| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | binder | Details |
| DB00977 | Ethinylestradiol | approved | unknown | agonist | Details |
| DB01892 | Hyperforin | nutraceutical | unknown | | Details |
| DB04466 | SR12813 | experimental | unknown | | Details |
| DB00163 | Vitamin E | approved, nutraceutical, vet_approved | unknown | | Details |
| DB01045 | Rifampicin | approved | unknown | agonist | Details |
| DB01220 | Rifaximin | approved, investigational | no | agonist | Details |
| DB07080 | TO-901317 | experimental | unknown | | Details |
| DB00530 | Erlotinib | approved, investigational | yes | agonist | Details |
| DB08864 | Rilpivirine | approved | unknown | agonist | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | inducer | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | binder | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | activator | Details |
| DB11605 | Myrrh | approved | unknown | partial agonist | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | activator | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | activator | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | activator | Details |
| DB00252 | Phenytoin | approved, vet_approved | unknown | | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | activator | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | activator | Details |
| DB00754 | Ethotoin | approved | unknown | activator | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | activator | Details |
| DB00849 | Methylphenobarbital | approved | unknown | activator | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | unknown | activator | Details |
| DB13179 | Troleandomycin | approved | unknown | activator | Details |
| DB04468 | Afimoxifene | investigational | unknown | | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | agonist | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | | Details |
| DB01645 | Genistein | investigational | unknown | | Details |
| DB00431 | Lindane | approved, withdrawn | unknown | | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | | Details |
| DB02789 | Pregnenolone | approved, experimental | unknown | | Details |
| DB00421 | Spironolactone | approved | unknown | agonist | Details |
| DB08604 | Triclosan | approved, investigational | unknown | | Details |
| DB00675 | Tamoxifen | approved | unknown | | Details |
| DB06777 | Chenodeoxycholic acid | approved | unknown | | Details |
| DB01127 | Econazole | approved | unknown | partial agonist | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | partial agonist | Details |
| DB00239 | Oxiconazole | approved | unknown | partial agonist | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | antagonist | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | | Details |
| DB00499 | Flutamide | approved, investigational | unknown | | Details |
| DB01181 | Ifosfamide | approved | unknown | | Details |
| DB01393 | Bezafibrate | approved, investigational | unknown | partial agonist | Details |
| DB01068 | Clonazepam | approved, illicit | unknown | partial agonist | Details |
| DB01039 | Fenofibrate | approved | unknown | partial agonist | Details |
| DB00682 | Warfarin | approved | unknown | | Details |
| DB07931 | Hexestrol | withdrawn | unknown | | Details |
| DB04824 | Phenolphthalein | approved, withdrawn | unknown | | Details |
| DB02709 | Resveratrol | investigational | unknown | | Details |
| DB04930 | Permethrin | approved, investigational | unknown | | Details |
| DB11087 | Pyrethrum extract | approved | unknown | | Details |
| DB01115 | Nifedipine | approved | unknown | agonist | Details |
| DB12582 | Piperine | investigational | unknown | | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | activator | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | | Details |
| DB13873 | Fenofibric acid | approved | unknown | partial agonist | Details |
| DB14001 | alpha-Tocopherol succinate | approved, nutraceutical, vet_approved | unknown | | Details |
| DB14002 | D-alpha-Tocopherol acetate | approved, nutraceutical, vet_approved | unknown | | Details |
| DB05928 | Dovitinib | investigational | unknown | suppressor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | agonist | Details |