| DB00248 | Cabergoline | approved | yes | agonist | Details |
| DB00268 | Ropinirole | approved, investigational | yes | agonist | Details |
| DB00391 | Sulpiride | approved, investigational | yes | antagonist | Details |
| DB00420 | Promazine | approved, vet_approved | yes | antagonist | Details |
| DB00433 | Prochlorperazine | approved, vet_approved | yes | antagonist | Details |
| DB00450 | Droperidol | approved, vet_approved | yes | antagonist | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | yes | antagonist | Details |
| DB00502 | Haloperidol | approved | yes | antagonist | Details |
| DB00623 | Fluphenazine | approved | yes | antagonist | Details |
| DB00714 | Apomorphine | approved, investigational | yes | agonist | Details |
| DB00831 | Trifluoperazine | approved, investigational | yes | antagonist | Details |
| DB00915 | Amantadine | approved | yes | agonist | Details |
| DB00933 | Mesoridazine | approved, investigational | yes | antagonist | Details |
| DB01063 | Acetophenazine | approved | yes | antagonist | Details |
| DB01069 | Promethazine | approved, investigational | unknown | antagonist | Details |
| DB01100 | Pimozide | approved | yes | antagonist | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | yes | antagonist | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | yes | agonist | Details |
| DB01238 | Aripiprazole | approved, investigational | yes | antagonistpartial agonist | Details |
| DB00246 | Ziprasidone | approved | yes | antagonist | Details |
| DB00334 | Olanzapine | approved, investigational | yes | antagonist | Details |
| DB00363 | Clozapine | approved | yes | antagonist | Details |
| DB00372 | Thiethylperazine | approved, withdrawn | unknown | antagonist | Details |
| DB00490 | Buspirone | approved, investigational | yes | antagonist | Details |
| DB00508 | Triflupromazine | approved, vet_approved | yes | antagonist | Details |
| DB00568 | Cinnarizine | approved, investigational | no | other/unknown | Details |
| DB00679 | Thioridazine | approved, withdrawn | yes | antagonist | Details |
| DB00777 | Propiomazine | approved | unknown | antagonist | Details |
| DB00805 | Minaprine | approved | unknown | agonist | Details |
| DB00850 | Perphenazine | approved | yes | antagonist | Details |
| DB00875 | Flupentixol | approved, investigational, withdrawn | yes | antagonist | Details |
| DB01224 | Quetiapine | approved | yes | antagonist | Details |
| DB01233 | Metoclopramide | approved, investigational | yes | antagonist | Details |
| DB01235 | Levodopa | approved | yes | agonist | Details |
| DB01239 | Chlorprothixene | approved, experimental, investigational, withdrawn | yes | antagonist | Details |
| DB01267 | Paliperidone | approved | yes | antagonist | Details |
| DB01624 | Zuclopenthixol | approved, investigational | yes | antagonist | Details |
| DB01618 | Molindone | approved | yes | antagonist | Details |
| DB04842 | Fluspirilene | approved, investigational | yes | antagonist | Details |
| DB00589 | Lisuride | approved, investigational | yes | agonist | Details |
| DB00408 | Loxapine | approved | yes | antagonist | Details |
| DB00413 | Pramipexole | approved, investigational | yes | agonist | Details |
| DB00409 | Remoxipride | approved, withdrawn | yes | antagonist | Details |
| DB00696 | Ergotamine | approved | unknown | agonist | Details |
| DB04857 | Brasofensine | investigational | unknown | | Details |
| DB04888 | Bifeprunox | investigational | unknown | | Details |
| DB04889 | Bicifadine | investigational | unknown | | Details |
| DB06144 | Sertindole | approved, investigational, withdrawn | yes | antagonist | Details |
| DB12061 | Pardoprunox | investigational | unknown | | Details |
| DB04924 | Itopride | investigational | unknown | | Details |
| DB04946 | Iloperidone | approved | yes | antagonist | Details |
| DB01038 | Carphenazine | withdrawn | yes | antagonist | Details |
| DB05687 | BL-1020 | investigational | unknown | | Details |
| DB05766 | Norclozapine | investigational | unknown | | Details |
| DB06077 | Lumateperone | approved, investigational | yes | partial agonist | Details |
| DB06109 | YKP-1358 | investigational | unknown | antagonist | Details |
| DB05964 | Amitifadine | investigational | unknown | | Details |
| DB06216 | Asenapine | approved | yes | antagonist | Details |
| DB06229 | Ocaperidone | investigational | unknown | | Details |
| DB06477 | Sumanirole | investigational | unknown | | Details |
| DB04599 | Aniracetam | experimental | unknown | | Details |
| DB06288 | Amisulpride | approved, investigational | yes | antagonist | Details |
| DB05271 | Rotigotine | approved | yes | agonist | Details |
| DB01403 | Methotrimeprazine | approved, investigational | yes | antagonist | Details |
| DB01549 | Rolicyclidine | experimental, illicit | unknown | | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB00726 | Trimipramine | approved | unknown | other/unknown | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | unknown | antagonist | Details |
| DB01221 | Ketamine | approved, vet_approved | unknown | agonistpartial agonist | Details |
| DB00988 | Dopamine | approved | yes | agonist | Details |
| DB01614 | Acepromazine | experimental, vet_approved | yes | antagonist | Details |
| DB01621 | Pipotiazine | approved, investigational | yes | antagonist | Details |
| DB01622 | Thioproperazine | experimental | yes | antagonist | Details |
| DB01623 | Thiothixene | approved | yes | antagonist | Details |
| DB01425 | Alizapride | investigational | yes | antagonist | Details |
| DB08815 | Lurasidone | approved, investigational | yes | antagonist | Details |
| DB04844 | Tetrabenazine | approved, investigational | unknown | inhibitor | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | unknown | binder | Details |
| DB00458 | Imipramine | approved | unknown | binder | Details |
| DB00540 | Nortriptyline | approved | unknown | antagonist | Details |
| DB01043 | Memantine | approved, investigational | unknown | antagonistagonist | Details |
| DB00934 | Maprotiline | approved, investigational | unknown | binder | Details |
| DB01151 | Desipramine | approved, investigational | unknown | binder | Details |
| DB06148 | Mianserin | approved, investigational | unknown | antagonist | Details |
| DB09018 | Bromopride | investigational | yes | antagonist | Details |
| DB09207 | AS-8112 | experimental | unknown | antagonist | Details |
| DB09128 | Brexpiprazole | approved, investigational | unknown | partial agonist | Details |
| DB13025 | Tiapride | investigational | yes | blocker | Details |
| DB08922 | Perospirone | experimental | yes | antagonist | Details |
| DB09097 | Quinagolide | approved, investigational | unknown | agonist | Details |
| DB12478 | Piribedil | investigational | unknown | | Details |
| DB06454 | Sarizotan | investigational | unknown | partial agonist | Details |
| DB12518 | Raclopride | investigational | unknown | antagonist | Details |
| DB12093 | Tetrahydropalmatine | investigational | unknown | antagonist | Details |
| DB09194 | Etoperidone | withdrawn | unknown | antagonist | Details |
| DB09223 | Blonanserin | investigational | yes | antagonist | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | agonistinhibitor | Details |
| DB09225 | Zotepine | approved, investigational, withdrawn | yes | antagonist | Details |
| DB09224 | Melperone | investigational | yes | antagonist | Details |
| DB09286 | Pipamperone | investigational | unknown | antagonist | Details |
| DB11274 | Dihydro-alpha-ergocryptine | approved | yes | agonist | Details |
| DB12579 | JNJ-37822681 | investigational | yes | antagonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | yes | partial agonist | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | other/unknown | Details |
| DB01175 | Escitalopram | approved | unknown | inhibitor | Details |
| DB00734 | Risperidone | approved, investigational | yes | antagonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | agonist | Details |
| DB06016 | Cariprazine | approved, investigational | unknown | partial agonist | Details |