| DB01032 | Probenecid | approved, investigational | yes | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | inducer | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrateinhibitor | Details |
| DB00936 | Salicylic acid | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB01053 | Benzylpenicillin | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB01092 | Ouabain | approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | inhibitor | Details |
| DB01050 | Ibuprofen | approved | unknown | inhibitor | Details |
| DB00536 | Guanidine | approved | unknown | inhibitor | Details |
| DB03553 | Glutaric Acid | experimental | unknown | substrateinhibitor | Details |
| DB00695 | Furosemide | approved, vet_approved | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inhibitor | Details |
| DB02659 | Cholic Acid | approved | unknown | substrateinhibitor | Details |
| DB00887 | Bumetanide | approved | unknown | inhibitor | Details |
| DB01597 | Cilastatin | approved, investigational | unknown | inhibitor | Details |
| DB00554 | Piroxicam | approved, investigational | unknown | inhibitor | Details |
| DB00345 | Aminohippuric acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB04519 | Caprylic acid | investigational | unknown | inhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00168 | Aspartame | investigational, nutraceutical | unknown | inhibitor | Details |
| DB00759 | Tetracycline | approved, vet_approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00595 | Oxytetracycline | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01004 | Ganciclovir | approved, investigational | unknown | inhibitor | Details |
| DB00787 | Acyclovir | approved | unknown | substrateinhibitor | Details |
| DB00917 | Dinoprostone | approved | unknown | substrateinhibitor | Details |
| DB00456 | Cefalotin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01329 | Cefoperazone | approved, investigational | unknown | inhibitor | Details |
| DB01327 | Cefazolin | approved | unknown | inhibitor | Details |
| DB01326 | Cefamandole | approved, experimental | unknown | inhibitor | Details |
| DB01140 | Cefadroxil | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB01212 | Ceftriaxone | approved | unknown | inhibitor | Details |
| DB00493 | Cefotaxime | approved | unknown | inhibitor | Details |
| DB00812 | Phenylbutazone | approved, vet_approved | unknown | inhibitor | Details |
| DB01009 | Ketoprofen | approved, vet_approved | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | no | substrateinhibitor | Details |
| DB00927 | Famotidine | approved | no | substrateinhibitor | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | inhibitor | Details |
| DB00563 | Methotrexate | approved | unknown | substrateinhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrateinhibitor | Details |
| DB00469 | Tenoxicam | approved | unknown | inhibitor | Details |
| DB00584 | Enalapril | approved, vet_approved | unknown | inhibitor | Details |
| DB01650 | trans-2-hydroxycinnamic acid | experimental | unknown | inhibitor | Details |
| DB00567 | Cephalexin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB03793 | Benzoic acid | approved, investigational | unknown | inhibitor | Details |
| DB01033 | Mercaptopurine | approved | unknown | substrateinhibitor | Details |
| DB01051 | Novobiocin | approved, investigational, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00213 | Pantoprazole | approved | unknown | inhibitor | Details |
| DB00139 | Succinic acid | approved, nutraceutical | unknown | substrate | Details |
| DB02527 | Cyclic adenosine monophosphate | experimental | unknown | substrate | Details |
| DB00577 | Valaciclovir | approved, investigational | unknown | substrate | Details |
| DB03902 | Oxalic Acid | experimental | unknown | substrate | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | substrate | Details |
| DB00583 | Levocarnitine | approved, investigational | unknown | substrate | Details |
| DB00437 | Allopurinol | approved | unknown | substrate | Details |
| DB00198 | Oseltamivir | approved | unknown | substrate | Details |
| DB01583 | Liotrix | approved | unknown | inhibitor | Details |
| DB01414 | Cefacetrile | experimental, vet_approved | unknown | substrateinhibitor | Details |
| DB06710 | Methyltestosterone | approved | unknown | inducer | Details |
| DB00495 | Zidovudine | approved | unknown | substrateinhibitor | Details |
| DB08844 | Uric acid | investigational | unknown | | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | | Details |
| DB01160 | Dinoprost tromethamine | approved, vet_approved | unknown | | Details |
| DB04133 | Degraded Cephaloridine | experimental | unknown | | Details |
| DB08837 | Tetraethylammonium | experimental, investigational | unknown | | Details |
| DB06335 | Saxagliptin | approved | unknown | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | no | inhibitor | Details |
| DB00300 | Tenofovir disoproxil | approved, investigational | unknown | substrate | Details |
| DB00493 | Cefotaxime | approved | unknown | | Details |
| DB01212 | Ceftriaxone | approved | unknown | | Details |
| DB01053 | Benzylpenicillin | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB09272 | Eluxadoline | approved, investigational | unknown | substrate | Details |
| DB09060 | Avibactam | approved | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB05016 | Ataluren | approved, investigational | no | inhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | unknown | inhibitor | Details |
| DB08930 | Dolutegravir | approved | no | inhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | inducer | Details |
| DB13944 | Testosterone enanthate | approved | unknown | inducer | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inducer | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | | Details |
| DB11901 | Apalutamide | approved, investigational | no | inhibitor | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00833 | Cefaclor | approved | unknown | substrateinhibitor | Details |
| DB00535 | Cefdinir | approved | unknown | substrate | Details |
| DB00229 | Cefotiam | approved, investigational | unknown | substrateinhibitor | Details |
| DB01415 | Ceftibuten | approved, investigational | unknown | substrateinhibitor | Details |
| DB01332 | Ceftizoxime | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB09008 | Cefaloridine | experimental, withdrawn | unknown | substrateinhibitor | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrate | Details |
| DB12243 | Edaravone | approved, investigational | no | substrate | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB00650 | Leucovorin | approved | unknown | substrateinhibitor | Details |
| DB00881 | Quinapril | approved, investigational | unknown | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrateinhibitor | Details |
| DB01261 | Sitagliptin | approved, investigational | unknown | substrate | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | | Details |
| DB14568 | Ivosidenib | approved, investigational | unknown | inhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB00319 | Piperacillin | approved | unknown | substrate | Details |
| DB01606 | Tazobactam | approved | unknown | substrateinhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inhibitor | Details |
| DB11751 | Cabotegravir | approved, investigational | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB12866 | Pradigastat | investigational | unknown | inhibitor | Details |
| DB00642 | Pemetrexed | approved, investigational | no | substrate | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inhibitor | Details |
| DB06211 | Doripenem | approved, investigational | no | substrate | Details |
| DB00945 | Acetylsalicylic acid | approved, vet_approved | unknown | inhibitor | Details |
| DB00736 | Esomeprazole | approved, investigational | unknown | inhibitor | Details |
| DB09299 | Tenofovir alafenamide | approved | no | substrate | Details |
| DB14126 | Tenofovir | experimental, investigational | no | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | | Details |
| DB12377 | Relebactam | approved, investigational | unknown | substrate | Details |
| DB05154 | Pretomanid | approved | unknown | inhibitor | Details |
| DB00654 | Latanoprost | approved, investigational | unknown | inhibitor | Details |
| DB00999 | Hydrochlorothiazide | approved, vet_approved | unknown | substrate | Details |
| DB01241 | Gemfibrozil | approved | unknown | inhibitor | Details |
| DB04855 | Dronedarone | approved | unknown | inhibitor | Details |
| DB01222 | Budesonide | approved | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB11644 | Tafamidis | approved, investigational | unknown | inhibitor | Details |
| DB12457 | Rimegepant | approved, investigational | unknown | inhibitor | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | inhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB00253 | Medrysone | approved | unknown | substrate | Details |
| DB00774 | Hydroflumethiazide | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB01324 | Polythiazide | approved | unknown | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | substrate | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | inhibitor | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | substrate | Details |
| DB00601 | Linezolid | approved, investigational | no | inhibitor | Details |
| DB01147 | Cloxacillin | approved, investigational, vet_approved | no | substrateinhibitor | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | inhibitor | Details |
| DB14973 | Abrocitinib | approved, investigational | unknown | substrate | Details |
| DB04847 | Roxadustat | approved, investigational | unknown | substrate | Details |
| DB17083 | Linzagolix | approved | no | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB11682 | Daprodustat | approved, investigational | no | substrate | Details |
| DB01250 | Olsalazine | approved | unknown | upregulator | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | substrateinhibitor | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB12218 | Capivasertib | approved, investigational | no | inhibitor | Details |
| DB11995 | Avatrombopag | approved, investigational | no | inhibitor | Details |