| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | | Details |
| DB01834 | (9R,10R)-9-(S-glutathionyl)-10-hydroxy-9,10-dihydrophenanthrene | experimental | unknown | | Details |
| DB01915 | S-Hydroxycysteine | experimental | unknown | | Details |
| DB02633 | Cibacron Blue | experimental | unknown | | Details |
| DB03814 | 2-(N-morpholino)ethanesulfonic acid | experimental | unknown | | Details |
| DB04132 | S-Hexylglutathione | experimental | unknown | | Details |
| DB03003 | Glutathione sulfonic acid | experimental | unknown | | Details |
| DB03686 | S-(4-nitrobenzyl)glutathione | experimental | unknown | | Details |
| DB04972 | Canfosfamide | investigational | unknown | | Details |
| DB05460 | Ezatiostat | investigational | unknown | | Details |
| DB07849 | S-NONYL-CYSTEINE | experimental | unknown | | Details |
| DB08370 | S-(4-BROMOBENZYL)CYSTEINE | experimental | unknown | | Details |
| DB00163 | Vitamin E | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB00291 | Chlorambucil | approved | unknown | substrate | Details |
| DB01008 | Busulfan | approved, investigational | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB00515 | Cisplatin | approved | unknown | substrate | Details |
| DB00958 | Carboplatin | approved | unknown | substrate | Details |
| DB00526 | Oxaliplatin | approved, investigational | no | substrate | Details |
| DB03619 | Deoxycholic acid | approved | unknown | | Details |
| DB06246 | Exisulind | investigational | unknown | inhibitor | Details |
| DB13014 | Hypericin | investigational | unknown | inhibitor | Details |
| DB00363 | Clozapine | approved | unknown | | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | | Details |
| DB11831 | Dinitrochlorobenzene | investigational | unknown | | Details |
| DB11672 | Curcumin | approved, investigational | unknown | | Details |
| DB00903 | Etacrynic acid | approved, investigational | unknown | inhibitor | Details |
| DB14001 | alpha-Tocopherol succinate | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB14002 | D-alpha-Tocopherol acetate | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB14924 | Ritlecitinib | approved, investigational | unknown | substrate | Details |