| DB01032 | Probenecid | approved, investigational | yes | inhibitor | Details |
| DB00759 | Tetracycline | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00595 | Oxytetracycline | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00917 | Dinoprostone | approved | unknown | inhibitor | Details |
| DB00456 | Cefalotin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01212 | Ceftriaxone | approved | unknown | inhibitor | Details |
| DB00493 | Cefotaxime | approved | unknown | inhibitor | Details |
| DB01329 | Cefoperazone | approved, investigational | unknown | inhibitor | Details |
| DB01327 | Cefazolin | approved | unknown | inhibitor | Details |
| DB01326 | Cefamandole | approved, experimental | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB00554 | Piroxicam | approved, investigational | unknown | inhibitor | Details |
| DB01053 | Benzylpenicillin | approved, vet_approved | unknown | inhibitor | Details |
| DB00345 | Aminohippuric acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB04519 | Caprylic acid | investigational | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | inhibitor | Details |
| DB00168 | Aspartame | investigational, nutraceutical | unknown | inhibitor | Details |
| DB00812 | Phenylbutazone | approved, vet_approved | unknown | inhibitor | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | inhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | inhibitor | Details |
| DB00936 | Salicylic acid | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB03553 | Glutaric Acid | experimental | unknown | inhibitor | Details |
| DB00695 | Furosemide | approved, vet_approved | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inhibitor | Details |
| DB00887 | Bumetanide | approved | unknown | inhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB01051 | Novobiocin | approved, investigational, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB00495 | Zidovudine | approved | unknown | | Details |
| DB01160 | Dinoprost tromethamine | approved, vet_approved | unknown | | Details |
| DB04133 | Degraded Cephaloridine | experimental | unknown | | Details |
| DB08846 | Ellagic acid | investigational | unknown | | Details |
| DB00493 | Cefotaxime | approved | unknown | | Details |
| DB01212 | Ceftriaxone | approved | unknown | | Details |
| DB11560 | Lesinurad | approved, investigational | yes | inhibitor | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB12377 | Relebactam | approved, investigational | unknown | substrate | Details |
| DB06282 | Levocetirizine | approved | unknown | substrate | Details |
| DB00999 | Hydrochlorothiazide | approved, vet_approved | unknown | substrate | Details |
| DB00642 | Pemetrexed | approved, investigational | no | substrate | Details |