| DB01138 | Sulfinpyrazone | approved | yes | inhibitor | Details |
| DB04851 | Biricodar | investigational | unknown | | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitorinducer | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | inhibitorinducer | Details |
| DB00570 | Vinblastine | approved | unknown | substrateinhibitorinducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | inhibitorinducer | Details |
| DB02659 | Cholic Acid | approved | unknown | inducer | Details |
| DB01165 | Ofloxacin | approved | unknown | inhibitor | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | inhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | inhibitor | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB03467 | Naringenin | experimental | unknown | inhibitor | Details |
| DB02375 | Myricetin | experimental | unknown | inhibitor | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | inhibitor | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | inhibitor | Details |
| DB01645 | Genistein | investigational | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inhibitor | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00694 | Daunorubicin | approved | unknown | substrateinhibitor | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | inhibitor | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | substrateinhibitor | Details |
| DB00563 | Methotrexate | approved | unknown | substrateinhibitor | Details |
| DB01177 | Idarubicin | approved | unknown | inhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrateinhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inhibitor | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitor | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | substrateinhibitor | Details |
| DB05294 | Vandetanib | approved | unknown | inhibitor | Details |
| DB00345 | Aminohippuric acid | approved, investigational | unknown | substrate | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00693 | Fluorescein | approved | unknown | substrate | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrate | Details |
| DB00445 | Epirubicin | approved | unknown | substrate | Details |
| DB03825 | Rhodamine 6G | experimental | unknown | substrate | Details |
| DB00970 | Dactinomycin | approved, investigational | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00399 | Zoledronic acid | approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB01072 | Atazanavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB06335 | Saxagliptin | approved | unknown | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB08881 | Vemurafenib | approved | unknown | substrateinhibitor | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB09161 | Technetium Tc-99m sestamibi | approved, investigational | no | substrate | Details |
| DB00171 | ATP | investigational, nutraceutical | unknown | | Details |
| DB08855 | Leukotriene C4 | experimental, investigational | unknown | | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | | Details |
| DB13783 | Acemetacin | approved, investigational | no | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB00115 | Cyanocobalamin | approved, nutraceutical | unknown | | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | unknown | substrate | Details |
| DB08868 | Fingolimod | approved, investigational | unknown | inhibitorinducer | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | unknown | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB04851 | Biricodar | investigational | unknown | modulator | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |