| DB01189 | Desflurane | approved | yes | positive allosteric modulator | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | yes | positive allosteric modulator | Details |
| DB00237 | Butabarbital | approved, illicit | yes | positive allosteric modulator | Details |
| DB00475 | Chlordiazepoxide | approved, illicit, investigational | yes | positive allosteric modulator | Details |
| DB00349 | Clobazam | approved, illicit | yes | positive allosteric modulator | Details |
| DB01068 | Clonazepam | approved, illicit | yes | positive allosteric modulator | Details |
| DB00628 | Clorazepic acid | approved, illicit | yes | positive allosteric modulator | Details |
| DB00186 | Lorazepam | approved | yes | positive allosteric modulator | Details |
| DB00189 | Ethchlorvynol | approved, illicit, withdrawn | yes | positive allosteric modulator | Details |
| DB00228 | Enflurane | approved, investigational, vet_approved | yes | potentiator | Details |
| DB00231 | Temazepam | approved, investigational | yes | positive allosteric modulator | Details |
| DB00241 | Butalbital | approved, illicit | yes | positive allosteric modulator | Details |
| DB00292 | Etomidate | approved | yes | positive allosteric modulator | Details |
| DB00306 | Talbutal | approved, illicit | yes | positive allosteric modulator | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | yes | positive allosteric modulator | Details |
| DB00371 | Meprobamate | approved, illicit | yes | positive allosteric modulator | Details |
| DB00402 | Eszopiclone | approved, investigational | yes | positive allosteric modulator | Details |
| DB00463 | Metharbital | withdrawn | yes | positive allosteric modulator | Details |
| DB00753 | Isoflurane | approved, vet_approved | yes | positive allosteric modulator | Details |
| DB00794 | Primidone | approved, vet_approved | yes | positive allosteric modulator | Details |
| DB00801 | Halazepam | approved, illicit, withdrawn | yes | positive allosteric modulator | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | yes | positive allosteric modulator | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | yes | positive allosteric modulator | Details |
| DB00842 | Oxazepam | approved | yes | positive allosteric modulator | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | yes | positive allosteric modulator | Details |
| DB01107 | Methyprylon | approved, illicit, withdrawn | yes | positive allosteric modulator | Details |
| DB01159 | Halothane | approved, vet_approved | yes | positive allosteric modulator | Details |
| DB01205 | Flumazenil | approved | yes | positive allosteric modulator | Details |
| DB01215 | Estazolam | approved, illicit | yes | positive allosteric modulator | Details |
| DB01236 | Sevoflurane | approved, vet_approved | yes | agonist | Details |
| DB01437 | Glutethimide | approved, illicit | yes | positive allosteric modulator | Details |
| DB01588 | Prazepam | approved, illicit | yes | positive allosteric modulator | Details |
| DB01589 | Quazepam | approved, illicit | yes | positive allosteric modulator | Details |
| DB00543 | Amoxapine | approved | unknown | binder | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | antagonist | Details |
| DB11582 | Thiocolchicoside | experimental | yes | antagonist | Details |
| DB09118 | Stiripentol | approved | yes | agonistpositive allosteric modulator | Details |
| DB01956 | Taurine | approved, nutraceutical | yes | agonist | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | antagonistinducer | Details |
| DB11901 | Apalutamide | approved, investigational | no | antagonist | Details |
| DB11859 | Brexanolone | approved, investigational | yes | positive allosteric modulator | Details |
| DB01043 | Memantine | approved, investigational | unknown | binder | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | inhibitor | Details |
| DB00252 | Phenytoin | approved, vet_approved | unknown | | Details |
| DB00683 | Midazolam | approved, illicit | yes | positive allosteric modulator | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | yes | positive allosteric modulator | Details |
| DB00897 | Triazolam | approved, investigational | yes | positive allosteric modulator | Details |
| DB01558 | Bromazepam | approved, illicit, investigational | yes | positive allosteric modulator | Details |
| DB01595 | Nitrazepam | approved | yes | positive allosteric modulator | Details |
| DB01489 | Camazepam | experimental, illicit | yes | positive allosteric modulator | Details |
| DB01511 | Delorazepam | experimental, illicit | yes | positive allosteric modulator | Details |
| DB01544 | Flunitrazepam | approved, illicit | yes | positive allosteric modulator | Details |
| DB09166 | Etizolam | experimental | yes | positive allosteric modulator | Details |
| DB13437 | Medazepam | experimental | yes | positive allosteric modulator | Details |
| DB13837 | Doxefazepam | experimental | yes | positive allosteric modulator | Details |
| DB13872 | Lormetazepam | approved | yes | positive allosteric modulator | Details |
| DB14028 | Nordazepam | experimental | yes | positive allosteric modulator | Details |
| DB00546 | Adinazolam | experimental | yes | positive allosteric modulator | Details |
| DB01545 | Ethyl loflazepate | experimental, illicit | yes | positive allosteric modulator | Details |
| DB01553 | Cloxazolam | experimental | yes | positive allosteric modulator | Details |
| DB01559 | Clotiazepam | approved, illicit | yes | positive allosteric modulator | Details |
| DB01587 | Ketazolam | approved | yes | positive allosteric modulator | Details |
| DB01594 | Cinolazepam | experimental | yes | positive allosteric modulator | Details |
| DB09017 | Brotizolam | investigational, withdrawn | yes | positive allosteric modulator | Details |
| DB13335 | Pinazepam | experimental | yes | positive allosteric modulator | Details |
| DB13643 | Loprazolam | experimental | yes | positive allosteric modulator | Details |
| DB14672 | Oxazepam acetate | experimental | yes | positive allosteric modulator | Details |
| DB12537 | 1,2-Benzodiazepine | approved, investigational | unknown | positive allosteric modulator | Details |
| DB14715 | Cinazepam | experimental | yes | positive allosteric modulator | Details |
| DB14719 | Bentazepam | experimental | yes | positive allosteric modulator | Details |
| DB15489 | Mexazolam | experimental | yes | positive allosteric modulator | Details |
| DB12404 | Remimazolam | approved, investigational | yes | positive allosteric modulator | Details |
| DB05087 | Ganaxolone | approved, investigational | yes | positive allosteric modulator | Details |
| DB15490 | Zuranolone | approved, experimental | yes | positive allosteric modulator | Details |