| DB00171 | ATP | investigational, nutraceutical | unknown | | Details |
| DB01138 | Sulfinpyrazone | approved | yes | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrate | Details |
| DB01892 | Hyperforin | nutraceutical | unknown | inducer | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | inducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB01169 | Arsenic trioxide | approved, investigational | unknown | inducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB00515 | Cisplatin | approved | unknown | inducer | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | inducer | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | inducer | Details |
| DB02659 | Cholic Acid | approved | unknown | inducer | Details |
| DB01115 | Nifedipine | approved | unknown | inducer | Details |
| DB00977 | Ethinylestradiol | approved | unknown | inhibitorinducer | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00570 | Vinblastine | approved | unknown | substrateinhibitorinducer | Details |
| DB00421 | Spironolactone | approved | unknown | inducer | Details |
| DB00876 | Eprosartan | approved | unknown | inducer | Details |
| DB00275 | Olmesartan | approved, investigational | unknown | substrateinducer | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | substrateinhibitor | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00206 | Reserpine | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrateinhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | substrateinhibitor | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | substrateinhibitor | Details |
| DB00695 | Furosemide | approved, vet_approved | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00563 | Methotrexate | approved | unknown | substrateinhibitor | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | inhibitor | Details |
| DB01208 | Sparfloxacin | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00978 | Lomefloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01165 | Ofloxacin | approved | unknown | inhibitor | Details |
| DB00116 | Tetrahydrofolic acid | nutraceutical | unknown | inhibitor | Details |
| DB04789 | 5-methyltetrahydrofolic acid | investigational, nutraceutical | unknown | inhibitor | Details |
| DB04100 | Tricarbonyl(1,10-phenanthroline)rhenium(1+) | experimental | unknown | inhibitor | Details |
| DB01411 | Pranlukast | investigational | unknown | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | inhibitor | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | inhibitor | Details |
| DB00345 | Aminohippuric acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrate | Details |
| DB00224 | Indinavir | approved | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | unknown | substrate | Details |
| DB00067 | Vasopressin | approved | unknown | substrate | Details |
| DB00795 | Sulfasalazine | approved | no | substrate | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | inhibitor | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB08907 | Canagliflozin | approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrate | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | | Details |
| DB00958 | Carboplatin | approved | unknown | substrate | Details |
| DB00526 | Oxaliplatin | approved, investigational | no | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00300 | Tenofovir disoproxil | approved, investigational | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB09272 | Eluxadoline | approved, investigational | unknown | substrate | Details |
| DB09060 | Avibactam | approved | no | substrate | Details |
| DB09374 | Indocyanine green acid form | approved, investigational | no | substrate | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB01095 | Fluvastatin | approved | no | substrate | Details |
| DB01098 | Rosuvastatin | approved | no | substrate | Details |
| DB12070 | Letermovir | approved, investigational | no | inhibitor | Details |
| DB14642 | Lypressin | approved | unknown | | Details |
| DB00177 | Valsartan | approved, investigational | unknown | substrate | Details |
| DB00207 | Azithromycin | approved | unknown | substrateinhibitor | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB00698 | Nitrofurantoin | approved, vet_approved | unknown | | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB11770 | Talinolol | investigational | unknown | substrate | Details |
| DB06813 | Pralatrexate | approved, investigational | no | substrateinhibitor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00104 | Octreotide | approved, investigational | unknown | substrateinhibitor | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB06448 | Lonafarnib | approved, investigational | no | inhibitor | Details |
| DB00798 | Gentamicin | approved, vet_approved | no | substrate | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | inhibitor | Details |
| DB16407 | Azvudine | investigational | unknown | regulator | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB08884 | Gadoxetic acid | approved | no | substrate | Details |
| DB00743 | Gadobenic acid | approved, investigational | no | substrate | Details |