| DB03147 | Flavin adenine dinucleotide | approved | unknown | | Details |
| DB01247 | Isocarboxazid | approved | yes | inhibitor | Details |
| DB01171 | Moclobemide | approved, investigational | yes | antagonistinhibitor | Details |
| DB00780 | Phenelzine | approved | yes | antagonist | Details |
| DB00752 | Tranylcypromine | approved, investigational | yes | inhibitor | Details |
| DB00191 | Phentermine | approved, illicit | yes | antagonist | Details |
| DB04850 | Posizolid | investigational | unknown | | Details |
| DB05205 | CX157 | investigational | unknown | | Details |
| DB00388 | Phenylephrine | approved | unknown | substrate | Details |
| DB00397 | Phenylpropanolamine | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00669 | Sumatriptan | approved, investigational | unknown | substrate | Details |
| DB00852 | Pseudoephedrine | approved | unknown | inhibitor | Details |
| DB00953 | Rizatriptan | approved | unknown | substrate | Details |
| DB01445 | Bufotenine | experimental, illicit | unknown | substrate | Details |
| DB00601 | Linezolid | approved, investigational | no | inhibitor | Details |
| DB00780 | Phenelzine | approved | unknown | substrate | Details |
| DB01171 | Moclobemide | approved, investigational | unknown | inhibitor | Details |
| DB00140 | Riboflavin | approved, investigational, nutraceutical, vet_approved | unknown | cofactor | Details |
| DB00315 | Zolmitriptan | approved, investigational | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | inducer | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB00988 | Dopamine | approved | unknown | substrate | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | no | inhibitor | Details |
| DB01104 | Sertraline | approved | unknown | substrate | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | inhibitor | Details |
| DB07641 | Decyl(dimethyl)phosphine oxide | experimental | unknown | | Details |
| DB07919 | Harmine | experimental | unknown | | Details |
| DB04017 | Clorgiline | experimental | unknown | | Details |
| DB00805 | Minaprine | approved | yes | inhibitor | Details |
| DB01626 | Pargyline | approved | unknown | inhibitor | Details |
| DB01472 | 4-Methoxyamphetamine | experimental, illicit | unknown | inhibitor | Details |
| DB01363 | Ephedra sinica root | nutraceutical | yes | inhibitor | Details |
| DB01442 | MMDA | experimental, illicit | yes | inhibitor | Details |
| DB01577 | Metamfetamine | approved, illicit, withdrawn | yes | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | inhibitor | Details |
| DB00614 | Furazolidone | experimental, vet_approved | unknown | inhibitor | Details |
| DB04832 | Zimelidine | approved, withdrawn | unknown | inhibitor | Details |
| DB04820 | Nialamide | approved, withdrawn | unknown | | Details |
| DB04821 | Nomifensine | approved, withdrawn | unknown | | Details |
| DB06774 | Capsaicin | approved | unknown | inhibitor | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | inhibitor | Details |
| DB00952 | Naratriptan | approved, investigational | unknown | substrate | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | inducer | Details |
| DB13876 | Brofaromine | experimental | unknown | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | inducer | Details |
| DB13944 | Testosterone enanthate | approved | unknown | inducer | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inducer | Details |
| DB09245 | Toloxatone | experimental | unknown | antagonist | Details |
| DB09245 | Toloxatone | experimental | yes | inhibitor | Details |
| DB09244 | Pirlindole | experimental | unknown | antagonist | Details |
| DB09244 | Pirlindole | experimental | unknown | inhibitor | Details |
| DB12329 | Eravacycline | approved, investigational | no | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | inhibitor | Details |
| DB04889 | Bicifadine | investigational | unknown | substrate | Details |
| DB04818 | Iproniazid | withdrawn | unknown | inhibitor | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | inhibitor | Details |
| DB14569 | Tedizolid | approved, investigational | no | inhibitor | Details |
| DB09042 | Tedizolid phosphate | approved | no | inhibitor | Details |
| DB14914 | Flortaucipir F-18 | approved, investigational | no | binder | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | unknown | inhibitor | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01175 | Escitalopram | approved | no | substrate | Details |
| DB00215 | Citalopram | approved | no | substrate | Details |