| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | binder | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | yes | binder | Details |
| DB09262 | Imidafenacin | investigational | no | substrate | Details |
| DB11828 | Neratinib | approved, investigational | no | substrate | Details |
| DB00512 | Vancomycin | approved | no | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | binder | Details |
| DB09053 | Ibrutinib | approved | no | substrate | Details |
| DB11641 | Vinflunine | approved, investigational | no | substrate | Details |
| DB14582 | Patisiran | approved, investigational | unknown | ligand | Details |
| DB00289 | Atomoxetine | approved | no | binder | Details |
| DB00332 | Ipratropium | approved, experimental | no | binder | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | binder | Details |
| DB00421 | Spironolactone | approved | unknown | binder | Details |
| DB00476 | Duloxetine | approved | unknown | ligand | Details |
| DB00497 | Oxycodone | approved, illicit, investigational | unknown | binder | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | binder | Details |
| DB01029 | Irbesartan | approved, investigational | unknown | binder | Details |
| DB01591 | Solifenacin | approved | unknown | binder | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB01203 | Nadolol | approved | unknown | binder | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | binder | Details |
| DB01045 | Rifampicin | approved | unknown | ligand | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | binder | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | binder | Details |
| DB00278 | Argatroban | approved, investigational | unknown | binder | Details |
| DB06216 | Asenapine | approved | unknown | binder | Details |
| DB01072 | Atazanavir | approved, investigational | no | binder | Details |
| DB11703 | Acalabrutinib | approved, investigational | unknown | binder | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | binder | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB01115 | Nifedipine | approved | unknown | binder | Details |
| DB00938 | Salmeterol | approved | unknown | binder | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | binder | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | carrier | Details |
| DB00907 | Cocaine | approved, illicit | unknown | binder | Details |
| DB11689 | Selumetinib | approved, investigational | unknown | carrier | Details |
| DB14840 | Ripretinib | approved | unknown | binder | Details |
| DB00808 | Indapamide | approved | unknown | binder | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | binder | Details |
| DB00960 | Pindolol | approved, investigational | unknown | binder | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | binder | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | binder | Details |
| DB08932 | Macitentan | approved | no | binder | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | binderregulator | Details |
| DB00748 | Carbinoxamine | approved | unknown | binderregulator | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | binder | Details |
| DB08930 | Dolutegravir | approved | no | binder | Details |
| DB12147 | Erdafitinib | approved, investigational | no | binder | Details |
| DB11978 | Glasdegib | approved, investigational | no | binder | Details |
| DB12005 | Nirogacestat | approved, investigational | no | binder | Details |