| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB00268 | Ropinirole | approved, investigational | yes | agonist | Details |
| DB00413 | Pramipexole | approved, investigational | yes | agonist | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | antagonist | Details |
| DB01239 | Chlorprothixene | approved, experimental, investigational, withdrawn | yes | antagonist | Details |
| DB00714 | Apomorphine | approved, investigational | yes | agonist | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | antagonist | Details |
| DB12061 | Pardoprunox | investigational | unknown | | Details |
| DB05766 | Norclozapine | investigational | unknown | | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB06477 | Sumanirole | investigational | unknown | | Details |
| DB06288 | Amisulpride | approved, investigational | yes | antagonist | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | yes | agonist | Details |
| DB00589 | Lisuride | approved, investigational | yes | agonist | Details |
| DB00248 | Cabergoline | approved | unknown | agonist | Details |
| DB05271 | Rotigotine | approved | yes | agonist | Details |
| DB00502 | Haloperidol | approved | unknown | inverse agonist | Details |
| DB01267 | Paliperidone | approved | yes | antagonist | Details |
| DB00363 | Clozapine | approved | unknown | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | antagonistpartial agonist | Details |
| DB01224 | Quetiapine | approved | unknown | ligand | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | antagonist | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | unknown | antagonist | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | antagonist | Details |
| DB00988 | Dopamine | approved | yes | agonist | Details |
| DB01235 | Levodopa | approved | yes | agonist | Details |
| DB01100 | Pimozide | approved | yes | antagonist | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | yes | antagonist | Details |
| DB04946 | Iloperidone | approved | unknown | antagonist | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB06148 | Mianserin | approved, investigational | unknown | binder | Details |
| DB09014 | Captodiame | experimental | yes | agonist | Details |
| DB09207 | AS-8112 | experimental | unknown | antagonist | Details |
| DB13025 | Tiapride | investigational | yes | blocker | Details |
| DB12478 | Piribedil | investigational | unknown | | Details |
| DB06454 | Sarizotan | investigational | unknown | ligand | Details |
| DB09223 | Blonanserin | investigational | yes | antagonist | Details |
| DB09286 | Pipamperone | investigational | unknown | | Details |
| DB11274 | Dihydro-alpha-ergocryptine | approved | yes | partial agonist | Details |
| DB09289 | Tianeptine | investigational | unknown | agonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | | Details |
| DB00490 | Buspirone | approved, investigational | unknown | antagonist | Details |
| DB00875 | Flupentixol | approved, investigational, withdrawn | unknown | antagonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | agonist | Details |
| DB06016 | Cariprazine | approved, investigational | unknown | partial agonist | Details |
| DB09128 | Brexpiprazole | approved, investigational | unknown | partial agonist | Details |