| DB00796 | Candesartan cilexetil | approved | unknown | substrate | Details |
| DB01029 | Irbesartan | approved, investigational | unknown | substrate | Details |
| DB00678 | Losartan | approved | unknown | substrate | Details |
| DB00749 | Etodolac | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00712 | Flurbiprofen | approved, investigational | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB00327 | Hydromorphone | approved, illicit | no | substrate | Details |
| DB01252 | Mitiglinide | investigational | unknown | substrate | Details |
| DB04725 | Licofelone | investigational | unknown | substrate | Details |
| DB06741 | Gavestinel | investigational | unknown | substrate | Details |
| DB06210 | Eltrombopag | approved | unknown | substrate | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB06510 | Muraglitazar | investigational | unknown | substrate | Details |
| DB00434 | Cyproheptadine | approved | unknown | substrate | Details |
| DB04953 | Ezogabine | approved, investigational | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | inhibitor | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB11691 | Naldemedine | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrate | Details |
| DB13919 | Candesartan | experimental | unknown | substrate | Details |
| DB12070 | Letermovir | approved, investigational | no | substrate | Details |
| DB06230 | Nalmefene | approved, investigational, withdrawn | no | substrate | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | no | substrate | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | substrate | Details |
| DB01241 | Gemfibrozil | approved | unknown | substrateinhibitor | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00455 | Loratadine | approved, investigational | unknown | | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | | Details |
| DB11689 | Selumetinib | approved, investigational | no | | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB00920 | Ketotifen | approved | unknown | substrate | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB08893 | Mirabegron | approved | no | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | substrate | Details |
| DB12020 | Tecovirimat | approved, investigational | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | no | substrate | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | substrate | Details |
| DB15114 | Vamorolone | approved, investigational | no | substrate | Details |
| DB16200 | Iptacopan | approved, investigational | no | substrate | Details |