| DB01045 | Rifampicin | approved | unknown | substrateinhibitor | Details |
| DB01132 | Pioglitazone | approved, investigational | unknown | inhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB02659 | Cholic Acid | approved | unknown | substrate | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | substrate | Details |
| DB01092 | Ouabain | approved | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00520 | Caspofungin | approved | unknown | substrate | Details |
| DB00275 | Olmesartan | approved, investigational | unknown | substrate | Details |
| DB00177 | Valsartan | approved, investigational | unknown | substrate | Details |
| DB01583 | Liotrix | approved | unknown | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | inhibitor | Details |
| DB08855 | Leukotriene C4 | experimental, investigational | unknown | | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | | Details |
| DB02691 | Glycocholic acid | experimental, investigational | unknown | | Details |
| DB05804 | Prasterone sulfate | investigational | unknown | | Details |
| DB00451 | Levothyroxine | approved | unknown | inhibitor | Details |
| DB08861 | DPDPE | experimental | unknown | | Details |
| DB08862 | Cholecystokinin | approved, investigational | unknown | substrate | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | | Details |
| DB06772 | Cabazitaxel | approved | unknown | inhibitor | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB08884 | Gadoxetic acid | approved | no | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrateinhibitor | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB00175 | Pravastatin | approved | no | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB01211 | Clarithromycin | approved | unknown | | Details |
| DB09054 | Idelalisib | approved | no | inhibitor | Details |
| DB09292 | Sacubitril | approved | unknown | inhibitor | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | inhibitor | Details |
| DB05239 | Cobimetinib | approved, investigational | no | inhibitor | Details |
| DB11362 | Selexipag | approved | no | substrate | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB11575 | Grazoprevir | approved | no | substrate | Details |
| DB09137 | Technetium Tc-99m mebrofenin | approved | no | substrate | Details |
| DB13154 | Parachlorophenol | approved | unknown | substrate | Details |
| DB13139 | Levosalbutamol | approved, investigational | no | substrate | Details |
| DB13153 | Levomenol | approved, experimental | unknown | substrate | Details |
| DB11613 | Velpatasvir | approved, investigational | no | inhibitortransporter | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB06749 | Ginsenoside Rb1 | nutraceutical | unknown | inhibitor | Details |
| DB06750 | Ginsenoside Rg1 | nutraceutical | unknown | | Details |
| DB05016 | Ataluren | approved, investigational | no | inhibitor | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrateinhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | inhibitor | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | inhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | substrateinhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | inhibitor | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | | Details |
| DB09297 | Paritaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00975 | Dipyridamole | approved | unknown | inhibitor | Details |
| DB01072 | Atazanavir | approved, investigational | unknown | inhibitor | Details |
| DB00541 | Vincristine | approved, investigational | unknown | inhibitor | Details |
| DB09142 | Sincalide | approved | no | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01149 | Nefazodone | approved, withdrawn | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB01051 | Novobiocin | approved, investigational, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00646 | Nystatin | approved, vet_approved | unknown | inhibitor | Details |
| DB11869 | Valspodar | investigational | unknown | inhibitor | Details |
| DB09298 | Silibinin | experimental, investigational | unknown | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | no | inhibitor | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | inhibitor | Details |
| DB09065 | Cobicistat | approved | unknown | inhibitor | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01601 | Lopinavir | approved | unknown | inhibitor | Details |
| DB00976 | Telithromycin | approved | unknown | inhibitor | Details |
| DB01590 | Everolimus | approved | unknown | inhibitor | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB11855 | Revefenacin | approved, investigational | no | substrate | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | no | inhibitor | Details |
| DB00834 | Mifepristone | approved, investigational | no | inhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inducer | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inducer | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB09299 | Tenofovir alafenamide | approved | no | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB11942 | Selinexor | approved, investigational | unknown | inhibitor | Details |
| DB00394 | Beclomethasone dipropionate | approved, investigational | unknown | inhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | inhibitor | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB01241 | Gemfibrozil | approved | unknown | inhibitor | Details |
| DB04855 | Dronedarone | approved | no | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | unknown | substrate | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | substrateinhibitor | Details |
| DB01211 | Clarithromycin | approved | unknown | inhibitor | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | inhibitor | Details |
| DB12457 | Rimegepant | approved, investigational | unknown | inhibitor | Details |
| DB11936 | Bempedoic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitor | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | inhibitor | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB00188 | Bortezomib | approved, investigational | no | inhibitor | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | inhibitor | Details |
| DB11796 | Fostemsavir | approved, investigational | unknown | inhibitor | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB11632 | Opicapone | approved, investigational | no | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB08995 | Diosmin | approved, investigational | unknown | | Details |
| DB11886 | Infigratinib | approved, investigational | no | inhibitor | Details |
| DB12471 | Ibrexafungerp | approved, investigational | unknown | inhibitor | Details |
| DB12151 | Brincidofovir | approved, investigational | no | substrate | Details |
| DB15463 | Belzutifan | approved, investigational | no | substrate | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | inhibitor | Details |
| DB16098 | Atogepant | approved, investigational | no | substrateinhibitor | Details |
| DB12597 | Asciminib | approved, investigational | no | inhibitor | Details |
| DB15413 | Pafolacianine | approved, investigational | no | substrate | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | inhibitor | Details |
| DB15575 | Padeliporfin | approved, experimental | unknown | inhibitor | Details |
| DB06813 | Pralatrexate | approved, investigational | no | substrate | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | inhibitor | Details |
| DB17083 | Linzagolix | approved | unknown | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB00244 | Mesalazine | approved | no | substrate | Details |
| DB11682 | Daprodustat | approved, investigational | no | inhibitor | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | inhibitor | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | substrate | Details |
| DB06045 | Trofinetide | approved, investigational | unknown | inhibitor | Details |
| DB16217 | Leniolisib | approved, investigational | no | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB01005 | Hydroxyurea | approved | unknown | | Details |
| DB05467 | Palovarotene | approved, investigational | no | inhibitor | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB12218 | Capivasertib | approved, investigational | no | inhibitor | Details |