| DB04851 | Biricodar | investigational | unknown | | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | inhibitor | Details |
| DB03467 | Naringenin | experimental | unknown | inhibitor | Details |
| DB01030 | Topotecan | approved, investigational | unknown | substrate | Details |
| DB01051 | Novobiocin | approved, investigational, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00655 | Estrone | approved | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01094 | Hesperetin | experimental | unknown | inhibitor | Details |
| DB01645 | Genistein | investigational | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB01016 | Glyburide | approved | unknown | substrate | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrate | Details |
| DB00213 | Pantoprazole | approved | unknown | substrateinhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | substrate | Details |
| DB02115 | Daidzin | experimental | unknown | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | no | substrateinhibitor | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | inhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00457 | Prazosin | approved | unknown | substrate | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inhibitor | Details |
| DB04881 | Elacridar | investigational | unknown | inhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | inhibitor | Details |
| DB05294 | Vandetanib | approved | unknown | inhibitor | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB00970 | Dactinomycin | approved, investigational | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00669 | Sumatriptan | approved, investigational | unknown | substrate | Details |
| DB00694 | Daunorubicin | approved | unknown | substrate | Details |
| DB04540 | Cholesterol | approved, investigational | unknown | inducer | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00158 | Folic acid | approved, nutraceutical, vet_approved | unknown | substrate | Details |
| DB03496 | Alvocidib | experimental, investigational | unknown | substrate | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrate | Details |
| DB00444 | Teniposide | approved | unknown | substrate | Details |
| DB00698 | Nitrofurantoin | approved, vet_approved | unknown | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | substrate | Details |
| DB04690 | Camptothecin | experimental | unknown | substrate | Details |
| DB00740 | Riluzole | approved, investigational | unknown | substrate | Details |
| DB00242 | Cladribine | approved, investigational | unknown | substrate | Details |
| DB00631 | Clofarabine | approved, investigational | unknown | substrate | Details |
| DB00526 | Oxaliplatin | approved, investigational | no | substrate | Details |
| DB06772 | Cabazitaxel | approved | unknown | inhibitor | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB06589 | Pazopanib | approved | unknown | substrate | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB08880 | Teriflunomide | approved | unknown | substrateinhibitor | Details |
| DB01097 | Leflunomide | approved, investigational | unknown | substrate | Details |
| DB08881 | Vemurafenib | approved | unknown | substrateinhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | inhibitor | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrateinhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | antagonist | Details |
| DB00285 | Venlafaxine | approved | unknown | inducer | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB08916 | Afatinib | approved | unknown | substrateinhibitor | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB00515 | Cisplatin | approved | unknown | substrate | Details |
| DB00958 | Carboplatin | approved | unknown | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB08934 | Sofosbuvir | approved | no | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | no | substrate | Details |
| DB09054 | Idelalisib | approved | no | substrate | Details |
| DB09065 | Cobicistat | approved | unknown | inhibitor | Details |
| DB09291 | Rolapitant | approved, investigational | no | inhibitor | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | inhibitor | Details |
| DB05239 | Cobimetinib | approved, investigational | no | weak inhibitor | Details |
| DB09330 | Osimertinib | approved | no | substrate | Details |
| DB11363 | Alectinib | approved, investigational | no | inhibitor | Details |
| DB08931 | Riociguat | approved | no | substrate | Details |
| DB09183 | Dasabuvir | approved | unknown | inhibitor | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrateinhibitor | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB09027 | Ledipasvir | approved | no | transporter | Details |
| DB09296 | Ombitasvir | approved, investigational | no | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrateinhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | substrateinhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | no | substrateinhibitor | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | substrateinhibitor | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB11827 | Ertugliflozin | approved, investigational | unknown | substrate | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11901 | Apalutamide | approved, investigational | unknown | inducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB12010 | Fostamatinib | approved, investigational | no | inhibitor | Details |
| DB09297 | Paritaprevir | approved, investigational | unknown | inhibitor | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitorinducer | Details |
| DB13125 | Lusutrombopag | approved, investigational | unknown | substrate | Details |
| DB06210 | Eltrombopag | approved | unknown | inhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inhibitorinducer | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | inhibitor | Details |
| DB11952 | Duvelisib | approved, investigational | no | substrate | Details |
| DB11760 | Talazoparib | approved, investigational | unknown | substrate | Details |
| DB11963 | Dacomitinib | approved, investigational | no | substrateinhibitor | Details |
| DB11581 | Venetoclax | approved, investigational | unknown | inhibitor | Details |
| DB11855 | Revefenacin | approved, investigational | no | substrate | Details |
| DB12141 | Gilteritinib | approved, investigational | no | inhibitor | Details |
| DB06228 | Rivaroxaban | approved | unknown | substrate | Details |
| DB09279 | Fimasartan | investigational | unknown | substrate | Details |
| DB11978 | Glasdegib | approved, investigational | no | substrateinhibitor | Details |
| DB09074 | Olaparib | approved | no | inhibitor | Details |
| DB00437 | Allopurinol | approved | unknown | substrate | Details |
| DB09073 | Palbociclib | approved, investigational | no | substrateinhibitor | Details |
| DB08907 | Canagliflozin | approved | unknown | | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | substrate | Details |
| DB09299 | Tenofovir alafenamide | approved | no | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB12015 | Alpelisib | approved, investigational | unknown | substrate | Details |
| DB00394 | Beclomethasone dipropionate | approved, investigational | unknown | inhibitor | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | substrate | Details |
| DB00843 | Donepezil | approved | unknown | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | inhibitor | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB09079 | Nintedanib | approved | unknown | | Details |
| DB00201 | Caffeine | approved | unknown | inhibitor | Details |
| DB11732 | Lasmiditan | approved, investigational | unknown | inhibitor | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | unknown | substrate | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | substrateinhibitor | Details |
| DB15091 | Upadacitinib | approved, investigational | no | substrateinhibitor | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | substrate | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitormodulator | Details |
| DB11644 | Tafamidis | approved, investigational | unknown | inhibitor | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | substrate | Details |
| DB14723 | Larotrectinib | approved, investigational | no | substrate | Details |
| DB11712 | Tezacaftor | approved, investigational | no | substrateinhibitor | Details |
| DB12457 | Rimegepant | approved, investigational | unknown | substrate | Details |
| DB12612 | Ozanimod | approved, investigational | unknown | substrate | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB11689 | Selumetinib | approved, investigational | unknown | substrate | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | substrate | Details |
| DB15102 | Pemigatinib | approved, investigational | no | substrate | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | inhibitor | Details |
| DB06813 | Pralatrexate | approved, investigational | no | substrate | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB14840 | Ripretinib | approved | unknown | substrateinhibitor | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11796 | Fostemsavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB11820 | Nifurtimox | approved, investigational | unknown | substrate | Details |
| DB15822 | Pralsetinib | approved, investigational | no | substrateinhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | inhibitor | Details |
| DB15982 | Berotralstat | approved | unknown | substrate | Details |
| DB11853 | Relugolix | approved, investigational | unknown | inhibitor | Details |
| DB11632 | Opicapone | approved, investigational | no | substrate | Details |
| DB15456 | Vericiguat | approved, investigational | unknown | substrate | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | substrate | Details |
| DB15133 | Tepotinib | approved, investigational | no | inhibitor | Details |
| DB15442 | Trilaciclib | approved, investigational | unknown | substrate | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | substrate | Details |
| DB00853 | Temozolomide | approved, investigational | no | substrate | Details |
| DB06237 | Avanafil | approved | unknown | inhibitor | Details |
| DB04854 | Febuxostat | approved | no | inhibitor | Details |
| DB11800 | Tivozanib | approved, investigational | no | inhibitor | Details |
| DB06288 | Amisulpride | approved, investigational | no | substrate | Details |
| DB15569 | Sotorasib | approved, investigational | unknown | inhibitor | Details |
| DB11886 | Infigratinib | approved, investigational | no | substrateinhibitor | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB16703 | Belumosudil | approved, investigational | no | inhibitor | Details |
| DB16390 | Mobocertinib | approved, investigational | unknown | inhibitor | Details |
| DB16098 | Atogepant | approved, investigational | no | substrate | Details |
| DB12597 | Asciminib | approved, investigational | no | substrateinhibitor | Details |
| DB06234 | Maribavir | approved, investigational | no | inhibitor | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | inhibitor | Details |
| DB04847 | Roxadustat | approved, investigational | unknown | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB11697 | Pacritinib | approved, investigational | no | inhibitor | Details |
| DB13055 | Oteseconazole | approved, investigational | no | inhibitor | Details |
| DB16407 | Azvudine | investigational | unknown | regulator | Details |
| DB12020 | Tecovirimat | approved, investigational | unknown | inhibitor | Details |
| DB09118 | Stiripentol | approved | unknown | inhibitor | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | unknown | inhibitor | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | binder | Details |
| DB15149 | Futibatinib | approved, investigational | no | substrate | Details |
| DB17083 | Linzagolix | approved | no | substrate | Details |
| DB11793 | Niraparib | approved, investigational | no | substrateinhibitor | Details |
| DB00642 | Pemetrexed | approved, investigational | no | | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06374 | Elacestrant | approved, investigational | unknown | inhibitor | Details |
| DB11682 | Daprodustat | approved, investigational | no | substrate | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | substrateinhibitor | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrateinhibitor | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | inhibitor | Details |
| DB12874 | Quizartinib | approved, investigational | no | inhibitor | Details |
| DB05467 | Palovarotene | approved, investigational | no | inhibitor | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB15097 | Gefapixant | approved, investigational | no | substrate | Details |
| DB11967 | Binimetinib | approved, investigational | no | substrate | Details |
| DB12218 | Capivasertib | approved, investigational | no | inhibitor | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inhibitor | Details |
| DB06636 | Isavuconazonium | approved, investigational | unknown | inhibitor | Details |
| DB11995 | Avatrombopag | approved, investigational | no | inhibitor | Details |