| DB00331 | Metformin | approved | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00567 | Cephalexin | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00877 | Sirolimus | approved, investigational | no | | Details |
| DB00787 | Acyclovir | approved | unknown | substrate | Details |
| DB08840 | N-methylnicotinamide | experimental | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | no | inhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB11799 | Bictegravir | approved, investigational | unknown | inhibitor | Details |
| DB04948 | Lofexidine | approved, investigational | no | inhibitor | Details |
| DB12615 | Plazomicin | approved, investigational | unknown | inhibitor | Details |
| DB06608 | Tafenoquine | approved, investigational | no | inhibitor | Details |
| DB01333 | Cefradine | approved | unknown | substrate | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB04574 | Estrone sulfate | approved | unknown | substrate | Details |
| DB01004 | Ganciclovir | approved, investigational | unknown | substrate | Details |
| DB08837 | Tetraethylammonium | experimental, investigational | unknown | substrate | Details |
| DB00536 | Guanidine | approved | unknown | substrate | Details |
| DB01035 | Procainamide | approved | unknown | substrate | Details |
| DB01030 | Topotecan | approved, investigational | unknown | substrateinhibitor | Details |
| DB00205 | Pyrimethamine | approved, investigational, vet_approved | no | inhibitor | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB09343 | Tipiracil | approved, investigational | unknown | substrate | Details |
| DB12141 | Gilteritinib | approved, investigational | no | inhibitor | Details |
| DB11978 | Glasdegib | approved, investigational | no | inhibitor | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inducer | Details |
| DB01043 | Memantine | approved, investigational | unknown | | Details |
| DB12377 | Relebactam | approved, investigational | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB01203 | Nadolol | approved | unknown | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | inhibitor | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB11901 | Apalutamide | approved, investigational | no | inhibitor | Details |
| DB11732 | Lasmiditan | approved, investigational | unknown | inhibitor | Details |
| DB00879 | Emtricitabine | approved, investigational | unknown | substrate | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB00927 | Famotidine | approved | no | inhibitor | Details |
| DB01018 | Guanfacine | approved, investigational | unknown | inhibitor | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | inhibitor | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00243 | Ranolazine | approved, investigational | unknown | inhibitor | Details |
| DB12457 | Rimegepant | approved, investigational | unknown | inhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | inhibitor | Details |
| DB15102 | Pemigatinib | approved, investigational | no | inhibitor | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | inhibitor | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | inhibitor | Details |
| DB14840 | Ripretinib | approved | unknown | inhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitor | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB15442 | Trilaciclib | approved, investigational | unknown | inhibitor | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | substrate | Details |
| DB16628 | Fosdenopterin | approved | unknown | substrate | Details |
| DB06288 | Amisulpride | approved, investigational | no | substrateinhibitor | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB11886 | Infigratinib | approved, investigational | no | inhibitor | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitor | Details |
| DB08930 | Dolutegravir | approved | no | inhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | inhibitor | Details |
| DB16098 | Atogepant | approved, investigational | no | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitor | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | inhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | no | inhibitor | Details |
| DB11793 | Niraparib | approved, investigational | no | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | substrate | Details |
| DB15097 | Gefapixant | approved, investigational | no | substrate | Details |
| DB12218 | Capivasertib | approved, investigational | no | inhibitor | Details |