| DB00858 | Drostanolone | illicit | unknown | | Details |
| DB01185 | Fluoxymesterone | approved, illicit | unknown | antagonist | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | binder | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | binder | Details |
| DB01406 | Danazol | approved | no | antagonist | Details |
| DB02901 | Stanolone | illicit, investigational | unknown | | Details |
| DB03882 | 5-Alpha-Androstane-3-Beta,17beta-Diol | experimental | unknown | | Details |
| DB03926 | 5alpha-androstane-3beta,17alpha-diol | experimental | unknown | | Details |
| DB00648 | Mitotane | approved | unknown | upregulator | Details |
| DB02342 | 2-Methoxyestradiol | investigational | unknown | | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | | Details |
| DB00624 | Testosterone | approved, investigational | no | binder | Details |
| DB04574 | Estrone sulfate | approved | unknown | | Details |
| DB06710 | Methyltestosterone | approved | unknown | | Details |
| DB00717 | Norethisterone | approved | unknown | substrate | Details |
| DB00367 | Levonorgestrel | approved, investigational | unknown | inhibitorbinder | Details |
| DB01593 | Zinc | approved, investigational | unknown | | Details |
| DB04429 | 4'-Hydroxyflavanone | experimental | unknown | | Details |
| DB04468 | Afimoxifene | investigational | unknown | | Details |
| DB00882 | Clomifene | approved, investigational | unknown | | Details |
| DB00890 | Dienestrol | approved, investigational | unknown | | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | | Details |
| DB11221 | Dioxybenzone | approved | unknown | binder | Details |
| DB11674 | Equol | investigational | unknown | | Details |
| DB04573 | Estriol | approved, investigational, vet_approved | unknown | | Details |
| DB00655 | Estrone | approved | unknown | | Details |
| DB01645 | Genistein | investigational | unknown | | Details |
| DB01094 | Hesperetin | experimental | unknown | | Details |
| DB00179 | Masoprocol | approved, investigational | unknown | | Details |
| DB03467 | Naringenin | experimental | unknown | | Details |
| DB09371 | Norethynodrel | approved | unknown | | Details |
| DB04824 | Phenolphthalein | approved, withdrawn | unknown | | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | binderpotentiator | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | | Details |
| DB00675 | Tamoxifen | approved | yes | inducer | Details |
| DB00539 | Toremifene | approved, investigational | unknown | | Details |
| DB11478 | Zeranol | experimental, vet_approved | unknown | | Details |
| DB09124 | Medrogestone | approved, withdrawn | no | binder | Details |
| DB13943 | Testosterone cypionate | approved | no | other/unknown | Details |
| DB13944 | Testosterone enanthate | approved | no | other/unknown | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | no | binder | Details |
| DB13951 | Stanolone acetate | experimental | unknown | | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | | Details |
| DB01420 | Testosterone propionate | approved, investigational, vet_approved, withdrawn | no | substrate | Details |
| DB11619 | Gestrinone | approved | unknown | antagonist | Details |
| DB14487 | Zinc acetate | approved, investigational | unknown | | Details |
| DB14533 | Zinc chloride | approved, investigational | unknown | modulator | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | | Details |
| DB14641 | Estriol tripropionate | experimental | unknown | | Details |
| DB00286 | Conjugated estrogens | approved | no | binder | Details |
| DB00294 | Etonogestrel | approved, investigational | no | binder | Details |
| DB00304 | Desogestrel | approved | no | binder | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | ligand | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | binder | Details |
| DB00977 | Ethinylestradiol | approved | unknown | binder | Details |
| DB14548 | Zinc sulfate, unspecified form | approved, experimental | unknown | modulator | Details |
| DB15690 | Fluoroestradiol F-18 | approved | unknown | binder | Details |
| DB00080 | Daptomycin | approved, investigational | no | binder | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | binder | Details |