| DB00199 | Erythromycin | approved, investigational, vet_approved | no | substrateinhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | substrate | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | substrate | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00897 | Triazolam | approved, investigational | unknown | substrate | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | substrate | Details |
| DB01114 | Chlorpheniramine | approved | unknown | substrate | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | substrate | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrateinhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | substrate | Details |
| DB00528 | Lercanidipine | approved, investigational | unknown | substrate | Details |
| DB00401 | Nisoldipine | approved | unknown | substrate | Details |
| DB01054 | Nitrendipine | approved, investigational | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | substrate | Details |
| DB01238 | Aripiprazole | approved, investigational | no | substrate | Details |
| DB00490 | Buspirone | approved, investigational | unknown | substrate | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB01216 | Finasteride | approved | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB01227 | Levacetylmethadol | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrate | Details |
| DB01100 | Pimozide | approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB00468 | Quinine | approved | unknown | substrate | Details |
| DB00938 | Salmeterol | approved | unknown | substrate | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrate | Details |
| DB00877 | Sirolimus | approved, investigational | no | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrate | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB06287 | Temsirolimus | approved | unknown | substrate | Details |
| DB00656 | Trazodone | approved, investigational | unknown | substrate | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrate | Details |
| DB00962 | Zaleplon | approved, illicit, investigational | unknown | substrate | Details |
| DB01167 | Itraconazole | approved, investigational | no | inhibitor | Details |
| DB00446 | Chloramphenicol | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00705 | Delavirdine | approved | unknown | inhibitor | Details |
| DB06730 | Gestodene | investigational | unknown | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB06731 | Seproxetine | investigational | unknown | inhibitor | Details |
| DB00582 | Voriconazole | approved | unknown | substrateinhibitor | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inducer | Details |
| DB00458 | Imipramine | approved | unknown | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00588 | Fluticasone propionate | approved | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB04946 | Iloperidone | approved | unknown | substrate | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrateinhibitor | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | no | inducer | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | substrate | Details |
| DB09054 | Idelalisib | approved | no | substrateinhibitor | Details |
| DB09065 | Cobicistat | approved | no | substrate | Details |
| DB06412 | Oxymetholone | approved, illicit | no | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | no | substrateinhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inducer | Details |
| DB11574 | Elbasvir | approved | unknown | substrate | Details |
| DB12483 | Copanlisib | approved, investigational | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inducer | Details |
| DB13179 | Troleandomycin | approved | unknown | inhibitor | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | substrate | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | substrate | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | substrate | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | substrate | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | substrate | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | substrate | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | substrate | Details |
| DB13867 | Fluticasone | approved, experimental | unknown | substrate | Details |
| DB08906 | Fluticasone furoate | approved | no | substrate | Details |
| DB00916 | Metronidazole | approved | unknown | substrate | Details |
| DB00683 | Midazolam | approved, illicit | unknown | substrate | Details |
| DB00238 | Nevirapine | approved | unknown | substrate | Details |
| DB01016 | Glyburide | approved | unknown | substrate | Details |
| DB00620 | Triamcinolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB01224 | Quetiapine | approved | unknown | | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB01059 | Norfloxacin | approved | no | inhibitor | Details |
| DB16390 | Mobocertinib | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | no | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB09065 | Cobicistat | approved | yes | inhibitor | Details |
| DB12874 | Quizartinib | approved, investigational | no | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB01072 | Atazanavir | approved, investigational | no | inhibitor | Details |
| DB11679 | Fruquintinib | approved, investigational | no | substrate | Details |
| DB00648 | Mitotane | approved | unknown | inducer | Details |