| DB00521 | Carteolol | approved | yes | antagonist | Details |
| DB00816 | Orciprenaline | approved | yes | agonist | Details |
| DB00867 | Ritodrine | approved, investigational | yes | agonist | Details |
| DB00871 | Terbutaline | approved | yes | agonist | Details |
| DB00901 | Bitolterol | withdrawn | yes | | Details |
| DB00938 | Salmeterol | approved | yes | agonist | Details |
| DB00983 | Formoterol | approved, investigational | yes | agonist | Details |
| DB01001 | Salbutamol | approved, vet_approved | yes | agonist | Details |
| DB00373 | Timolol | approved | yes | antagonist | Details |
| DB00571 | Propranolol | approved, investigational | unknown | antagonist | Details |
| DB00598 | Labetalol | approved | yes | antagonist | Details |
| DB00612 | Bisoprolol | approved | no | antagonist | Details |
| DB00668 | Epinephrine | approved, vet_approved | yes | agonist | Details |
| DB00852 | Pseudoephedrine | approved | unknown | partial agonist | Details |
| DB00866 | Alprenolol | experimental, withdrawn | yes | antagonist | Details |
| DB00960 | Pindolol | approved, investigational | yes | partial agonist | Details |
| DB01064 | Isoprenaline | approved, investigational | yes | agonistbinder | Details |
| DB01151 | Desipramine | approved, investigational | unknown | antagonist | Details |
| DB01203 | Nadolol | approved | unknown | antagonist | Details |
| DB01210 | Levobunolol | approved | yes | antagonist | Details |
| DB01214 | Metipranolol | approved | yes | antagonist | Details |
| DB01274 | Arformoterol | approved, investigational | yes | agonist | Details |
| DB01366 | Procaterol | approved, investigational | yes | agonist | Details |
| DB01407 | Clenbuterol | approved, investigational, vet_approved | yes | agonist | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | antagonist | Details |
| DB01288 | Fenoterol | approved, investigational | yes | agonist | Details |
| DB01291 | Pirbuterol | approved | yes | agonist | Details |
| DB01580 | Oxprenolol | approved | unknown | antagonist | Details |
| DB01359 | Penbutolol | approved, investigational | yes | antagonistpartial agonist | Details |
| DB00368 | Norepinephrine | approved | yes | agonist | Details |
| DB01408 | Bambuterol | investigational | yes | agonist | Details |
| DB05039 | Indacaterol | approved | yes | agonist | Details |
| DB05849 | NCX 950 | investigational | unknown | | Details |
| DB06262 | Droxidopa | approved, investigational | yes | agonist | Details |
| DB00264 | Metoprolol | approved, investigational | no | antagonist | Details |
| DB00195 | Betaxolol | approved, investigational | unknown | antagonist | Details |
| DB00489 | Sotalol | approved | yes | antagonist | Details |
| DB01295 | Bevantolol | experimental | unknown | antagonist | Details |
| DB01193 | Acebutolol | approved, investigational | unknown | partial agonist | Details |
| DB01102 | Arbutamine | approved | unknown | agonist | Details |
| DB00841 | Dobutamine | approved | unknown | agonist | Details |
| DB07543 | (S)-carazolol | experimental | unknown | | Details |
| DB00449 | Dipivefrin | approved | yes | agonist | Details |
| DB08807 | Bopindolol | experimental | yes | antagonistpartial agonist | Details |
| DB08808 | Bupranolol | experimental | unknown | antagonist | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | antagonist | Details |
| DB00925 | Phenoxybenzamine | approved | unknown | | Details |
| DB01363 | Ephedra sinica root | nutraceutical | yes | agonist | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB00248 | Cabergoline | approved | unknown | binder | Details |
| DB00221 | Isoetharine | approved | unknown | agonist | Details |
| DB00335 | Atenolol | approved | unknown | antagonist | Details |
| DB00397 | Phenylpropanolamine | approved, vet_approved, withdrawn | unknown | agonist | Details |
| DB09080 | Olodaterol | approved | yes | agonist | Details |
| DB09082 | Vilanterol | approved | yes | agonist | Details |
| DB04846 | Celiprolol | approved, investigational | yes | agonist | Details |
| DB13139 | Levosalbutamol | approved, investigational | yes | agonist | Details |
| DB09013 | Befunolol | experimental | unknown | | Details |
| DB12248 | Tulobuterol | investigational | unknown | regulator | Details |
| DB01917 | Putrescine | experimental | unknown | | Details |
| DB03566 | Spermidine | experimental | unknown | | Details |
| DB00127 | Spermine | experimental, nutraceutical | unknown | | Details |
| DB01182 | Propafenone | approved | unknown | antagonist | Details |
| DB09204 | Arotinolol | investigational | yes | antagonist | Details |
| DB09273 | Doxofylline | experimental | yes | agonist | Details |
| DB06814 | Protokylol | approved, vet_approved | yes | agonist | Details |
| DB11124 | Racepinephrine | approved | yes | agonist | Details |
| DB11587 | Etafedrine | approved | yes | agonist | Details |
| DB05590 | Bedoradrine | investigational | yes | agonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | ligand | Details |
| DB01364 | Ephedrine | approved | yes | agonist | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | unknown | antagonist | Details |
| DB13624 | Methoxyphenamine | approved | unknown | regulator | Details |