| DB00563 | Methotrexate | approved | unknown | substrateinhibitor | Details |
| DB02527 | Cyclic adenosine monophosphate | experimental | unknown | substrateinhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB00975 | Dipyridamole | approved | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | inhibitor | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | inhibitor | Details |
| DB00158 | Folic acid | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | inhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | inhibitor | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | inhibitor | Details |
| DB02659 | Cholic Acid | approved | unknown | inhibitor | Details |
| DB00533 | Rofecoxib | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | inhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | inhibitor | Details |
| DB00712 | Flurbiprofen | approved, investigational | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inhibitor | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | inhibitor | Details |
| DB00352 | Tioguanine | approved | unknown | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | inhibitor | Details |
| DB01033 | Mercaptopurine | approved | unknown | substrate | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB00917 | Dinoprostone | approved | unknown | substrate | Details |
| DB00770 | Alprostadil | approved, investigational | unknown | substrate | Details |
| DB00718 | Adefovir dipivoxil | approved, investigational | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrate | Details |
| DB00198 | Oseltamivir | approved | unknown | substrate | Details |
| DB00814 | Meloxicam | approved, vet_approved | unknown | binder | Details |
| DB01327 | Cefazolin | approved | unknown | substrate | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB00300 | Tenofovir disoproxil | approved, investigational | unknown | substrate | Details |
| DB00171 | ATP | investigational, nutraceutical | unknown | | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB13146 | Fluciclovine (18F) | approved | no | substrate | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB09299 | Tenofovir alafenamide | approved | no | substrate | Details |
| DB14126 | Tenofovir | experimental, investigational | no | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB00999 | Hydrochlorothiazide | approved, vet_approved | unknown | substrate | Details |
| DB01069 | Promethazine | approved, investigational | unknown | inhibitor | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB08884 | Gadoxetic acid | approved | no | substrate | Details |