| DB00728 | Rocuronium | approved | unknown | substrate | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB01004 | Ganciclovir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00787 | Acyclovir | approved | unknown | substrateinhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inhibitor | Details |
| DB00457 | Prazosin | approved | unknown | substrateinhibitor | Details |
| DB00925 | Phenoxybenzamine | approved | unknown | inhibitor | Details |
| DB00914 | Phenformin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00331 | Metformin | approved | unknown | substrate | Details |
| DB00152 | Thiamine | approved, investigational, nutraceutical, vet_approved | unknown | substrate | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB01035 | Procainamide | approved | unknown | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | inhibitor | Details |
| DB05381 | Histamine | approved, investigational | unknown | | Details |
| DB00988 | Dopamine | approved | unknown | substrate | Details |
| DB00406 | Gentian violet cation | approved | unknown | | Details |
| DB00122 | Choline | approved, nutraceutical | unknown | substrateinhibitor | Details |
| DB00915 | Amantadine | approved | unknown | substrateinhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitor | Details |
| DB01337 | Pancuronium | approved | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00280 | Disopyramide | approved | unknown | inhibitor | Details |
| DB01151 | Desipramine | approved, investigational | unknown | inhibitor | Details |
| DB00520 | Caspofungin | approved | unknown | | Details |
| DB00536 | Guanidine | approved | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB01114 | Chlorpheniramine | approved | unknown | inhibitor | Details |
| DB00668 | Epinephrine | approved, vet_approved | unknown | substrate | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB00206 | Reserpine | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB00368 | Norepinephrine | approved | unknown | substrate | Details |
| DB03128 | Acetylcholine | approved, investigational | unknown | substrate | Details |
| DB00127 | Spermine | experimental, nutraceutical | unknown | substrate | Details |
| DB03566 | Spermidine | experimental | unknown | substrate | Details |
| DB01199 | Tubocurarine | approved | unknown | substrate | Details |
| DB04830 | Buformin | investigational, withdrawn | unknown | substrate | Details |
| DB00413 | Pramipexole | approved, investigational | unknown | substrate | Details |
| DB01621 | Pipotiazine | approved, investigational | unknown | | Details |
| DB01623 | Thiothixene | approved | unknown | | Details |
| DB08837 | Tetraethylammonium | experimental, investigational | unknown | | Details |
| DB08838 | Agmatine | experimental | unknown | substrate | Details |
| DB00318 | Codeine | approved, illicit | unknown | substrateinhibitor | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB09555 | Dexchlorpheniramine maleate | approved | unknown | substrateinhibitor | Details |
| DB12598 | Nafamostat | investigational | unknown | substrate | Details |
| DB12267 | Brigatinib | approved, investigational | no | | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11642 | Pitolisant | approved, investigational | unknown | inhibitor | Details |
| DB14006 | Choline salicylate | approved, nutraceutical | unknown | substrateinhibitor | Details |
| DB00758 | Clopidogrel | approved | no | inhibitor | Details |
| DB00590 | Doxazosin | approved | no | inhibitor | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inhibitor | Details |
| DB00238 | Nevirapine | approved | unknown | inhibitor | Details |
| DB11963 | Dacomitinib | approved, investigational | no | inhibitor | Details |
| DB12141 | Gilteritinib | approved, investigational | no | inhibitor | Details |
| DB09073 | Palbociclib | approved, investigational | no | inhibitor | Details |
| DB08882 | Linagliptin | approved | unknown | inhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | | Details |
| DB09079 | Nintedanib | approved | unknown | substrateinhibitor | Details |
| DB04855 | Dronedarone | approved | no | inhibitor | Details |
| DB11732 | Lasmiditan | approved, investigational | no | inhibitor | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrateinhibitor | Details |
| DB01018 | Guanfacine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00938 | Salmeterol | approved | unknown | substrateinhibitor | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | substrate | Details |
| DB00434 | Cyproheptadine | approved | unknown | inhibitor | Details |
| DB06288 | Amisulpride | approved, investigational | no | substrate | Details |
| DB08893 | Mirabegron | approved | no | substrate | Details |
| DB11886 | Infigratinib | approved, investigational | no | inhibitor | Details |
| DB16098 | Atogepant | approved, investigational | no | inhibitor | Details |
| DB12597 | Asciminib | approved, investigational | no | inhibitor | Details |
| DB14973 | Abrocitinib | approved, investigational | unknown | inhibitor | Details |
| DB11697 | Pacritinib | approved, investigational | no | inhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | no | inhibitor | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB09076 | Umeclidinium | approved | no | substrate | Details |
| DB05467 | Palovarotene | approved, investigational | no | inhibitor | Details |