| DB00280 | Disopyramide | approved | no | other/unknown | Details |
| DB00706 | Tamsulosin | approved, investigational | no | | Details |
| DB00908 | Quinidine | approved, investigational | unknown | binder | Details |
| DB00946 | Phenprocoumon | approved, investigational | no | | Details |
| DB01359 | Penbutolol | approved, investigational | unknown | other/unknown | Details |
| DB01429 | Aprindine | experimental | unknown | | Details |
| DB01418 | Acenocoumarol | approved, investigational | no | | Details |
| DB00682 | Warfarin | approved | no | | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | | Details |
| DB00540 | Nortriptyline | approved | no | binder | Details |
| DB00321 | Amitriptyline | approved | no | binder | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | | Details |
| DB00334 | Olanzapine | approved, investigational | no | binder | Details |
| DB00543 | Amoxapine | approved | no | | Details |
| DB00457 | Prazosin | approved | no | substrate | Details |
| DB00571 | Propranolol | approved, investigational | no | | Details |
| DB00458 | Imipramine | approved | no | | Details |
| DB01151 | Desipramine | approved, investigational | no | | Details |
| DB04821 | Nomifensine | approved, withdrawn | no | | Details |
| DB01156 | Bupropion | approved | no | antagonist | Details |
| DB00934 | Maprotiline | approved, investigational | no | | Details |
| DB01426 | Ajmaline | approved, experimental | unknown | | Details |
| DB00454 | Meperidine | approved | unknown | binder | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | | Details |
| DB08867 | Ulipristal | approved | no | substrate | Details |
| DB05294 | Vandetanib | approved | unknown | binder | Details |
| DB05521 | Telaprevir | approved, withdrawn | no | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | binder | Details |
| DB08881 | Vemurafenib | approved | unknown | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | binder | Details |
| DB08893 | Mirabegron | approved | no | binder | Details |
| DB08820 | Ivacaftor | approved | no | carrier | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB08907 | Canagliflozin | approved | unknown | substrate | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrate | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | binder | Details |
| DB00864 | Tacrolimus | approved, investigational | unknown | substrate | Details |
| DB08931 | Riociguat | approved | unknown | substrate | Details |
| DB11575 | Grazoprevir | approved | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | binder | Details |
| DB00276 | Amsacrine | approved, investigational | unknown | | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | binder | Details |
| DB00975 | Dipyridamole | approved | unknown | | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | | Details |
| DB09236 | Lacidipine | approved, investigational | unknown | binder | Details |
| DB09204 | Arotinolol | investigational | no | substrate | Details |
| DB09229 | Aranidipine | experimental | no | binder | Details |
| DB11148 | Butamben | approved, withdrawn | no | substrate | Details |
| DB11637 | Delamanid | approved, investigational | unknown | substrate | Details |
| DB00243 | Ranolazine | approved, investigational | no | binder | Details |
| DB01142 | Doxepin | approved, investigational | no | binder | Details |
| DB01126 | Dutasteride | approved, investigational | no | binder | Details |
| DB00343 | Diltiazem | approved, investigational | no | binder | Details |
| DB00481 | Raloxifene | approved, investigational | no | binder | Details |
| DB00490 | Buspirone | approved, investigational | unknown | binder | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | binder | Details |
| DB00333 | Methadone | approved | no | | Details |
| DB01233 | Metoclopramide | approved, investigational | unknown | binder | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | binder | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB01190 | Clindamycin | approved, vet_approved | unknown | substrate | Details |
| DB00246 | Ziprasidone | approved | unknown | | Details |
| DB01264 | Darunavir | approved | unknown | substrate | Details |
| DB01601 | Lopinavir | approved | unknown | substrate | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrate | Details |
| DB11642 | Pitolisant | approved, investigational | no | binder | Details |
| DB00734 | Risperidone | approved, investigational | unknown | binder | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | binder | Details |
| DB11853 | Relugolix | approved, investigational | unknown | binder | Details |
| DB15133 | Tepotinib | approved, investigational | unknown | binder | Details |
| DB00346 | Alfuzosin | approved, investigational | unknown | binder | Details |
| DB00853 | Temozolomide | approved, investigational | no | binder | Details |
| DB06237 | Avanafil | approved | unknown | binder | Details |
| DB00080 | Daptomycin | approved, investigational | no | binder | Details |
| DB12235 | Estetrol | approved, investigational | unknown | binder | Details |
| DB01627 | Lincomycin | approved, vet_approved | no | binder | Details |
| DB16703 | Belumosudil | approved, investigational | no | binder | Details |
| DB00877 | Sirolimus | approved, investigational | no | binder | Details |
| DB06234 | Maribavir | approved, investigational | no | binder | Details |
| DB09074 | Olaparib | approved | unknown | binder | Details |
| DB00220 | Nelfinavir | approved | no | binder | Details |
| DB00296 | Ropivacaine | approved | no | binder | Details |
| DB00572 | Atropine | approved, vet_approved | unknown | binder | Details |
| DB15149 | Futibatinib | approved, investigational | no | binder | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | binder | Details |
| DB05239 | Cobimetinib | approved, investigational | no | binder | Details |
| DB00363 | Clozapine | approved | no | binder | Details |
| DB00349 | Clobazam | approved, illicit | no | binder | Details |
| DB00683 | Midazolam | approved, illicit | no | binder | Details |
| DB09128 | Brexpiprazole | approved, investigational | no | substrate | Details |
| DB08906 | Fluticasone furoate | approved | no | binder | Details |
| DB09076 | Umeclidinium | approved | unknown | binder | Details |
| DB01042 | Melphalan | approved | unknown | binder | Details |
| DB08903 | Bedaquiline | approved | no | binder | Details |
| DB16200 | Iptacopan | approved, investigational | yes | binder | Details |