| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB00861 | Diflunisal | approved, investigational | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB06230 | Nalmefene | approved, investigational, withdrawn | no | substrate | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB06401 | Bazedoxifene | approved, investigational | unknown | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | no | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB09079 | Nintedanib | approved | unknown | substrate | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB09038 | Empagliflozin | approved | unknown | substrate | Details |
| DB08893 | Mirabegron | approved | no | substrate | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | substrateinhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB12243 | Edaravone | approved, investigational | no | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | substrate | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | substrate | Details |
| DB16200 | Iptacopan | approved, investigational | no | substrate | Details |