| DB00216 | Eletriptan | approved, investigational | yes | agonist | Details |
| DB00315 | Zolmitriptan | approved, investigational | yes | agonist | Details |
| DB00952 | Naratriptan | approved, investigational | yes | agonist | Details |
| DB00953 | Rizatriptan | approved | yes | agonist | Details |
| DB00998 | Frovatriptan | approved, investigational | yes | agonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | yes | agonist | Details |
| DB00669 | Sumatriptan | approved, investigational | yes | agonist | Details |
| DB00696 | Ergotamine | approved | yes | agonist | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | agonist | Details |
| DB00960 | Pindolol | approved, investigational | unknown | other/unknownligand | Details |
| DB04884 | Dapoxetine | investigational | unknown | | Details |
| DB00571 | Propranolol | approved, investigational | unknown | other/unknown | Details |
| DB06096 | NXN-188 | investigational | unknown | | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | unknown | agonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | agonist | Details |
| DB00589 | Lisuride | approved, investigational | unknown | agonist | Details |
| DB00248 | Cabergoline | approved | unknown | agonist | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | agonist | Details |
| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB00363 | Clozapine | approved | unknown | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | antagonistligand | Details |
| DB01224 | Quetiapine | approved | unknown | ligand | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | unknown | partial agonist | Details |
| DB08807 | Bopindolol | experimental | unknown | | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | other/unknown | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB00247 | Methysergide | approved | unknown | binder | Details |
| DB00321 | Amitriptyline | approved | unknown | binder | Details |
| DB01359 | Penbutolol | approved, investigational | unknown | antagonist | Details |
| DB09068 | Vortioxetine | approved, investigational | yes | partial agonist | Details |
| DB06153 | Pizotifen | approved | unknown | antagonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | | Details |
| DB00935 | Oxymetazoline | approved, investigational | unknown | agonist | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | modulator | Details |