| DB12243 | Edaravone | approved, investigational | no | binder | Details |
| DB00795 | Sulfasalazine | approved | no | binder | Details |
| DB00303 | Ertapenem | approved, investigational | no | binder | Details |
| DB01119 | Diazoxide | approved | unknown | binder | Details |
| DB01101 | Capecitabine | approved, investigational | no | binder | Details |
| DB00363 | Clozapine | approved | no | binder | Details |
| DB00349 | Clobazam | approved, illicit | no | binder | Details |
| DB00770 | Alprostadil | approved, investigational | unknown | binder | Details |
| DB00683 | Midazolam | approved, illicit | no | binder | Details |
| DB11901 | Apalutamide | approved, investigational | no | binder | Details |
| DB09128 | Brexpiprazole | approved, investigational | no | substrate | Details |
| DB08906 | Fluticasone furoate | approved | no | binder | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | binder | Details |
| DB09076 | Umeclidinium | approved | no | binder | Details |
| DB01005 | Hydroxyurea | approved | no | binder | Details |
| DB00526 | Oxaliplatin | approved, investigational | no | binder | Details |
| DB06772 | Cabazitaxel | approved | unknown | binder | Details |
| DB12874 | Quizartinib | approved, investigational | no | binder | Details |
| DB01042 | Melphalan | approved | unknown | binder | Details |
| DB08903 | Bedaquiline | approved | no | binder | Details |
| DB11718 | Encorafenib | approved, investigational | no | binder | Details |
| DB11967 | Binimetinib | approved, investigational | no | binder | Details |
| DB12005 | Nirogacestat | approved, investigational | no | binder | Details |
| DB16200 | Iptacopan | approved, investigational | no | binder | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | binder | Details |
| DB13874 | Enasidenib | approved, investigational | no | binder | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | no | binder | Details |