| DB00678 | Losartan | approved | unknown | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00749 | Etodolac | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00712 | Flurbiprofen | approved, investigational | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB01252 | Mitiglinide | investigational | unknown | substrate | Details |
| DB06737 | Zaltoprofen | experimental | unknown | substrate | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | inhibitor | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB06777 | Chenodeoxycholic acid | approved | unknown | inhibitor | Details |
| DB06235 | Vadimezan | investigational | unknown | substrate | Details |
| DB00445 | Epirubicin | approved | unknown | substrate | Details |
| DB06204 | Tapentadol | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB06695 | Dabigatran etexilate | approved | unknown | substrate | Details |
| DB06207 | Silodosin | approved | unknown | substrate | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB00842 | Oxazepam | approved | unknown | substrate | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrate | Details |
| DB00318 | Codeine | approved, illicit | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrate | Details |
| DB06230 | Nalmefene | approved, investigational, withdrawn | no | substrate | Details |
| DB13783 | Acemetacin | approved, investigational | no | substrate | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | substrate | Details |
| DB11638 | Artenimol | approved, experimental, investigational | no | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB00465 | Ketorolac | approved | unknown | substrate | Details |
| DB00327 | Hydromorphone | approved, illicit | no | substrate | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB01241 | Gemfibrozil | approved | unknown | substrate | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrate | Details |
| DB09212 | Loxoprofen | approved | unknown | substrate | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrate | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB01006 | Letrozole | approved, investigational | unknown | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | inhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | substrate | Details |
| DB11936 | Bempedoic acid | approved, investigational | unknown | substrate | Details |
| DB00870 | Suprofen | approved, withdrawn | unknown | substrate | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | substrate | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB00784 | Mefenamic acid | approved | unknown | inhibitor | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB12016 | Ponesimod | approved, investigational | unknown | substrate | Details |
| DB08893 | Mirabegron | approved | no | substrate | Details |
| DB12235 | Estetrol | approved, investigational | unknown | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | substrate | Details |
| DB12597 | Asciminib | approved, investigational | no | substrate | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | no | substrateinhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | substrateinducer | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitorinducer | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inducer | Details |
| DB05239 | Cobimetinib | approved, investigational | no | substrate | Details |
| DB12243 | Edaravone | approved, investigational | no | substrate | Details |
| DB00683 | Midazolam | approved, illicit | no | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB06045 | Trofinetide | approved, investigational | unknown | inhibitor | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | substrate | Details |
| DB15114 | Vamorolone | approved, investigational | no | substrate | Details |
| DB12218 | Capivasertib | approved, investigational | no | substrate | Details |