| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB01048 | Abacavir | approved, investigational | unknown | substrate | Details |
| DB00173 | Adenine | approved, nutraceutical | unknown | inhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00678 | Losartan | approved | unknown | substrate | Details |
| DB00712 | Flurbiprofen | approved, investigational | unknown | substrateinhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00870 | Suprofen | approved, withdrawn | unknown | substrate | Details |
| DB06741 | Gavestinel | investigational | unknown | substrate | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | inhibitor | Details |
| DB06210 | Eltrombopag | approved | unknown | substrateinhibitor | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB05039 | Indacaterol | approved | unknown | substrate | Details |
| DB06510 | Muraglitazar | investigational | unknown | substrate | Details |
| DB00704 | Naltrexone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB06817 | Raltegravir | approved | unknown | substrate | Details |
| DB04953 | Ezogabine | approved, investigational | unknown | substrate | Details |
| DB01420 | Testosterone propionate | approved, investigational, vet_approved, withdrawn | unknown | inducer | Details |
| DB06589 | Pazopanib | approved | unknown | inhibitor | Details |
| DB06626 | Axitinib | approved, investigational | no | substrate | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | no | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | inhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | inhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB09101 | Elvitegravir | approved | no | substrate | Details |
| DB09183 | Dasabuvir | approved | unknown | inhibitor | Details |
| DB05015 | Belinostat | approved, investigational | unknown | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | inhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | inhibitor | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB11799 | Bictegravir | approved, investigational | unknown | substrate | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB00564 | Carbamazepine | approved, investigational | no | inducer | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB01174 | Phenobarbital | approved, investigational | no | inducer | Details |
| DB00932 | Tipranavir | approved, investigational | no | inducer | Details |
| DB00220 | Nelfinavir | approved | no | inducer | Details |
| DB00625 | Efavirenz | approved, investigational | no | inducer | Details |
| DB00906 | Tiagabine | approved, investigational | no | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | no | substrateinhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | no | substrate | Details |
| DB01136 | Carvedilol | approved, investigational | no | substrate | Details |
| DB03496 | Alvocidib | experimental, investigational | no | substrate | Details |
| DB00695 | Furosemide | approved, vet_approved | no | substrate | Details |
| DB01241 | Gemfibrozil | approved | no | substrateinhibitor | Details |
| DB01067 | Glipizide | approved, investigational | no | substrate | Details |
| DB00451 | Levothyroxine | approved | no | substrate | Details |
| DB00916 | Metronidazole | approved | no | substrate | Details |
| DB01183 | Naloxone | approved, vet_approved | no | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | no | substrate | Details |
| DB00193 | Tramadol | approved, investigational | no | substrate | Details |
| DB00495 | Zidovudine | approved | no | substrateinducer | Details |
| DB09298 | Silibinin | experimental, investigational | no | inhibitor | Details |
| DB09276 | Sodium aurothiomalate | approved, investigational | no | inhibitor | Details |
| DB00977 | Ethinylestradiol | approved | no | substrateinducer | Details |
| DB00439 | Cerivastatin | approved, withdrawn | no | substrate | Details |
| DB00947 | Fulvestrant | approved, investigational | no | substrate | Details |
| DB01009 | Ketoprofen | approved, vet_approved | no | substrate | Details |
| DB11967 | Binimetinib | approved, investigational | no | substrate | Details |
| DB01072 | Atazanavir | approved, investigational | no | inhibitor | Details |
| DB12020 | Tecovirimat | approved, investigational | unknown | substrate | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | substrate | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | substrateinhibitor | Details |
| DB14575 | Eslicarbazepine | approved | unknown | substrate | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB09119 | Eslicarbazepine acetate | approved | unknown | substrate | Details |
| DB11963 | Dacomitinib | approved, investigational | no | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | no | inhibitor | Details |
| DB00350 | Minoxidil | approved, investigational | no | substrate | Details |
| DB00279 | Liothyronine | approved, vet_approved | no | substrate | Details |
| DB00304 | Desogestrel | approved | no | inducer | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB09297 | Paritaprevir | approved, investigational | unknown | inhibitor | Details |
| DB09079 | Nintedanib | approved | unknown | substrate | Details |
| DB00455 | Loratadine | approved, investigational | unknown | | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | inhibitor | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | substrate | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB12893 | Sacituzumab govitecan | approved, investigational | no | substrate | Details |
| DB15456 | Vericiguat | approved, investigational | unknown | substrate | Details |
| DB09296 | Ombitasvir | approved, investigational | unknown | inhibitor | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | substrate | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB12016 | Ponesimod | approved, investigational | unknown | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | substrate | Details |
| DB16703 | Belumosudil | approved, investigational | no | inhibitor | Details |
| DB12597 | Asciminib | approved, investigational | no | inhibitor | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | substrate | Details |
| DB16236 | Mitapivat | approved, investigational | no | inducer | Details |
| DB09074 | Olaparib | approved | unknown | inhibitor | Details |
| DB08912 | Dabrafenib | approved, investigational | no | inhibitor | Details |
| DB15673 | Lenacapavir | approved, investigational | no | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | no | substrate | Details |
| DB12243 | Edaravone | approved, investigational | no | substrate | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | no | upregulator | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | substrateinducer | Details |
| DB12874 | Quizartinib | approved, investigational | no | inhibitor | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | substrate | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | inhibitorinducer | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inhibitor | Details |
| DB16200 | Iptacopan | approved, investigational | no | substrate | Details |