| DB00357 | Aminoglutethimide | approved, investigational | yes | inhibitor | Details |
| DB01217 | Anastrozole | approved, investigational | yes | inhibitor | Details |
| DB00990 | Exemestane | approved, investigational | yes | inhibitor | Details |
| DB01006 | Letrozole | approved, investigational | yes | antagonist | Details |
| DB00894 | Testolactone | approved, investigational | yes | inhibitor | Details |
| DB05749 | MPI-674 | investigational | unknown | | Details |
| DB01006 | Letrozole | approved, investigational | unknown | inhibitor | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB01406 | Danazol | approved | unknown | inhibitor | Details |
| DB02901 | Stanolone | illicit, investigational | unknown | substrate | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB04794 | Bifonazole | approved, investigational | unknown | inhibitor | Details |
| DB06719 | Buserelin | approved, investigational | unknown | inducer | Details |
| DB01127 | Econazole | approved | no | inhibitor | Details |
| DB00926 | Etretinate | withdrawn | unknown | inhibitor | Details |
| DB00990 | Exemestane | approved, investigational | unknown | inhibitor | Details |
| DB00358 | Mefloquine | approved, investigational | unknown | inhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | inhibitor | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | inhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | inhibitor | Details |
| DB01007 | Tioconazole | approved | unknown | inhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB02342 | 2-Methoxyestradiol | investigational | unknown | | Details |
| DB00858 | Drostanolone | illicit | unknown | inhibitor | Details |
| DB00974 | Edetic acid | approved, vet_approved | unknown | substrate | Details |
| DB00389 | Carbimazole | approved, investigational | unknown | inhibitor | Details |
| DB00856 | Chlorphenesin | approved, experimental | unknown | inducer | Details |
| DB00269 | Chlorotrianisene | investigational, withdrawn | unknown | inducer | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | inducer | Details |
| DB06423 | Endostatin | investigational | unknown | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | inducer | Details |
| DB05875 | Sar9, Met (O2)11-Substance P | investigational | unknown | inhibitor | Details |
| DB06147 | Sulfathiazole | approved, vet_approved, withdrawn | unknown | inducer | Details |
| DB00184 | Nicotine | approved | unknown | inhibitor | Details |
| DB09389 | Norgestrel | approved | unknown | inhibitor | Details |
| DB04539 | Glyphosate | experimental | unknown | | Details |
| DB00655 | Estrone | approved | unknown | | Details |
| DB03467 | Naringenin | experimental | unknown | inhibitor | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB14600 | Edetate disodium anhydrous | approved, vet_approved | unknown | modulator | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB06710 | Methyltestosterone | approved | unknown | substrateinducer | Details |
| DB04839 | Cyproterone acetate | approved, investigational | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB14598 | Edetate calcium disodium anhydrous | approved | unknown | modulator | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitor | Details |
| DB16236 | Mitapivat | approved, investigational | unknown | inhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | product of | Details |
| DB13009 | Carbendazim | investigational | no | regulator | Details |