| DB00171 | ATP | investigational, nutraceutical | unknown | | Details |
| DB00778 | Roxithromycin | approved, investigational, withdrawn | unknown | | Details |
| DB04881 | Elacridar | investigational | unknown | | Details |
| DB04905 | Tesmilifene | investigational | yes | inducer | Details |
| DB05449 | FM-VP4 | investigational | unknown | | Details |
| DB06240 | Tariquidar | investigational | unknown | | Details |
| DB06191 | Zosuquidar | investigational | yes | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | substrateinhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00220 | Nelfinavir | approved | no | substrateinhibitorinducer | Details |
| DB00224 | Indinavir | approved | unknown | substrateinhibitorinducer | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | substrateinducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00206 | Reserpine | approved, investigational, withdrawn | unknown | substrateinhibitorinducer | Details |
| DB01115 | Nifedipine | approved | unknown | substrateinducer | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | inhibitorinducer | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitorinducer | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | inducer | Details |
| DB00656 | Trazodone | approved, investigational | unknown | inducer | Details |
| DB01149 | Nefazodone | approved, withdrawn | unknown | inhibitorinducer | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00390 | Digoxin | approved | unknown | substrateinhibitorinducer | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | inducer | Details |
| DB00451 | Levothyroxine | approved | unknown | inducer | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB02261 | Platelet Activating Factor | experimental | unknown | substrateinducer | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrateinducer | Details |
| DB04630 | Aldosterone | experimental, investigational | unknown | substrateinducer | Details |
| DB00864 | Tacrolimus | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00877 | Sirolimus | approved, investigational | no | substrateinhibitorinducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | substrateinducer | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | no | substrateinhibitor | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | inhibitorinducer | Details |
| DB01323 | St. John's Wort | approved, investigational, nutraceutical | unknown | inducer | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00570 | Vinblastine | approved | unknown | substrateinhibitorinducer | Details |
| DB02659 | Cholic Acid | approved | unknown | inducer | Details |
| DB00675 | Tamoxifen | approved | unknown | substrateinhibitorinducer | Details |
| DB00428 | Streptozocin | approved, investigational | unknown | inducer | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00694 | Daunorubicin | approved | unknown | substrateinhibitorinducer | Details |
| DB00908 | Quinidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB04540 | Cholesterol | approved, investigational | unknown | inhibitor | Details |
| DB00358 | Mefloquine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00381 | Amlodipine | approved | unknown | substrateinhibitor | Details |
| DB00972 | Azelastine | approved | unknown | inhibitor | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrateinhibitor | Details |
| DB00333 | Methadone | approved | unknown | inhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | inhibitor | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | inhibitor | Details |
| DB01076 | Atorvastatin | approved | no | substrateinhibitor | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00457 | Prazosin | approved | unknown | substrateinhibitormodulator | Details |
| DB01054 | Nitrendipine | approved, investigational | unknown | inhibitor | Details |
| DB00975 | Dipyridamole | approved | unknown | substrateinhibitor | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrateinhibitor | Details |
| DB01394 | Colchicine | approved | unknown | substrateinducer | Details |
| DB01211 | Clarithromycin | approved | unknown | substrateinhibitor | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00970 | Dactinomycin | approved, investigational | unknown | substrateinhibitor | Details |
| DB13179 | Troleandomycin | approved | unknown | inhibitor | Details |
| DB00831 | Trifluoperazine | approved, investigational | unknown | inhibitor | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | inhibitor | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitor | Details |
| DB01167 | Itraconazole | approved, investigational | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB02587 | Colforsin | experimental, investigational | unknown | inhibitor | Details |
| DB00623 | Fluphenazine | approved | unknown | inhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | inhibitor | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | inhibitor | Details |
| DB00421 | Spironolactone | approved | unknown | inducer | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | substrate | Details |
| DB00207 | Azithromycin | approved | unknown | substrateinhibitor | Details |
| DB00316 | Acetaminophen | approved | unknown | substrateinhibitor | Details |
| DB00196 | Fluconazole | approved, investigational | unknown | inhibitor | Details |
| DB00213 | Pantoprazole | approved | unknown | substrateinhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00678 | Losartan | approved | unknown | substrateinhibitor | Details |
| DB00584 | Enalapril | approved, vet_approved | unknown | inhibitor | Details |
| DB00590 | Doxazosin | approved | unknown | inhibitor | Details |
| DB01340 | Cilazapril | approved | unknown | inhibitor | Details |
| DB01197 | Captopril | approved | unknown | inhibitor | Details |
| DB00796 | Candesartan cilexetil | approved | unknown | inhibitor | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00696 | Ergotamine | approved | unknown | inhibitor | Details |
| DB01253 | Ergometrine | approved | unknown | inhibitor | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | inhibitor | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00836 | Loperamide | approved | unknown | substrate | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | inhibitor | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | inhibitor | Details |
| DB00401 | Nisoldipine | approved | unknown | inhibitor | Details |
| DB04832 | Zimelidine | approved, withdrawn | unknown | inhibitor | Details |
| DB00382 | Tacrine | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00669 | Sumatriptan | approved, investigational | unknown | substrate | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00458 | Imipramine | approved | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrateinhibitor | Details |
| DB00176 | Fluvoxamine | approved, investigational | unknown | inhibitor | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | unknown | inhibitor | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | inhibitor | Details |
| DB01142 | Doxepin | approved, investigational | unknown | substrate | Details |
| DB01151 | Desipramine | approved, investigational | unknown | inhibitor | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01239 | Chlorprothixene | approved, experimental, investigational, withdrawn | unknown | inhibitor | Details |
| DB00490 | Buspirone | approved, investigational | unknown | inhibitor | Details |
| DB01100 | Pimozide | approved | unknown | inhibitor | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | inhibitor | Details |
| DB00508 | Triflupromazine | approved, vet_approved | unknown | inhibitor | Details |
| DB00344 | Protriptyline | approved | unknown | inhibitor | Details |
| DB01069 | Promethazine | approved, investigational | unknown | inhibitor | Details |
| DB01244 | Bepridil | approved, withdrawn | unknown | inhibitor | Details |
| DB00455 | Loratadine | approved, investigational | no | substrateinhibitor | Details |
| DB00967 | Desloratadine | approved, investigational | unknown | inhibitor | Details |
| DB00285 | Venlafaxine | approved | unknown | substrateinhibitor | Details |
| DB01104 | Sertraline | approved | unknown | inhibitor | Details |
| DB00234 | Reboxetine | approved, experimental | unknown | inhibitor | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | inhibitor | Details |
| DB00215 | Citalopram | approved | unknown | substrateinhibitor | Details |
| DB01196 | Estramustine | approved, investigational | unknown | inhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrateinhibitor | Details |
| DB00875 | Flupentixol | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00351 | Megestrol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB02010 | Staurosporine | experimental | unknown | inhibitor | Details |
| DB01103 | Quinacrine | investigational | unknown | inhibitor | Details |
| DB01645 | Genistein | investigational | unknown | inhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | inhibitor | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB03467 | Naringenin | experimental | unknown | downregulator | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB00726 | Trimipramine | approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00276 | Amsacrine | approved, investigational | unknown | inhibitor | Details |
| DB00027 | Gramicidin D | approved | unknown | substrateinhibitor | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | inhibitor | Details |
| DB01601 | Lopinavir | approved | unknown | inhibitorinducer | Details |
| DB00520 | Caspofungin | approved | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | inhibitor | Details |
| DB01162 | Terazosin | approved | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | unknown | inhibitor | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | inhibitor | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | inhibitor | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00655 | Estrone | approved | unknown | substrateinducer | Details |
| DB01259 | Lapatinib | approved, investigational | unknown | inhibitor | Details |
| DB01263 | Posaconazole | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB01396 | Digitoxin | approved, investigational | unknown | substrate | Details |
| DB01208 | Sparfloxacin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB01224 | Quetiapine | approved | unknown | substrate | Details |
| DB00334 | Olanzapine | approved, investigational | no | substrate | Details |
| DB00363 | Clozapine | approved | unknown | substrate | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | substrate | Details |
| DB04690 | Camptothecin | experimental | unknown | substrate | Details |
| DB00860 | Prednisolone | approved, vet_approved | unknown | substrate | Details |
| DB01193 | Acebutolol | approved, investigational | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB00945 | Acetylsalicylic acid | approved, vet_approved | unknown | substrateinducermodulator | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | substrate | Details |
| DB00539 | Toremifene | approved, investigational | unknown | substrate | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00882 | Clomifene | approved, investigational | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substratedownregulatorregulator | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00373 | Timolol | approved | unknown | substrate | Details |
| DB01203 | Nadolol | approved | unknown | substrate | Details |
| DB00523 | Alitretinoin | approved, investigational | unknown | substrate | Details |
| DB01339 | Vecuronium | approved, investigational | unknown | substrate | Details |
| DB04840 | Debrisoquine | approved, investigational | unknown | substrate | Details |
| DB00441 | Gemcitabine | approved | no | substrate | Details |
| DB01030 | Topotecan | approved, investigational | unknown | substrate | Details |
| DB02901 | Stanolone | illicit, investigational | unknown | substrate | Details |
| DB00751 | Epinastine | approved, investigational | unknown | substrate | Details |
| DB00717 | Norethisterone | approved | unknown | inhibitor | Details |
| DB04573 | Estriol | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB03203 | Sphingosine | experimental | unknown | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB01202 | Levetiracetam | approved | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | unknown | substrate | Details |
| DB00585 | Nizatidine | approved | unknown | substrate | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01261 | Sitagliptin | approved, investigational | unknown | substrate | Details |
| DB01072 | Atazanavir | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB01169 | Arsenic trioxide | approved, investigational | unknown | inhibitor | Details |
| DB06772 | Cabazitaxel | approved | unknown | substrateinhibitor | Details |
| DB01583 | Liotrix | approved | unknown | inducer | Details |
| DB06287 | Temsirolimus | approved | unknown | substrateinhibitor | Details |
| DB01587 | Ketazolam | approved | unknown | substrate | Details |
| DB04877 | Voacamine | experimental | unknown | inhibitor | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB01182 | Propafenone | approved | unknown | inhibitor | Details |
| DB00216 | Eletriptan | approved, investigational | unknown | substrate | Details |
| DB04855 | Dronedarone | approved | no | inhibitor | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB06207 | Silodosin | approved | unknown | substrate | Details |
| DB06414 | Etravirine | approved | unknown | inhibitor | Details |
| DB06228 | Rivaroxaban | approved | unknown | substrate | Details |
| DB06695 | Dabigatran etexilate | approved | unknown | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB06702 | Fesoterodine | approved | unknown | substrate | Details |
| DB06212 | Tolvaptan | approved | no | substrateinhibitor | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB06589 | Pazopanib | approved | unknown | substrate | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB08873 | Boceprevir | approved, withdrawn | unknown | inhibitor | Details |
| DB05521 | Telaprevir | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB08874 | Fidaxomicin | approved | no | substrate | Details |
| DB05039 | Indacaterol | approved | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB08882 | Linagliptin | approved | unknown | substrate | Details |
| DB08827 | Lomitapide | approved, investigational | no | inhibitor | Details |
| DB08816 | Ticagrelor | approved | unknown | substrateinhibitor | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB06626 | Axitinib | approved, investigational | no | substrateinhibitor | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | substrate | Details |
| DB08889 | Carfilzomib | approved, investigational | unknown | substrateinhibitor | Details |
| DB08893 | Mirabegron | approved | unknown | substrateinhibitor | Details |
| DB08896 | Regorafenib | approved | unknown | substrateinhibitor | Details |
| DB08899 | Enzalutamide | approved | no | inhibitor | Details |
| DB08820 | Ivacaftor | approved | no | inhibitor | Details |
| DB06616 | Bosutinib | approved | no | substrate | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB08906 | Fluticasone furoate | approved | no | substrateinducer | Details |
| DB08907 | Canagliflozin | approved | unknown | substrateinhibitor | Details |
| DB08910 | Pomalidomide | approved | unknown | substrate | Details |
| DB00480 | Lenalidomide | approved | no | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrate | Details |
| DB05773 | Trastuzumab emtansine | approved, investigational | unknown | substrate | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB00758 | Clopidogrel | approved | no | substrate | Details |
| DB08916 | Afatinib | approved | unknown | substrateinhibitor | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB08934 | Sofosbuvir | approved | no | substrate | Details |
| DB06292 | Dapagliflozin | approved | unknown | substrate | Details |
| DB09076 | Umeclidinium | approved | no | substrate | Details |
| DB09075 | Edoxaban | approved | no | substrate | Details |
| DB09063 | Ceritinib | approved | no | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | no | substrateinhibitor | Details |
| DB09079 | Nintedanib | approved | no | substrateinhibitor | Details |
| DB09054 | Idelalisib | approved | no | substrateinhibitor | Details |
| DB09065 | Cobicistat | approved | unknown | inhibitor | Details |
| DB09291 | Rolapitant | approved, investigational | no | inhibitor | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | substrateinhibitor | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | inhibitor | Details |
| DB06603 | Panobinostat | approved, investigational | no | substrate | Details |
| DB09330 | Osimertinib | approved | no | substrate | Details |
| DB11362 | Selexipag | approved | no | substrate | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB09296 | Ombitasvir | approved, investigational | no | substrate | Details |
| DB11574 | Elbasvir | approved | no | substrateinhibitor | Details |
| DB11575 | Grazoprevir | approved | no | substrate | Details |
| DB09161 | Technetium Tc-99m sestamibi | approved, investigational | no | substrate | Details |
| DB11581 | Venetoclax | approved, investigational | no | substrateinhibitor | Details |
| DB05015 | Belinostat | approved, investigational | unknown | substrate | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrateinhibitor | Details |
| DB09027 | Ledipasvir | approved | no | substratetransporter | Details |
| DB09198 | Lobeglitazone | experimental | no | | Details |
| DB09031 | Miltefosine | approved, investigational | unknown | | Details |
| DB09280 | Lumacaftor | approved | no | inhibitorinducer | Details |
| DB11828 | Neratinib | approved, investigational | unknown | inhibitor | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrateinhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB05889 | Inotuzumab ozogamicin | approved, investigational | unknown | substrate | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | substrateinhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12364 | Betrixaban | approved, investigational | no | substrate | Details |
| DB13919 | Candesartan | experimental | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | substrateinhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | substrateinhibitor | Details |
| DB09270 | Ubidecarenone | approved, investigational, nutraceutical | no | substrate | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | substrate | Details |
| DB13943 | Testosterone cypionate | approved | unknown | inhibitor | Details |
| DB13944 | Testosterone enanthate | approved | unknown | inhibitor | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inhibitor | Details |
| DB09160 | Technetium Tc-99m tetrofosmin | approved | no | binder | Details |
| DB13951 | Stanolone acetate | experimental | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01420 | Testosterone propionate | approved, investigational, vet_approved, withdrawn | no | substrate | Details |
| DB11901 | Apalutamide | approved, investigational | unknown | inducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB11251 | Tocopherol | approved, investigational | no | transporter | Details |
| DB14003 | alpha-Tocopherol acetate | approved | no | substrate | Details |
| DB09099 | Somatostatin | approved, investigational | unknown | substrate | Details |
| DB11635 | Tocofersolan | approved | unknown | antagonist | Details |
| DB11641 | Vinflunine | approved, investigational | no | substrate | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB11995 | Avatrombopag | approved, investigational | no | substrate | Details |
| DB09297 | Paritaprevir | approved, investigational | unknown | substrate | Details |
| DB09183 | Dasabuvir | approved | unknown | substrate | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | | Details |
| DB14062 | Concanamycin A | experimental | yes | inhibitor | Details |
| DB14061 | Hycanthone | experimental | yes | inhibitor | Details |
| DB14063 | Dexverapamil | experimental | yes | inhibitor | Details |
| DB14064 | Emopamil | experimental | yes | inhibitor | Details |
| DB14065 | Lomerizine | experimental | yes | inhibitor | Details |
| DB14066 | Tetrandrine | experimental | unknown | inhibitor | Details |
| DB14067 | Dofequidar | experimental, investigational | unknown | inhibitor | Details |
| DB14068 | Dexniguldipine | experimental | unknown | inhibitor | Details |
| DB14069 | ONT-093 | investigational | yes | inhibitor | Details |
| DB14070 | HM-30181 | experimental | yes | inhibitor | Details |
| DB14071 | Desmethylsertraline | experimental | unknown | inhibitor | Details |
| DB14072 | Reversin 121 | experimental | yes | inhibitor | Details |
| DB14146 | Loxicodegol | investigational | unknown | | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | | Details |
| DB14568 | Ivosidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11979 | Elagolix | approved, investigational | unknown | substrateinhibitor | Details |
| DB13867 | Fluticasone | approved, experimental | no | substrate | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00613 | Amodiaquine | approved, investigational | unknown | inhibitor | Details |
| DB01087 | Primaquine | approved | unknown | inhibitor | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | inhibitor | Details |
| DB01267 | Paliperidone | approved | unknown | substrateinhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB13125 | Lusutrombopag | approved, investigational | unknown | substrate | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | | Details |
| DB14641 | Estriol tripropionate | experimental | unknown | | Details |
| DB11952 | Duvelisib | approved, investigational | no | substrate | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB11760 | Talazoparib | approved, investigational | unknown | substrate | Details |
| DB12455 | Omadacycline | approved, investigational | unknown | substrate | Details |
| DB12836 | Grapiprant | investigational, vet_approved | no | substrate | Details |
| DB12035 | Sarecycline | approved, investigational | unknown | inhibitor | Details |
| DB11753 | Rifamycin | approved, investigational | no | substrateinhibitor | Details |
| DB11963 | Dacomitinib | approved, investigational | no | substrateinhibitor | Details |
| DB11855 | Revefenacin | approved, investigational | no | substrate | Details |
| DB12141 | Gilteritinib | approved, investigational | no | substrate | Details |
| DB14126 | Tenofovir | experimental, investigational | no | substrate | Details |
| DB00300 | Tenofovir disoproxil | approved, investigational | unknown | substrateinhibitor | Details |
| DB09299 | Tenofovir alafenamide | approved | unknown | substrate | Details |
| DB01264 | Darunavir | approved | unknown | substrateinhibitorinducer | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrateinhibitor | Details |
| DB00862 | Vardenafil | approved | unknown | substrateinhibitor | Details |
| DB00776 | Oxcarbazepine | approved | unknown | substrate | Details |
| DB00248 | Cabergoline | approved | no | substrate | Details |
| DB06480 | Prucalopride | approved | no | substrate | Details |
| DB00734 | Risperidone | approved, investigational | unknown | substrate | Details |
| DB01117 | Atovaquone | approved | no | inhibitor | Details |
| DB00788 | Naproxen | approved, vet_approved | no | inhibitor | Details |
| DB00615 | Rifabutin | approved, investigational | unknown | inducer | Details |
| DB12582 | Piperine | investigational | unknown | inhibitor | Details |
| DB11978 | Glasdegib | approved, investigational | no | substrateinhibitor | Details |
| DB09074 | Olaparib | approved | no | substrateinhibitor | Details |
| DB00243 | Ranolazine | approved, investigational | no | substrateinhibitor | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00341 | Cetirizine | approved | no | substrateinhibitor | Details |
| DB09073 | Palbociclib | approved, investigational | no | substrateinhibitor | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | substrate | Details |
| DB13867 | Fluticasone | approved, experimental | unknown | substrate | Details |
| DB12147 | Erdafitinib | approved, investigational | no | substrateinhibitor | Details |
| DB00736 | Esomeprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00476 | Duloxetine | approved | unknown | inhibitor | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB12015 | Alpelisib | approved, investigational | unknown | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | substrateinhibitor | Details |
| DB00768 | Olopatadine | approved | no | substrate | Details |
| DB00698 | Nitrofurantoin | approved, vet_approved | unknown | substrate | Details |
| DB00451 | Levothyroxine | approved | no | inducer | Details |
| DB00394 | Beclomethasone dipropionate | approved, investigational | unknown | substrateinducer | Details |
| DB00612 | Bisoprolol | approved | unknown | substrateinhibitor | Details |
| DB00916 | Metronidazole | approved | unknown | inhibitor | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | substrate | Details |
| DB11986 | Entrectinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12825 | Lefamulin | approved, investigational | unknown | substrate | Details |
| DB01222 | Budesonide | approved | no | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB01233 | Metoclopramide | approved, investigational | unknown | substrate | Details |
| DB01175 | Escitalopram | approved | unknown | substrate | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | inhibitor | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrate | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | substrate | Details |
| DB01418 | Acenocoumarol | approved, investigational | unknown | substrate | Details |
| DB05676 | Apremilast | approved, investigational | unknown | substrate | Details |
| DB11732 | Lasmiditan | approved, investigational | unknown | substrateinhibitor | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | substrateinhibitor | Details |
| DB15566 | Prednisolone acetate | approved, vet_approved | unknown | substrate | Details |
| DB15035 | Zanubrutinib | approved, investigational | no | substrate | Details |
| DB00273 | Topiramate | approved | unknown | substrate | Details |
| DB09237 | Levamlodipine | approved, investigational | unknown | substrate | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | no | substrate | Details |
| DB13007 | Enfortumab vedotin | approved, investigational | unknown | substrate | Details |
| DB11951 | Lemborexant | approved, investigational | unknown | substrate | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | substrate | Details |
| DB15091 | Upadacitinib | approved, investigational | no | substrateinhibitor | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | substrate | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitormodulator | Details |
| DB00993 | Azathioprine | approved | unknown | substrate | Details |
| DB00557 | Hydroxyzine | approved | unknown | substrate | Details |
| DB11077 | Polyethylene glycol 400 | approved | unknown | inhibitor | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | substrate | Details |
| DB01006 | Letrozole | approved, investigational | unknown | substrate | Details |
| DB00246 | Ziprasidone | approved | unknown | | Details |
| DB01190 | Clindamycin | approved, vet_approved | unknown | substrate | Details |
| DB09287 | Polyethylene glycol | approved, vet_approved | no | inhibitor | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | inhibitor | Details |
| DB11770 | Talinolol | investigational | unknown | substrate | Details |
| DB04881 | Elacridar | investigational | unknown | inhibitor | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB11869 | Valspodar | investigational | unknown | inhibitor | Details |
| DB00518 | Albendazole | approved, vet_approved | no | substrate | Details |
| DB05239 | Cobimetinib | approved, investigational | no | substrate | Details |
| DB06670 | Odanacatib | investigational | unknown | substrate | Details |
| DB04877 | Voacamine | experimental | no | inhibitor | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inducer | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrate | Details |
| DB11363 | Alectinib | approved, investigational | unknown | inhibitor | Details |
| DB14723 | Larotrectinib | approved, investigational | no | substrate | Details |
| DB00588 | Fluticasone propionate | approved | unknown | substrate | Details |
| DB11430 | Monensin | experimental, vet_approved | unknown | substrate | Details |
| DB03825 | Rhodamine 6G | experimental | unknown | substrate | Details |
| DB09239 | Niguldipine | experimental | unknown | inhibitor | Details |
| DB04851 | Biricodar | investigational | unknown | inhibitor | Details |
| DB06240 | Tariquidar | investigational | unknown | inhibitor | Details |
| DB12799 | Laniquidar | investigational | unknown | inhibitor | Details |
| DB12923 | Gallopamil | investigational | unknown | inhibitor | Details |
| DB06420 | Annamycin | investigational | unknown | | Details |
| DB00540 | Nortriptyline | approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | substrate | Details |
| DB00652 | Pentazocine | approved, vet_approved | unknown | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01590 | Everolimus | approved | unknown | substrateinhibitor | Details |
| DB01212 | Ceftriaxone | approved | unknown | inhibitor | Details |
| DB00872 | Conivaptan | approved, investigational | unknown | inhibitor | Details |
| DB11544 | Salinomycin | vet_approved | unknown | inhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | inhibitor | Details |
| DB14057 | Valinomycin | experimental | unknown | substrateinhibitor | Details |
| DB04908 | Flibanserin | approved, investigational | unknown | inhibitor | Details |
| DB09039 | Eliglustat | approved, investigational | no | substrateinhibitor | Details |
| DB01128 | Bicalutamide | approved | unknown | inhibitor | Details |
| DB00648 | Mitotane | approved | unknown | inhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrateinhibitor | Details |
| DB04960 | Tipifarnib | investigational | unknown | inhibitor | Details |
| DB09048 | Netupitant | approved, investigational | unknown | inhibitor | Details |
| DB09034 | Suvorexant | approved, investigational | unknown | | Details |
| DB09030 | Vorapaxar | approved | unknown | | Details |
| DB05294 | Vandetanib | approved | unknown | inhibitor | Details |
| DB14062 | Concanamycin A | experimental | unknown | inhibitor | Details |
| DB14061 | Hycanthone | experimental | unknown | inhibitor | Details |
| DB08881 | Vemurafenib | approved | unknown | substrateinhibitor | Details |
| DB14063 | Dexverapamil | experimental | unknown | inhibitor | Details |
| DB14064 | Emopamil | experimental | unknown | inhibitor | Details |
| DB14065 | Lomerizine | experimental | unknown | inhibitor | Details |
| DB14066 | Tetrandrine | experimental | unknown | inhibitor | Details |
| DB14069 | ONT-093 | investigational | unknown | inhibitor | Details |
| DB14067 | Dofequidar | experimental, investigational | unknown | inhibitor | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | inhibitor | Details |
| DB12457 | Rimegepant | approved, investigational | unknown | substrate | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | inhibitor | Details |
| DB00253 | Medrysone | approved | unknown | substrate | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | substrateinhibitor | Details |
| DB12612 | Ozanimod | approved, investigational | unknown | substrate | Details |
| DB08868 | Fingolimod | approved, investigational | no | inhibitor | Details |
| DB07565 | Chloramphenicol succinate | approved | unknown | substrate | Details |
| DB11689 | Selumetinib | approved, investigational | unknown | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | substrateinducer | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | substrate | Details |
| DB15102 | Pemigatinib | approved, investigational | no | substrateinhibitor | Details |
| DB00315 | Zolmitriptan | approved, investigational | no | | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | substrate | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB04845 | Ixabepilone | approved, investigational | unknown | substrateinhibitor | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB14840 | Ripretinib | approved | unknown | substrateinhibitor | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | substrateinhibitor | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB06419 | Cethromycin | investigational | unknown | substrateinhibitor | Details |
| DB00674 | Galantamine | approved | no | inhibitor | Details |
| DB09026 | Aliskiren | approved, investigational | no | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | substrate | Details |
| DB00188 | Bortezomib | approved, investigational | no | substrate | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | substrateinducer | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | substrateinhibitor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB00104 | Octreotide | approved, investigational | unknown | substrate | Details |
| DB11796 | Fostemsavir | approved, investigational | unknown | substrate | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB15822 | Pralsetinib | approved, investigational | no | substrateinhibitor | Details |
| DB14845 | Filgotinib | approved, investigational | unknown | substrate | Details |
| DB15982 | Berotralstat | approved | no | substrateinhibitor | Details |
| DB11853 | Relugolix | approved, investigational | unknown | substrateinhibitor | Details |
| DB14895 | Vibegron | approved, investigational | no | substrate | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | substrateinducer | Details |
| DB11632 | Opicapone | approved, investigational | no | substrate | Details |
| DB15456 | Vericiguat | approved, investigational | unknown | substrate | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | substrate | Details |
| DB11693 | Voclosporin | approved, investigational | unknown | substrateinhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | no | substrateinhibitor | Details |
| DB00052 | Somatotropin | approved, investigational | unknown | substrate | Details |
| DB00346 | Alfuzosin | approved, investigational | unknown | substrate | Details |
| DB15442 | Trilaciclib | approved, investigational | unknown | substrate | Details |
| DB14989 | Umbralisib | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | substrate | Details |
| DB00853 | Temozolomide | approved, investigational | no | substrate | Details |
| DB06237 | Avanafil | approved | unknown | substrate | Details |
| DB11800 | Tivozanib | approved, investigational | unknown | substrate | Details |
| DB00080 | Daptomycin | approved, investigational | no | substrate | Details |
| DB06288 | Amisulpride | approved, investigational | no | substrate | Details |
| DB08995 | Diosmin | approved, investigational | unknown | inhibitor | Details |
| DB04876 | Vildagliptin | approved, investigational | no | substrate | Details |
| DB08822 | Azilsartan medoxomil | approved, investigational | no | inhibitor | Details |
| DB00360 | Sapropterin | approved, investigational | unknown | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitor | Details |
| DB16222 | Loncastuximab tesirine | approved, investigational | unknown | substrate | Details |
| DB15569 | Sotorasib | approved, investigational | unknown | inhibitor | Details |
| DB11886 | Infigratinib | approved, investigational | no | substrateinhibitor | Details |
| DB12471 | Ibrexafungerp | approved, investigational | unknown | substratetransporter | Details |
| DB16703 | Belumosudil | approved, investigational | no | substrateinhibitor | Details |
| DB16261 | Odevixibat | approved, investigational | unknown | substrate | Details |
| DB15463 | Belzutifan | approved, investigational | no | substrate | Details |
| DB16220 | Lonapegsomatropin | approved, investigational | unknown | substrate | Details |
| DB16390 | Mobocertinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB16732 | Tisotumab vedotin | approved | no | substrate | Details |
| DB16098 | Atogepant | approved, investigational | no | substrate | Details |
| DB08931 | Riociguat | approved | no | substrate | Details |
| DB15011 | Avacopan | approved, investigational | no | substrate | Details |
| DB12597 | Asciminib | approved, investigational | no | substrateinhibitor | Details |
| DB06234 | Maribavir | approved, investigational | no | inhibitor | Details |
| DB16691 | Nirmatrelvir | approved, investigational | no | substrateinhibitor | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | inhibitor | Details |
| DB14973 | Abrocitinib | approved, investigational | unknown | inhibitor | Details |
| DB16236 | Mitapivat | approved, investigational | no | substrateinhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB11697 | Pacritinib | approved, investigational | no | inhibitor | Details |
| DB06016 | Cariprazine | approved, investigational | unknown | inhibitor | Details |
| DB16407 | Azvudine | investigational | unknown | activatorregulator | Details |
| DB12541 | SAR-405838 | investigational | no | substrate | Details |
| DB00661 | Verapamil | approved | unknown | inhibitorblocker | Details |
| DB09118 | Stiripentol | approved | unknown | inhibitor | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | inhibitor | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | unknown | substrateinhibitor | Details |
| DB15673 | Lenacapavir | approved, investigational | no | substrate | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | substrateinhibitor | Details |
| DB15149 | Futibatinib | approved, investigational | no | substrateinhibitor | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | inhibitor | Details |
| DB11793 | Niraparib | approved, investigational | no | substrate | Details |
| DB12489 | Mirvetuximab soravtansine | approved, investigational | no | substrate | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB12240 | Polatuzumab vedotin | approved, investigational | no | substrate | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | inhibitor | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06374 | Elacestrant | approved, investigational | unknown | inhibitor | Details |
| DB00683 | Midazolam | approved, illicit | no | substrate | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | substrateinhibitor | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | substrate | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrate | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | inhibitor | Details |
| DB09082 | Vilanterol | approved | no | substrate | Details |
| DB12874 | Quizartinib | approved, investigational | no | substrateinhibitor | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | substrateinhibitor | Details |
| DB15097 | Gefapixant | approved, investigational | no | substrate | Details |
| DB11967 | Binimetinib | approved, investigational | no | substrate | Details |
| DB16826 | Repotrectinib | approved, investigational | no | substrateinhibitor | Details |
| DB12005 | Nirogacestat | approved, investigational | no | substrateinhibitor | Details |