Janus Kinase Inhibitors

Name
Janus Kinase Inhibitors
Accession Number
DBCAT004108
Description

Agents that inhibit JANUS KINASES.

Drugs
DrugDrug Description
TofacitinibA Janus kinase (JAK) inhibitor used to treat rheumatic conditions, such as rheumatoid arthritis and ankylosing spondylitis, and ulcerative colitis.
BaricitinibA Janus kinase inhibitor used to treat moderate to severe rheumatoid arthritis that has responded poorly to at least one TNF antagonist.
UpadacitinibAn oral Janus kinase (JAK)1-selective inhibitor used in the treatment of moderate to severe rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, and severe atopic dermatitis, including in patients who did not respond well to other therapies.
AbrocitinibA kinase inhibitor used to treat moderate-to-severe atopic dermatitis in adults.
DeucravacitinibA TYK2 inhibitor being investigated as a treatment for psoriasis.
RitlecitinibA kinase inhibitor used to treat severe alopecia areata in adults and adolescents 12 years and older.
Drugs & Drug Targets
DrugTargetType
TofacitinibNon-receptor tyrosine-protein kinase TYK2target
TofacitinibCytochrome P450 3A4enzyme
TofacitinibCytochrome P450 2C19enzyme
TofacitinibTyrosine-protein kinase JAK2target
TofacitinibTyrosine-protein kinase JAK1target
TofacitinibTyrosine-protein kinase JAK3target
TofacitinibSerum albumincarrier
BaricitinibSolute carrier family 22 member 8transporter
BaricitinibATP-binding cassette sub-family G member 2transporter
BaricitinibMultidrug and toxin extrusion protein 2transporter
BaricitinibCytochrome P450 3A4enzyme
BaricitinibTyrosine-protein kinase JAK1target
BaricitinibTyrosine-protein kinase JAK2target
BaricitinibSolute carrier family 22 member 6transporter
BaricitinibSolute carrier family 22 member 2transporter
BaricitinibSolute carrier organic anion transporter family member 1B3transporter
BaricitinibTyrosine-protein kinase JAK3target
BaricitinibP-glycoprotein 1transporter
BaricitinibNon-receptor tyrosine-protein kinase TYK2target
UpadacitinibTyrosine-protein kinase JAK1target
UpadacitinibCytochrome P450 3A4enzyme
UpadacitinibCytochrome P450 2D6enzyme
UpadacitinibP-glycoprotein 1transporter
UpadacitinibATP-binding cassette sub-family G member 2transporter
UpadacitinibSolute carrier organic anion transporter family member 1B1transporter
AbrocitinibCytochrome P450 2C19enzyme
AbrocitinibCytochrome P450 2C9enzyme
AbrocitinibCytochrome P450 3A4enzyme
AbrocitinibCytochrome P450 2B6enzyme
AbrocitinibTyrosine-protein kinase JAK1target
AbrocitinibP-glycoprotein 1transporter
AbrocitinibSolute carrier family 22 member 1transporter
AbrocitinibTyrosine-protein kinase JAK2target
AbrocitinibTyrosine-protein kinase JAK3target
AbrocitinibNon-receptor tyrosine-protein kinase TYK2target
AbrocitinibSerum albumincarrier
AbrocitinibSolute carrier family 22 member 8transporter
DeucravacitinibNon-receptor tyrosine-protein kinase TYK2target
DeucravacitinibCytochrome P450 1A2enzyme
DeucravacitinibCytochrome P450 2B6enzyme
DeucravacitinibCytochrome P450 2D6enzyme
DeucravacitinibCocaine esteraseenzyme
DeucravacitinibUDP-glucuronosyltransferase 1-9enzyme
DeucravacitinibP-glycoprotein 1transporter
DeucravacitinibATP-binding cassette sub-family G member 2transporter
DeucravacitinibSolute carrier family 22 member 1transporter
DeucravacitinibSolute carrier organic anion transporter family member 1B3transporter
RitlecitinibTyrosine-protein kinase JAK3target
RitlecitinibTyrosine-protein kinase Tectarget
RitlecitinibTyrosine-protein kinase ITK/TSKtarget
RitlecitinibTyrosine-protein kinase TXKtarget
RitlecitinibTyrosine-protein kinase BTKtarget
RitlecitinibCytoplasmic tyrosine-protein kinase BMXtarget
RitlecitinibCytochrome P450 3A4enzyme
RitlecitinibCytochrome P450 2C8enzyme
RitlecitinibCytochrome P450 1A2enzyme
RitlecitinibCytochrome P450 2C9enzyme
RitlecitinibGlutathione S-transferase A1enzyme
RitlecitinibGlutathione S-transferase A3enzyme
RitlecitinibGlutathione S-transferase Mu 1enzyme
RitlecitinibGlutathione S-transferase Mu 3enzyme
RitlecitinibGlutathione S-transferase Mu 5enzyme
RitlecitinibGlutathione S-transferase Penzyme
RitlecitinibGlutathione S-transferase theta-2enzyme
RitlecitinibMaleylacetoacetate isomeraseenzyme
RitlecitinibMicrosomal glutathione S-transferase 1enzyme
RitlecitinibMicrosomal glutathione S-transferase 2enzyme
RitlecitinibMicrosomal glutathione S-transferase 3enzyme