| DB01782 | Pyrazolanthrone | experimental | unknown | | Details |
| DB02388 | Cyclohexyl-{4-[5-(3,4-Dichlorophenyl)-2-Piperidin-4-Yl-3-Propyl-3h-Imidazol-4-Yl]-Pyrimidin-2-Yl}Amine | experimental | unknown | | Details |
| DB03084 | Cyclopropyl-{4-[5-(3,4-Dichlorophenyl)-2-[(1-Methyl)-Piperidin]-4-Yl-3-Propyl-3h-Imidazol-4-Yl]-Pyrimidin-2-Yl}Amine | experimental | unknown | | Details |
| DB03623 | 9-(4-Hydroxyphenyl)-2,7-Phenanthroline | experimental | unknown | | Details |
| DB04395 | Phosphoaminophosphonic Acid-Adenylate Ester | experimental | unknown | | Details |
| DB06933 | N-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | experimental | unknown | | Details |
| DB07010 | N-BENZYL-4-[4-(3-CHLOROPHENYL)-1H-PYRAZOL-3-YL]-1H-PYRROLE-2-CARBOXAMIDE | experimental | unknown | | Details |
| DB07217 | N-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamide | experimental | unknown | | Details |
| DB08005 | 4-{[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino}-N-ethylpiperidine-1-carboxamide | experimental | unknown | | Details |
| DB08010 | (3Z)-1-[(6-fluoro-4H-1,3-benzodioxin-8-yl)methyl]-4-[(E)-2-phenylethenyl]-1H-indole-2,3-dione 3-oxime | experimental | unknown | | Details |
| DB08011 | (3E)-5-fluoro-1-[(6-fluoro-4H-1,3-benzodioxin-8-yl)methyl]-1H-indole-2,3-dione 3-oxime | experimental | unknown | | Details |
| DB08015 | (3Z)-1-[(6-fluoro-4H-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1H-indole-2,3-dione 3-oxime | experimental | unknown | | Details |
| DB08021 | 5-bromo-N-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | experimental | unknown | | Details |
| DB08023 | N-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-N-methylpyrimidin-2-amine | experimental | unknown | | Details |
| DB08025 | N-{2'-[(4-FLUOROPHENYL)AMINO]-4,4'-BIPYRIDIN-2-YL}-4-METHOXYCYCLOHEXANECARBOXAMIDE | experimental | unknown | | Details |
| DB08026 | 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-N-methylacetamide | experimental | unknown | | Details |
| DB08555 | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | experimental | unknown | | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB11718 | Encorafenib | approved, investigational | yes | inhibitor | Details |