| DB00787 | Acyclovir | approved | unknown | substrate | Details |
| DB08840 | N-methylnicotinamide | experimental | unknown | substrate | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | inhibitor | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | unknown | inhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11901 | Apalutamide | approved, investigational | no | inhibitor | Details |
| DB12615 | Plazomicin | approved, investigational | unknown | inhibitor | Details |
| DB06608 | Tafenoquine | approved, investigational | no | inhibitor | Details |
| DB01137 | Levofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB04574 | Estrone sulfate | approved | unknown | substrate | Details |
| DB01004 | Ganciclovir | approved, investigational | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00331 | Metformin | approved | unknown | substrate | Details |
| DB01035 | Procainamide | approved | unknown | substrate | Details |
| DB01030 | Topotecan | approved, investigational | unknown | substrate | Details |
| DB00536 | Guanidine | approved | unknown | | Details |
| DB00205 | Pyrimethamine | approved, investigational, vet_approved | no | inhibitor | Details |
| DB11978 | Glasdegib | approved, investigational | no | inhibitor | Details |
| DB12377 | Relebactam | approved, investigational | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB01203 | Nadolol | approved | unknown | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | inhibitor | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB11732 | Lasmiditan | approved, investigational | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | unknown | substrate | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | inhibitor | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00243 | Ranolazine | approved, investigational | unknown | inhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | inhibitor | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | inhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB15442 | Trilaciclib | approved, investigational | unknown | inhibitor | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | substrate | Details |
| DB16628 | Fosdenopterin | approved | unknown | inhibitor | Details |
| DB06288 | Amisulpride | approved, investigational | no | substrateinhibitor | Details |
| DB11886 | Infigratinib | approved, investigational | no | inhibitor | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitor | Details |
| DB15463 | Belzutifan | approved, investigational | no | inhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | inhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | no | inhibitor | Details |
| DB11793 | Niraparib | approved, investigational | no | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | inhibitor | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | | Details |
| DB09128 | Brexpiprazole | approved, investigational | no | inhibitor | Details |
| DB15097 | Gefapixant | approved, investigational | unknown | substrate | Details |
| DB12218 | Capivasertib | approved, investigational | no | inhibitor | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inhibitor | Details |