| DB03796 | Palmitic Acid | approved | unknown | | Details |
| DB00214 | Torasemide | approved | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | substrateinhibitor | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrateinducer | Details |
| DB00682 | Warfarin | approved | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB00912 | Repaglinide | approved, investigational | unknown | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | no | substrate | Details |
| DB01132 | Pioglitazone | approved, investigational | unknown | substrateinhibitor | Details |
| DB01198 | Zopiclone | approved | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB01261 | Sitagliptin | approved, investigational | unknown | substrate | Details |
| DB01259 | Lapatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrate | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00471 | Montelukast | approved | unknown | substrateinhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00613 | Amodiaquine | approved, investigational | unknown | substrate | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | substrateinhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitorinducer | Details |
| DB01124 | Tolbutamide | approved, investigational | unknown | substrateinhibitor | Details |
| DB01241 | Gemfibrozil | approved | unknown | inhibitor | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrateinhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | inhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00796 | Candesartan cilexetil | approved | unknown | inhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitor | Details |
| DB00764 | Mometasone | experimental | no | inhibitor | Details |
| DB00938 | Salmeterol | approved | unknown | inhibitor | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | inhibitor | Details |
| DB01039 | Fenofibrate | approved | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitorinducer | Details |
| DB00451 | Levothyroxine | approved | unknown | inhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | inhibitor | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrateinhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | inhibitor | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | inhibitor | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrateinhibitor | Details |
| DB00421 | Spironolactone | approved | unknown | inhibitor | Details |
| DB01029 | Irbesartan | approved, investigational | unknown | substrateinhibitor | Details |
| DB01181 | Ifosfamide | approved | unknown | substrateinducer | Details |
| DB01115 | Nifedipine | approved | unknown | inhibitor | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitor | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00946 | Phenprocoumon | approved, investigational | unknown | substrate | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB01201 | Rifapentine | approved, investigational | unknown | inducer | Details |
| DB00418 | Secobarbital | approved, vet_approved | unknown | inducer | Details |
| DB06210 | Eltrombopag | approved | unknown | substrateinhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | inhibitorinducer | Details |
| DB00661 | Verapamil | approved | unknown | substrateinhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB00201 | Caffeine | approved | unknown | substrate | Details |
| DB04725 | Licofelone | investigational | unknown | substrateinhibitor | Details |
| DB06739 | Seratrodast | experimental | unknown | substrate | Details |
| DB00402 | Eszopiclone | approved, investigational | unknown | substrate | Details |
| DB08607 | (5R)-5-(4-{[(2R)-6-HYDROXY-2,5,7,8-TETRAMETHYL-3,4-DIHYDRO-2H-CHROMEN-2-YL]METHOXY}BENZYL)-1,3-THIAZOLIDINE-2,4-DIONE | experimental | unknown | | Details |
| DB06772 | Cabazitaxel | approved | unknown | substrate | Details |
| DB01583 | Liotrix | approved | unknown | inhibitor | Details |
| DB00321 | Amitriptyline | approved | unknown | substrateinhibitor | Details |
| DB00381 | Amlodipine | approved | unknown | inhibitor | Details |
| DB01076 | Atorvastatin | approved | no | substrateinhibitor | Details |
| DB01393 | Bezafibrate | approved, investigational | unknown | inhibitor | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00758 | Clopidogrel | approved | no | inhibitor | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB00907 | Cocaine | approved, illicit | unknown | downregulator | Details |
| DB01394 | Colchicine | approved | unknown | inhibitor | Details |
| DB00169 | Cholecalciferol | approved, nutraceutical | unknown | inhibitor | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrateinducer | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB01218 | Halofantrine | approved | unknown | substrate | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inducer | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB01221 | Ketamine | approved, vet_approved | unknown | substrate | Details |
| DB06738 | Ketobemidone | investigational | unknown | substrate | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | inhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | substrate | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB00784 | Mefenamic acid | approved | unknown | inhibitor | Details |
| DB00814 | Meloxicam | approved, vet_approved | unknown | substrate | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00916 | Metronidazole | approved | unknown | inhibitor | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00184 | Nicotine | approved | unknown | substrate | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB00554 | Piroxicam | approved, investigational | unknown | substrate | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inducer | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00205 | Pyrimethamine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00533 | Rofecoxib | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00359 | Sulfadiazine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB06729 | Sulfaphenazole | approved | unknown | inhibitor | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | inhibitor | Details |
| DB00799 | Tazarotene | approved, investigational | unknown | substrate | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00208 | Ticlopidine | approved | unknown | inhibitor | Details |
| DB00897 | Triazolam | approved, investigational | unknown | inhibitor | Details |
| DB00347 | Trimethadione | approved | unknown | substrate | Details |
| DB13179 | Troleandomycin | approved | unknown | inhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00617 | Paramethadione | approved | unknown | substrate | Details |
| DB06589 | Pazopanib | approved | unknown | substrateinhibitor | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00836 | Loperamide | approved | unknown | substrate | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB05229 | Beraprost | investigational | unknown | substrate | Details |
| DB06510 | Muraglitazar | investigational | unknown | substrate | Details |
| DB06770 | Benzyl alcohol | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | inhibitor | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB08899 | Enzalutamide | approved | no | substrateinhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrate | Details |
| DB08911 | Trametinib | approved | unknown | inhibitor | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrateinhibitor | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | | Details |
| DB09080 | Olodaterol | approved | no | substrate | Details |
| DB09054 | Idelalisib | approved | no | inhibitor | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09280 | Lumacaftor | approved | no | inhibitorinducer | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB11362 | Selexipag | approved | no | substrate | Details |
| DB08931 | Riociguat | approved | unknown | substrate | Details |
| DB09183 | Dasabuvir | approved | no | substrate | Details |
| DB09296 | Ombitasvir | approved, investigational | no | substrate | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | substrate | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inhibitor | Details |
| DB08880 | Teriflunomide | approved | unknown | inhibitor | Details |
| DB05219 | Crisaborole | approved, investigational | no | inhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inhibitorinducer | Details |
| DB05015 | Belinostat | approved, investigational | unknown | inhibitor | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrate | Details |
| DB06670 | Odanacatib | investigational | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB08922 | Perospirone | experimental | unknown | substrate | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13919 | Candesartan | experimental | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB11901 | Apalutamide | approved, investigational | no | substrate | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitorinducer | Details |
| DB11632 | Opicapone | approved, investigational | no | inhibitor | Details |
| DB13746 | Bioallethrin | approved, experimental | no | substrate | Details |
| DB00486 | Nabilone | approved, investigational | no | substrateinhibitor | Details |
| DB11995 | Avatrombopag | approved, investigational | no | inducer | Details |
| DB00973 | Ezetimibe | approved | unknown | inhibitor | Details |
| DB14512 | Mometasone furoate | approved, investigational, vet_approved | no | inhibitor | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | inducer | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | inducer | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | inducer | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | inducer | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | inducer | Details |
| DB14568 | Ivosidenib | approved, investigational | unknown | inducer | Details |
| DB14545 | Hydrocortisone succinate | approved | unknown | inducer | Details |
| DB11979 | Elagolix | approved, investigational | no | substrate | Details |
| DB13867 | Fluticasone | approved, experimental | no | inhibitor | Details |
| DB08906 | Fluticasone furoate | approved | no | inhibitor | Details |
| DB00588 | Fluticasone propionate | approved | no | inhibitor | Details |
| DB00615 | Rifabutin | approved, investigational | no | inducer | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB01220 | Rifaximin | approved, investigational | no | inducer | Details |
| DB12781 | Balaglitazone | investigational | no | substrateinhibitor | Details |
| DB09201 | Ciglitazone | experimental | no | substrateinhibitor | Details |
| DB09198 | Lobeglitazone | experimental | no | substrateinhibitor | Details |
| DB09199 | Netoglitazone | experimental | no | substrateinhibitor | Details |
| DB09200 | Rivoglitazone | experimental, investigational | no | substrateinhibitor | Details |
| DB06616 | Bosutinib | approved | unknown | inhibitor | Details |
| DB08875 | Cabozantinib | approved, investigational | unknown | inhibitor | Details |
| DB01645 | Genistein | investigational | unknown | inhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB01072 | Atazanavir | approved, investigational | no | inhibitor | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB14055 | (S)-Warfarin | experimental, investigational | unknown | substrate | Details |
| DB09256 | Tegafur | approved, investigational | unknown | substrate | Details |
| DB00307 | Bexarotene | approved, investigational | no | inhibitor | Details |
| DB01357 | Mestranol | approved | no | substrate | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | inhibitor | Details |
| DB00908 | Quinidine | approved, investigational | no | inhibitor | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | inhibitor | Details |
| DB08881 | Vemurafenib | approved | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | no | substrate | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB11978 | Glasdegib | approved, investigational | no | substrate | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | inhibitor | Details |
| DB00465 | Ketorolac | approved | unknown | substrate | Details |
| DB12015 | Alpelisib | approved, investigational | unknown | inhibitor | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB00678 | Losartan | approved | no | inhibitor | Details |
| DB08502 | Capravirine | investigational | unknown | substrate | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrateinhibitor | Details |
| DB12808 | Trifarotene | approved, investigational | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | inducer | Details |
| DB01222 | Budesonide | approved | unknown | inducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | inducer | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | inhibitor | Details |
| DB01060 | Amoxicillin | approved, vet_approved | unknown | inhibitor | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | inhibitor | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB12612 | Ozanimod | approved, investigational | unknown | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | substrate | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | substrate | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | substrate | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | inhibitor | Details |
| DB14840 | Ripretinib | approved | no | inhibitor | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitorinducer | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrateinhibitor | Details |
| DB15935 | Lumasiran | approved, investigational | no | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | substrateinhibitor | Details |
| DB11853 | Relugolix | approved, investigational | unknown | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | unknown | substrate | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB08822 | Azilsartan medoxomil | approved, investigational | no | substrate | Details |
| DB15569 | Sotorasib | approved, investigational | unknown | inducer | Details |
| DB12471 | Ibrexafungerp | approved, investigational | unknown | inhibitor | Details |
| DB12543 | Samidorphan | approved, investigational | no | substrate | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB16165 | Finerenone | approved, investigational | unknown | substrate | Details |
| DB16703 | Belumosudil | approved, investigational | no | substrate | Details |
| DB08932 | Macitentan | approved | no | substrate | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitor | Details |
| DB05467 | Palovarotene | approved, investigational | no | substrate | Details |
| DB04847 | Roxadustat | approved, investigational | unknown | substrate | Details |
| DB16236 | Mitapivat | approved, investigational | no | substrateinducer | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB14921 | Mavacamten | approved, investigational | no | substrate | Details |
| DB12020 | Tecovirimat | approved, investigational | no | inducer | Details |
| DB00374 | Treprostinil | approved, investigational | unknown | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB16536 | Birch bark extract | approved, experimental | unknown | inhibitor | Details |
| DB09118 | Stiripentol | approved | unknown | inhibitor | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | unknown | inhibitor | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inhibitor | Details |
| DB17083 | Linzagolix | approved | no | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | substrateinducer | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | substrate | Details |
| DB17449 | Anacaulase | approved, investigational | unknown | inhibitor | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inhibitor | Details |
| DB11682 | Daprodustat | approved, investigational | no | substrateinhibitor | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB12513 | Omaveloxolone | approved, investigational | unknown | substrateinducer | Details |
| DB00862 | Vardenafil | approved | unknown | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB01194 | Brinzolamide | approved | no | substrate | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | inhibitor | Details |
| DB14924 | Ritlecitinib | approved, investigational | unknown | substrate | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB14766 | Etrasimod | approved | no | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB15114 | Vamorolone | approved, investigational | no | substrate | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inducer | Details |
| DB11679 | Fruquintinib | approved, investigational | no | substrate | Details |
| DB16200 | Iptacopan | approved, investigational | no | substrate | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | inhibitorinducer | Details |
| DB12005 | Nirogacestat | approved, investigational | no | inducer | Details |