| DB00176 | Fluvoxamine | approved, investigational | unknown | inhibitor | Details |
| DB00599 | Thiopental | approved, vet_approved | unknown | substrate | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB13174 | Rhein | experimental | unknown | inhibitor | Details |
| DB11994 | Diacerein | approved, investigational | unknown | inhibitor | Details |
| DB11605 | Myrrh | approved | unknown | inducer | Details |
| DB11691 | Naldemedine | approved, investigational | no | substrate | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | inhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB09205 | Moxisylyte | approved, investigational | no | substrate | Details |
| DB09568 | Omega-3-carboxylic acids | approved, investigational | no | substrate | Details |
| DB01601 | Lopinavir | approved | no | inhibitor | Details |
| DB01149 | Nefazodone | approved, withdrawn | no | inhibitor | Details |
| DB13141 | Ambroxol acefyllinate | experimental, investigational | no | substrate | Details |
| DB11792 | Mirodenafil | investigational | unknown | substrate | Details |
| DB11979 | Elagolix | approved, investigational | no | substrate | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11703 | Acalabrutinib | approved, investigational | unknown | substrate | Details |
| DB12267 | Brigatinib | approved, investigational | unknown | inducer | Details |
| DB12307 | Foretinib | investigational | unknown | substrate | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB00593 | Ethosuximide | approved | unknown | substrate | Details |
| DB01201 | Rifapentine | approved, investigational | unknown | inducer | Details |
| DB00643 | Mebendazole | approved, vet_approved | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | inhibitor | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | inhibitor | Details |
| DB09212 | Loxoprofen | approved | unknown | substrate | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB01222 | Budesonide | approved | unknown | substrateinducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB11951 | Lemborexant | approved, investigational | unknown | inhibitorinducer | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB11652 | Tucatinib | approved, investigational | unknown | substrate | Details |
| DB15035 | Zanubrutinib | approved, investigational | unknown | substrate | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | inhibitor | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | inhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | inhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrateinhibitor | Details |
| DB11853 | Relugolix | approved, investigational | unknown | substrateinducer | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | inducer | Details |
| DB11742 | Ebastine | approved, investigational | unknown | substrate | Details |
| DB15569 | Sotorasib | approved, investigational | unknown | substrate | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB00647 | Dextropropoxyphene | approved, illicit, investigational, withdrawn | unknown | inhibitor | Details |
| DB00333 | Methadone | approved | no | inhibitor | Details |
| DB01167 | Itraconazole | approved, investigational | no | inhibitor | Details |
| DB16536 | Birch bark extract | approved, experimental | unknown | inhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | substrateinhibitor | Details |