| DB04348 | Taurocholic acid | approved, experimental | unknown | substrateinhibitorinducer | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB02659 | Cholic Acid | approved | unknown | substrateinhibitorinducer | Details |
| DB00669 | Sumatriptan | approved, investigational | unknown | inducer | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | inhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrateinhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | inhibitor | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB01124 | Tolbutamide | approved, investigational | unknown | inhibitor | Details |
| DB00468 | Quinine | approved | unknown | inhibitor | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | inhibitor | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | inhibitor | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB02123 | Glycochenodeoxycholic Acid | experimental | unknown | substrateinhibitor | Details |
| DB03619 | Deoxycholic acid | approved | unknown | substrateinhibitor | Details |
| DB00421 | Spironolactone | approved | unknown | inhibitor | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inhibitor | Details |
| DB04630 | Aldosterone | experimental, investigational | unknown | inhibitor | Details |
| DB00655 | Estrone | approved | unknown | inhibitor | Details |
| DB04573 | Estriol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inhibitor | Details |
| DB00860 | Prednisolone | approved, vet_approved | unknown | inhibitor | Details |
| DB01396 | Digitoxin | approved, investigational | unknown | inhibitor | Details |
| DB01092 | Ouabain | approved | unknown | substrateinhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00584 | Enalapril | approved, vet_approved | unknown | substrate | Details |
| DB00917 | Dinoprostone | approved | unknown | substrate | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | substrate | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB00728 | Rocuronium | approved | unknown | substrate | Details |
| DB00390 | Digoxin | approved | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00887 | Bumetanide | approved | unknown | substrate | Details |
| DB01583 | Liotrix | approved | unknown | substrate | Details |
| DB06710 | Methyltestosterone | approved | unknown | inhibitorinducer | Details |
| DB02691 | Glycocholic acid | experimental, investigational | unknown | | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | | Details |
| DB00451 | Levothyroxine | approved | unknown | substrate | Details |
| DB00291 | Chlorambucil | approved | unknown | | Details |
| DB08833 | Taurochenodeoxycholic acid | experimental | unknown | | Details |
| DB08834 | Tauroursodeoxycholic acid | approved, investigational | unknown | substrate | Details |
| DB08836 | Temocapril | experimental, investigational | unknown | | Details |
| DB01098 | Rosuvastatin | approved | unknown | | Details |
| DB08893 | Mirabegron | approved | unknown | substrate | Details |
| DB11611 | Lifitegrast | approved | unknown | substrate | Details |
| DB11591 | Bilastine | approved, investigational | no | substrate | Details |
| DB13943 | Testosterone cypionate | approved | unknown | inhibitorinducer | Details |
| DB13944 | Testosterone enanthate | approved | unknown | inhibitorinducer | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inhibitorinducer | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01590 | Everolimus | approved | unknown | inhibitor | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | | Details |
| DB14641 | Estriol tripropionate | experimental | unknown | | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | inhibitor | Details |
| DB15566 | Prednisolone acetate | approved, vet_approved | unknown | inhibitor | Details |
| DB01222 | Budesonide | approved | unknown | substrate | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | inhibitor | Details |
| DB00253 | Medrysone | approved | unknown | substrate | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inhibitor | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | inhibitor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | inhibitor | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrate | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB01005 | Hydroxyurea | approved | no | substrate | Details |