| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | substrateinhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | substrateinhibitor | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB02709 | Resveratrol | investigational | no | substrateinhibitor | Details |
| DB00613 | Amodiaquine | approved, investigational | unknown | substrate | Details |
| DB00121 | Biotin | approved, investigational, nutraceutical | unknown | inducer | Details |
| DB00201 | Caffeine | approved | unknown | substrate | Details |
| DB00694 | Daunorubicin | approved | unknown | inhibitor | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | binder | Details |
| DB00997 | Doxorubicin | approved, investigational | no | inhibitorinducer | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inducer | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | inhibitor | Details |
| DB01087 | Primaquine | approved | unknown | inducer | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00277 | Theophylline | approved | unknown | substrate | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrate | Details |
| DB02342 | 2-Methoxyestradiol | investigational | unknown | | Details |
| DB06732 | beta-Naphthoflavone | experimental | unknown | | Details |
| DB07776 | Flavone | approved, experimental | unknown | | Details |
| DB01645 | Genistein | investigational | unknown | | Details |
| DB03467 | Naringenin | experimental | unknown | | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB11155 | Triclocarban | approved | unknown | inducer | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inducer | Details |
| DB01222 | Budesonide | approved | unknown | inducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | inducer | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | no | inhibitor | Details |
| DB01064 | Isoprenaline | approved, investigational | unknown | inducer | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |