| DB00171 | ATP | investigational, nutraceutical | unknown | | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB03619 | Deoxycholic acid | approved | unknown | inducer | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrateinducer | Details |
| DB02659 | Cholic Acid | approved | unknown | substrateinhibitorinducer | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB00977 | Ethinylestradiol | approved | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitor | Details |
| DB02123 | Glycochenodeoxycholic Acid | experimental | unknown | substrateinhibitor | Details |
| DB01016 | Glyburide | approved | unknown | substrateinhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00206 | Reserpine | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00570 | Vinblastine | approved | no | substrateinhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01229 | Paclitaxel | approved, vet_approved | no | substrateinhibitor | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | inhibitor | Details |
| DB00559 | Bosentan | approved, investigational | unknown | inhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrate | Details |
| DB00693 | Fluorescein | approved | unknown | substrate | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrate | Details |
| DB00390 | Digoxin | approved | unknown | substrate | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrate | Details |
| DB06290 | Simeprevir | approved | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | unknown | inhibitor | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB00966 | Telmisartan | approved, investigational | no | substrate | Details |
| DB09374 | Indocyanine green acid form | approved, investigational | no | substrate | Details |
| DB01149 | Nefazodone | approved, withdrawn | no | substrate | Details |
| DB01232 | Saquinavir | approved, investigational | no | substrate | Details |
| DB01601 | Lopinavir | approved | no | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | no | inhibitor | Details |
| DB00834 | Mifepristone | approved, investigational | no | substrate | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrate | Details |
| DB13345 | Dihydroergocristine | approved, experimental | no | substrate | Details |
| DB12319 | Benzbromarone | investigational, withdrawn | no | substrate | Details |
| DB00622 | Nicardipine | approved, investigational | no | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | no | substrate | Details |
| DB01023 | Felodipine | approved, investigational | no | substrate | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | no | substrate | Details |
| DB00678 | Losartan | approved | no | substrate | Details |
| DB00222 | Glimepiride | approved | no | substrate | Details |
| DB00822 | Disulfiram | approved | no | substrate | Details |
| DB00641 | Simvastatin | approved | no | substrate | Details |
| DB00421 | Spironolactone | approved | no | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | no | substrate | Details |
| DB00270 | Isradipine | approved, investigational | no | substrate | Details |
| DB00973 | Ezetimibe | approved | no | substrate | Details |
| DB00975 | Dipyridamole | approved | no | substrate | Details |
| DB08860 | Pitavastatin | approved | no | substrate | Details |
| DB01039 | Fenofibrate | approved | no | substrate | Details |
| DB01072 | Atazanavir | approved, investigational | no | substrate | Details |
| DB00912 | Repaglinide | approved, investigational | no | substrate | Details |
| DB01138 | Sulfinpyrazone | approved | no | substrate | Details |
| DB00243 | Ranolazine | approved, investigational | no | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | no | substrate | Details |
| DB00220 | Nelfinavir | approved | no | substrate | Details |
| DB01222 | Budesonide | approved | no | substrate | Details |
| DB00224 | Indinavir | approved | no | substrate | Details |
| DB00482 | Celecoxib | approved, investigational | no | inhibitor | Details |
| DB00833 | Cefaclor | approved | no | substrate | Details |
| DB05804 | Prasterone sulfate | investigational | no | substrate | Details |
| DB00637 | Astemizole | approved, withdrawn | no | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | no | substrateinhibitor | Details |
| DB00911 | Tinidazole | approved, investigational | no | substrate | Details |
| DB12712 | Pilsicainide | investigational | no | substrate | Details |
| DB00698 | Nitrofurantoin | approved, vet_approved | no | substrate | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB00328 | Indomethacin | approved, investigational | no | substrate | Details |
| DB00176 | Fluvoxamine | approved, investigational | no | substrate | Details |
| DB01165 | Ofloxacin | approved | no | substrate | Details |
| DB01067 | Glipizide | approved, investigational | no | substrate | Details |
| DB00275 | Olmesartan | approved, investigational | no | inhibitor | Details |
| DB00335 | Atenolol | approved | no | substrate | Details |
| DB00625 | Efavirenz | approved, investigational | no | substrate | Details |
| DB00342 | Terfenadine | approved, withdrawn | no | substrate | Details |
| DB01211 | Clarithromycin | approved | no | substrate | Details |
| DB13751 | Glycyrrhizic acid | approved, experimental | no | substrate | Details |
| DB00572 | Atropine | approved, vet_approved | no | substrate | Details |
| DB00301 | Flucloxacillin | approved, investigational | no | substrate | Details |
| DB01054 | Nitrendipine | approved, investigational | no | substrate | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | no | substrateinhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | no | substrate | Details |
| DB01115 | Nifedipine | approved | no | inhibitor | Details |
| DB01015 | Sulfamethoxazole | approved | no | inhibitor | Details |
| DB00788 | Naproxen | approved, vet_approved | no | substrate | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | no | inhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00908 | Quinidine | approved, investigational | no | inhibitor | Details |
| DB00675 | Tamoxifen | approved | no | inhibitor | Details |
| DB14057 | Valinomycin | experimental | no | inhibitor | Details |
| DB05990 | Obeticholic acid | approved | unknown | inhibitorinducer | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | inhibitor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitor | Details |
| DB11886 | Infigratinib | approved, investigational | no | inhibitor | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitor | Details |
| DB06176 | Romidepsin | approved, investigational | no | inhibitor | Details |
| DB08834 | Tauroursodeoxycholic acid | approved, investigational | unknown | regulator | Details |
| DB15133 | Tepotinib | approved, investigational | no | inhibitor | Details |
| DB05467 | Palovarotene | approved, investigational | no | inhibitor | Details |