| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrate | Details |
| DB00494 | Entacapone | approved, investigational | unknown | substrate | Details |
| DB00749 | Etodolac | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB00744 | Zileuton | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00712 | Flurbiprofen | approved, investigational | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB01283 | Lumiracoxib | approved, investigational | unknown | substrate | Details |
| DB00580 | Valdecoxib | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB06739 | Seratrodast | experimental | unknown | substrate | Details |
| DB06741 | Gavestinel | investigational | unknown | substrate | Details |
| DB06738 | Ketobemidone | investigational | unknown | substrate | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB04824 | Phenolphthalein | approved, withdrawn | unknown | | Details |
| DB04552 | Niflumic acid | experimental | unknown | | Details |
| DB06235 | Vadimezan | investigational | unknown | substrate | Details |
| DB04953 | Ezogabine | approved, investigational | unknown | substrate | Details |
| DB06204 | Tapentadol | approved | unknown | substrate | Details |
| DB06695 | Dabigatran etexilate | approved | unknown | substrate | Details |
| DB08896 | Regorafenib | approved | unknown | substrateinhibitor | Details |
| DB08907 | Canagliflozin | approved | unknown | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB00842 | Oxazepam | approved | unknown | substrate | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | substrate | Details |
| DB05016 | Ataluren | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrate | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | substrate | Details |
| DB11638 | Artenimol | approved, experimental, investigational | no | substrate | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB09285 | Morniflumate | experimental | unknown | inhibitor | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | substrate | Details |
| DB01039 | Fenofibrate | approved | no | substrate | Details |
| DB01320 | Fosphenytoin | approved, investigational | no | inhibitor | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinhibitor | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB06210 | Eltrombopag | approved | no | inhibitor | Details |
| DB00784 | Mefenamic acid | approved | no | inhibitor | Details |
| DB00861 | Diflunisal | approved, investigational | no | inhibitor | Details |
| DB04552 | Niflumic acid | experimental | no | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitor | Details |
| DB11978 | Glasdegib | approved, investigational | no | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB01241 | Gemfibrozil | approved | unknown | substrate | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | substrateinhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | substrate | Details |
| DB00935 | Oxymetazoline | approved, investigational | no | substrate | Details |
| DB15456 | Vericiguat | approved, investigational | unknown | substrate | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | substrate | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB16703 | Belumosudil | approved, investigational | no | substrateinhibitor | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | substrate | Details |
| DB04847 | Roxadustat | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | no | substrateinhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | substrateinhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | substrate | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | no | substrate | Details |
| DB12243 | Edaravone | approved, investigational | no | substrate | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | substrate | Details |
| DB06045 | Trofinetide | approved, investigational | unknown | inhibitor | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | substrate | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | inhibitor | Details |