Accession Number

Peptides composed of between two and twelve amino acids.

DrugDrug Description
LeuprolideA peptide-based GnRH receptor superagonist used for the palliative treatment of prostate cancer, uterine leiomyomata, endometriosis, and central precocious puberty.
GoserelinA synthetic analog of luteinizing hormone-releasing hormone used to treat breast cancer and prostate cancer by reducing secretion of gonadotropins from the pituitary.
DesmopressinA synthetic analog of vasopressin used to reduce renal excretion of water in central diabetes insipidus and nocturia.
CetrorelixA synthetic peptide antagonist of gonadotropin releasing hormone used to prevent luteinizing hormone surges in women undergoing assisted reproduction therapy.
VasopressinA peptide hormone used to increase blood pressure in patients with vasodilatory shock who are resistant to fluid and catecholamine therapy.
GlutathioneFor nutritional supplementation, also for treating dietary shortage or imbalance
PentagastrinA gastrin-like molecule used as a diagnostic aid for the evaluation of gastric acid secretory function, gastric hypersecretion, and Zollinger-Ellison tumors.
CeruletideCaerulein is used in the treatment of paralytic ileus and as diagnostic aid in pancreatic malfunction.
EnalaprilA prodrug of an ACE inhibitor used to treat hypertension and congestive heart failure.
GonadorelinA synthetic GnRH used to test the function of gonadotropes and the pituitary.
NafarelinA gonadotropin releasing hormone agonist used to treat central precocious puberty.
LisinoprilAn ACE inhibitor used to treat hypertension, heart failure, and acute myocardial infarction.
SpiraprilSpirapril is an ACE inhibitor class drug used to treat hypertension.
BuserelinA LHRH agonist used for the palliative treatment of hormone-dependent advanced carcinoma of the prostate gland in males and treatment of endometriosis in females.
GanirelixA GnRH antagonist used in assisted reproduction in women undergoing controlled ovarian hyperstimulation to control ovulation by inhibiting the premature LH surges.
HistrelinA GnRH agonist found in subcutaneous implants used for the treatment of pediatric patients with central precocious puberty and the palliative treatment of advanced prostate cancer.
TriptorelinA GnRH agonist indicated for the palliative treatment of advanced prostate cancer.
ProtirelinA synthetic analogue of thyrotropin-releasing hormone that has been used during diagnostic tests to evaluate function of the thyroid gland.
EnalaprilatAn antihypertensive agent used for the management of hypertension when oral therapy is not practical.
DeslorelinDeslorelin acetate is an injectable gonadotropin releasing hormone super-agonist also known as an LHRH agonist. It stops the production of sex hormones.
Angiotensin IIA peptide hormone of the RAAS system used to raise blood pressure in septic or other forms of shock.
LypressinNot Annotated
Glutathione disulfideAn ingredient of ophthalmic irrigation solutions used during ophthalmological procedures.
AntipainAntipain is a serine/cysteine protease inhibitor originally isolated from various strains of actinomycetes. Early studies investigated the potential for antipain to alter DNA damage and chromosomal aberrations in irradiated cells...
OrnithineAn amino acid commonly found as a component in total parenteral nutrition.
AtazanavirAn antiviral protease inhibitor used in combination with other antiretrovirals for the treatment of HIV.
Angiotensin 1-7TXA127 has been investigated for the treatment of Miscellaneous Peripheral Blood Cell Abnormalities.
BradykininBradykinin has been investigated for the basic science and treatment of Hypertension and Diabetes Type 2.
AclerastideAclerastide has been investigated for the treatment of Diabetic Foot, Diabetic Foot Ulcers, and Foot Ulcer, Diabetic.
AngiotensinamideNot Annotated
FelypressinFor use as an alternative to adrenaline as a localising agent, provided that local ischaemia is not essential.
AspartameUsed as a diet supplement and sugar substitute.
IlomastatIlomastat is a broad-spectrum matrix metalloproteinase inhibitor.
N-(1-carboxy-3-phenylpropyl)phenylalanyl-alpha-asparagineNot Available
S-(2,4-dinitrophenyl)glutathioneNot Available
TerlipressinA drug used to treat bleeding caused by esophageal varices.
JE-2147Not Available
N-(3-Propylcarbamoyloxirane-2-Carbonyl)-Isoleucyl-ProlineNot Available
S-octylglutathioneNot Available
GlutathionylspermidineNot Available
EnalkirenNot Available
gamma-GlutamylcysteineNot Available
TrypanothioneNot Available
Z-Pro-ProlinalNot Available
S-benzylglutathioneNot Available
S-(4-nitrobenzyl)glutathioneNot Available
S-(N-hydroxy-N-bromophenylcarbamoyl)glutathioneNot Available
S-HexylglutathioneNot Available
S-Methyl glutathioneNot Available
OlcegepantFor the treatment of migraine headaches.
CanfosfamideIntended for the treatment of various forms of cancer.
NOV-002Investigated for use/treatment in breast cancer, lung cancer, and ovarian cancer.
EzatiostatInvestigated for use/treatment in myelodysplastic syndrome.
GolotimodInvestigated for use/treatment in hepatitis (viral, C), infectious and parasitic disease (unspecified), and tuberculosis.
VX-765Investigated for use/treatment in inflammatory disorders (unspecified) and psoriasis and psoriatic disorders.
FlovagatranInvestigated for use/treatment in thrombosis.
OglufanideInvestigated for use/treatment in hepatitis (viral, C).
Sar9, Met (O2)11-Substance PInvestigated for use/treatment in acute respiratory distress syndrome (ARDS) and viral infection.
DarinaparsinInvestigated for use/treatment in blood (blood forming organ disorders, unspecified), cancer/tumors (unspecified), solid tumors, multiple myeloma, and liver cancer.
TalabostatInvestigated for use/treatment in lymphoma (non-hodgkin's), leukemia (lymphoid), lung cancer, melanoma, and pancreatic cancer.
IcatibantA bradykinin B2 receptor antagonist used to treat acute episodes of swelling and inflammation associated with hereditary angioedema (HAE).
SaxagliptinAn DPP-4 inhibitor used for the management of type 2 diabetes mellitus.
LabradimilInvestigated for use/treatment in brain cancer and pediatric indications.
SaralasinNot Annotated
acetylleucyl-leucyl-norleucinalNot Available
KelatorphanNot Available
Brentuximab vedotinA CD30-directed antibody-drug conjugate used to treat various types of lymphoma.
PolaprezincPeptic ulcer disease, dyspepsia .
CarnosineCarnosine has been investigated for the treatment of Gulf War Illness.
BirinapantBirinapant has been investigated for the treatment of Myelodysplastic Syndrome (MDS) and Chronic Myelomonocytic Leukemia (CMML).
DanegaptideDanegaptide has been investigated for the treatment of Focus of Study is STEMI.
Alanyl glutamineA dipeptide consisting of alanine and glutamine used for supplementation.
IbodutantIbodutant has been used in trials studying the treatment of Irritable Bowel Syndrome and Irritable Bowel Syndrome With Diarrhea.
ElobixibatElobixibat has been used in trials studying the treatment and basic science of Dyslipidemia, Constipation, Chronic Constipation, Functional Constipation, and Chronic Idiopathic Constipation.
SelepressinSelepressin has been used in trials studying the treatment of Septic Shock.
Zoptarelin doxorubicinZoptarelin doxorubicin has been used in trials studying the treatment of Breast Cancer, Ovarian Cancer, Prostate Cancer, Endometrial Cancer, and Urothelial Carcinoma, among others.
CMX-2043CMX-2043 has been used in trials studying the treatment and prevention of Non STEMI, Unstable Angina, Stable Coronary Artery Disease, and Percutaneous Coronary Intervention.
Neladenoson bialanateNeladenoson bialanate has been investigated for the treatment of Heart Failure.
Arginine glutamateTwo amino acids indicated in the treatment of hyperammonemia and in combination for total parenteral nutrition.
OrnipressinNot Annotated
Aspartyl-alanyl-diketopiperazineAspartyl-alanyl-diketopiperazine is under investigation in clinical trial NCT03349645 (An Open Label Extension Study to Assess the Safety of Long-Term Treatment With Ampion for Severe OA of the Knee).
VM4-037VM4-037 is under investigation in clinical trial NCT00884520 (An Exploratory, Open Label, Multi-Center, Non-Randomized Study of [F-18]VM4-037).
GlycylglutamineAn ingredient in amino acid solutions for parenteral nutrition.
GlycyltyrosineAn ingredient in amino acid solutions for parenteral nutrition.
LeupeptinNot Annotated
CA-074 methyl esterCA-074 methyl ester (CA-074Me) is a cell-permeable cathepsin B inhibitor. It is converted by cellular esterases to CA-074.[A258234,A258239]
S-NitrosoglutathioneNot Annotated
Drugs & Drug Targets
LeuprolideGonadotropin-releasing hormone receptortarget
GoserelinLutropin-choriogonadotropic hormone receptortarget
GoserelinGonadotropin-releasing hormone receptortarget
DesmopressinVasopressin V1a receptortarget
DesmopressinVasopressin V1b receptortarget
DesmopressinVasopressin V2 receptortarget
DesmopressinProstaglandin G/H synthase 1enzyme
DesmopressinProstaglandin G/H synthase 2enzyme
CetrorelixLutropin-choriogonadotropic hormone receptortarget
CetrorelixGonadotropin-releasing hormone receptortarget
VasopressinVasopressin V1a receptortarget
VasopressinVasopressin V2 receptortarget
VasopressinVasopressin V1b receptortarget
VasopressinCanalicular multispecific organic anion transporter 1transporter
VasopressinOxytocin receptortarget
GlutathioneGlutathione reductase, mitochondrialtarget
GlutathioneGlutathione synthetasetarget
GlutathioneGlutathione S-transferase Mu 1target
GlutathioneGlutathione S-transferase kappa 1target
GlutathioneGlutathione S-transferase A3target
GlutathioneGlutathione S-transferase Mu 3target
GlutathioneGlutathione S-transferase A4target
GlutathioneGlutathione S-transferase Mu 4target
GlutathioneGlutathione S-transferase A5target
GlutathioneGlutathione S-transferase Ptarget
GlutathioneGlutathione S-transferase omega-1target
GlutathioneGlutathione peroxidase 1target
GlutathioneGlutathione peroxidase 2target
GlutathioneGlutathione S-transferase theta-1target
GlutathioneMaleylacetoacetate isomerasetarget
GlutathioneEpididymal secretory glutathione peroxidasetarget
GlutathioneGlutathione peroxidase 3target
GlutathioneLactoylglutathione lyasetarget
GlutathioneLeukotriene C4 synthasetarget
GlutathioneMicrosomal glutathione S-transferase 3target
GlutathioneHematopoietic prostaglandin D synthasetarget
GlutathioneGlutathione S-transferase A1target
GlutathioneGlutathione S-transferase A2target
GlutathioneMicrosomal glutathione S-transferase 1target
GlutathioneS-formylglutathione hydrolasetarget
GlutathioneGamma-glutamyltranspeptidase 1target
GlutathioneGlutathione S-transferase Mu 2target
GlutathionePhospholipid hydroperoxide glutathione peroxidase, mitochondrialtarget
GlutathioneGlutathione S-transferase Mu 5target
GlutathioneGlutathione peroxidase 6target
GlutathioneHydroxyacylglutathione hydrolase, mitochondrialtarget
GlutathioneGlutathione peroxidasetarget
GlutathioneGlutathione peroxidase 7target
GlutathioneMicrosomal glutathione S-transferase 2target
GlutathioneGlutathione S-transferase omega-2target
GlutathioneGlutaredoxin-2, mitochondrialtarget
GlutathioneGlutathione S-transferase A2enzyme
GlutathioneGlutathione S-transferase A1enzyme
GlutathioneMultidrug resistance-associated protein 1transporter
GlutathioneCanalicular multispecific organic anion transporter 1transporter
GlutathioneCanalicular multispecific organic anion transporter 2transporter
GlutathioneMultidrug resistance-associated protein 4transporter
GlutathioneMultidrug resistance-associated protein 5transporter
GlutathioneAldose reductasetarget
GlutathioneMatrix metalloproteinase-9target
GlutathioneCytochrome P450 3A4target
GlutathioneGlutathione peroxidasetarget
PentagastrinGastrin/cholecystokinin type B receptortarget
CeruletideCholecystokinin receptor type Atarget
EnalaprilAngiotensin-converting enzymetarget
EnalaprilP-glycoprotein 1transporter
EnalaprilSolute carrier family 15 member 1transporter
EnalaprilSolute carrier family 22 member 6transporter
EnalaprilSolute carrier family 22 member 8transporter
EnalaprilSolute carrier family 22 member 7transporter
EnalaprilSolute carrier organic anion transporter family member 1A2transporter
EnalaprilSerum albumincarrier
GonadorelinGonadotropin-releasing hormone receptortarget
GonadorelinPutative gonadotropin-releasing hormone II receptortarget
NafarelinGonadotropin-releasing hormone receptortarget
NafarelinPutative gonadotropin-releasing hormone II receptortarget
LisinoprilAngiotensin-converting enzymetarget
LisinoprilSolute carrier family 15 member 1transporter
LisinoprilSolute carrier family 15 member 2transporter
SpiraprilAngiotensin-converting enzymetarget
SpiraprilSolute carrier family 15 member 1transporter
SpiraprilSolute carrier family 15 member 2transporter
BuserelinLutropin-choriogonadotropic hormone receptortarget
BuserelinGonadotropin-releasing hormone receptortarget
BuserelinCytochrome P450 19A1enzyme
GanirelixGonadotropin-releasing hormone receptortarget
HistrelinGonadotropin-releasing hormone receptortarget
TriptorelinGonadotropin-releasing hormone receptortarget
ProtirelinThyrotropin Releasing Hormone Receptortarget
EnalaprilatAngiotensin-converting enzymetarget
EnalaprilatB1 bradykinin receptortarget
Angiotensin IIType-1 angiotensin II receptortarget
LypressinVasopressin V1a receptortarget
LypressinVasopressin V2 receptortarget
LypressinVasopressin V1b receptortarget
LypressinCanalicular multispecific organic anion transporter 1transporter
Glutathione disulfideGlutathione S-transferase Mu 2target
Glutathione disulfideGlutathione reductase, mitochondrialtarget
Glutathione disulfideGlutathione peroxidasetarget
Glutathione disulfideMicrosomal glutathione S-transferase 1target
Glutathione disulfideGlutathione S-transferases (Cytosolic)target
OrnithineOrnithine aminotransferase, mitochondrialtarget
OrnithineOrnithine carbamoyltransferase, mitochondrialtarget
OrnithineOrnithine decarboxylase antizyme 1target
OrnithineLow affinity cationic amino acid transporter 2target
OrnithineMitochondrial ornithine transporter 2target
OrnithineHigh affinity cationic amino acid transporter 1target
OrnithineArginase-2, mitochondrialtarget
OrnithineMitochondrial ornithine transporter 1target
OrnithineGlycine amidinotransferase, mitochondrialtarget
AtazanavirHuman immunodeficiency virus type 1 proteasetarget
AtazanavirCytochrome P450 3A4enzyme
AtazanavirCytochrome P450 2C9enzyme
AtazanavirP-glycoprotein 1transporter
AtazanavirMultidrug resistance-associated protein 1transporter
AtazanavirSerum albumincarrier
AtazanavirUDP-glucuronosyltransferase 1-1enzyme
AtazanavirSolute carrier organic anion transporter family member 1B1transporter
AtazanavirSolute carrier organic anion transporter family member 1B3transporter
AtazanavirCytochrome P450 2C8enzyme
AtazanavirBile salt export pumptransporter
Atazanaviralpha1-acid glycoproteincarrier
AtazanavirCytochrome P450 1A2enzyme
AtazanavirSolute carrier organic anion transporter family member 2B1transporter
AtazanavirCytochrome P450 3A5enzyme
AtazanavirCytochrome P450 3A7enzyme
FelypressinVasopressin V1a receptortarget
AspartameTaste receptor type 1 member 2target
AspartameTransient receptor potential cation channel subfamily V member 1target
AspartameSolute carrier family 22 member 6transporter
AspartameSolute carrier family 22 member 8transporter
AspartameSolute carrier family 22 member 11transporter
AspartameTaste receptor type 1 member 3target
IlomastatLethal factortarget
IlomastatDisintegrin and metalloproteinase domain-containing protein 28target
IlomastatAggrecan core proteintarget
S-(2,4-dinitrophenyl)glutathioneGlutathione S-transferase Mu 1target
S-(2,4-dinitrophenyl)glutathioneGlutathione S-transferase Mu 2target
TerlipressinVasopressin V1a receptortarget
TerlipressinVasopressin V2 receptortarget
TerlipressinVasopressin V1b receptortarget
JE-2147Gag-Pol polyproteintarget
N-(3-Propylcarbamoyloxirane-2-Carbonyl)-Isoleucyl-ProlineCathepsin Btarget
S-octylglutathioneGlutathione S-transferase Mu 4target
gamma-GlutamylcysteineGlutathione synthetasetarget
TrypanothioneTrypanothione reductasetarget
Z-Pro-ProlinalProlyl endopeptidasetarget
Z-Pro-ProlinalProlyl endopeptidasetarget
S-benzylglutathioneLactoylglutathione lyasetarget
S-benzylglutathioneGlutathione S-transferase A1target
S-benzylglutathioneGlutathione S-transferase A1enzyme
S-(4-nitrobenzyl)glutathioneGlutathione S-transferase Ptarget
S-(N-hydroxy-N-bromophenylcarbamoyl)glutathioneHydroxyacylglutathione hydrolase, mitochondrialtarget
S-HexylglutathioneLactoylglutathione lyasetarget
S-HexylglutathioneGlutathione S-transferase Mu 4target
S-HexylglutathioneGlutathione S-transferase Ptarget
S-HexylglutathioneGlutathione S-transferasetarget
S-HexylglutathioneGlutathione S-transferase A1target
S-HexylglutathioneGlutathione S-transferase theta-2target
S-HexylglutathioneGlutathione S-transferase A1enzyme
S-Methyl glutathioneGlutathione S-transferase Mu 2target
OlcegepantCalcitonin gene-related peptide 1target
OlcegepantCalcitonin gene-related peptide type 1 receptortarget
CanfosfamideGlutathione S-transferase Ptarget
EzatiostatGlutathione S-transferase Ptarget
GolotimodToll-like receptor 2target
GolotimodToll-like receptor 4target
GolotimodToll-like receptor 7target
GolotimodToll-like receptor 9target
VX-765Interleukin-1 betatarget
Sar9, Met (O2)11-Substance PCytochrome P450 19A1enzyme
Sar9, Met (O2)11-Substance PCholinesteraseenzyme
Sar9, Met (O2)11-Substance PProstaglandin G/H synthase 2enzyme
IcatibantB2 bradykinin receptortarget
IcatibantAminopeptidase Ntarget
SaxagliptinDipeptidyl peptidase 4target
SaxagliptinCytochrome P450 3A4enzyme
SaxagliptinCytochrome P450 3A5enzyme
SaxagliptinMultidrug resistance-associated protein 1transporter
SaxagliptinSolute carrier organic anion transporter family member 4C1transporter
SaxagliptinSolute carrier family 22 member 8transporter
LabradimilB2 bradykinin receptortarget
acetylleucyl-leucyl-norleucinalProteasome subunit alpha type-7target
KelatorphanLeukotriene A-4 hydrolasetarget
Brentuximab vedotinTumor necrosis factor receptor superfamily member 8target
Brentuximab vedotinCytochrome P450 3A4enzyme
Brentuximab vedotinATP-binding cassette sub-family B member 5transporter
PolaprezincTumor necrosis factortarget
PolaprezincSuperoxide dismutase [Cu-Zn]enzyme
PolaprezincHeme oxygenase 1enzyme
PolaprezincSuperoxide dismutase [Mn], mitochondrialenzyme
PolaprezincGlutathione S-transferase theta-1enzyme
PolaprezincGlutathione peroxidase 1enzyme
PolaprezincPeroxiredoxin-5, mitochondrialenzyme
PolaprezincVascular endothelial growth factor receptor 1target
PolaprezincBeta-nerve growth factortarget
PolaprezincPlatelet-derived growth factor receptor betatarget
PolaprezincHeat shock protein HSP 90-alphatarget
PolaprezincHeat shock protein HSP 90-betatarget
CA-074 methyl esterCathepsin Btarget