| DB00851 | Dacarbazine | approved, investigational | unknown | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitorinducer | Details |
| DB00176 | Fluvoxamine | approved, investigational | unknown | inhibitor | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrate | Details |
| DB00468 | Quinine | approved | unknown | inhibitorinducer | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00730 | Thiabendazole | approved, vet_approved | unknown | inducer | Details |
| DB00889 | Granisetron | approved, investigational | unknown | substrate | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitorinducer | Details |
| DB01087 | Primaquine | approved | unknown | inducer | Details |
| DB04905 | Tesmilifene | investigational | unknown | substrate | Details |
| DB02709 | Resveratrol | investigational | no | substrateinhibitor | Details |
| DB04957 | Azimilide | investigational | unknown | substrate | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | substrateinhibitor | Details |
| DB00381 | Amlodipine | approved | unknown | inhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | substrateinhibitor | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | substrate | Details |
| DB04841 | Flunarizine | approved | unknown | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | substrate | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrateinducer | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00518 | Albendazole | approved, vet_approved | unknown | inducer | Details |
| DB00613 | Amodiaquine | approved, investigational | unknown | substrate | Details |
| DB01393 | Bezafibrate | approved, investigational | unknown | inducer | Details |
| DB00201 | Caffeine | approved | unknown | inhibitor | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01407 | Clenbuterol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00636 | Clofibrate | approved, investigational | unknown | inducer | Details |
| DB00363 | Clozapine | approved | no | inducer | Details |
| DB00169 | Cholecalciferol | approved, nutraceutical | unknown | inhibitor | Details |
| DB04840 | Debrisoquine | approved, investigational | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inhibitorinducer | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00898 | Ethanol | approved | unknown | inhibitor | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB01064 | Isoprenaline | approved, investigational | unknown | inhibitorinducer | Details |
| DB01167 | Itraconazole | approved, investigational | no | inducer | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inducer | Details |
| DB00643 | Mebendazole | approved, vet_approved | unknown | inducer | Details |
| DB00553 | Methoxsalen | approved | unknown | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | substrateinducer | Details |
| DB01115 | Nifedipine | approved | unknown | inhibitor | Details |
| DB00325 | Nitroprusside | approved, investigational | unknown | inhibitor | Details |
| DB01059 | Norfloxacin | approved | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inducer | Details |
| DB00740 | Riluzole | approved, investigational | unknown | substrate | Details |
| DB00605 | Sulindac | approved, investigational | unknown | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00277 | Theophylline | approved | unknown | substrateinhibitor | Details |
| DB00539 | Toremifene | approved, investigational | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inducer | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB00738 | Pentamidine | approved, investigational | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrate | Details |
| DB00575 | Clonidine | approved | unknown | substrate | Details |
| DB02342 | 2-Methoxyestradiol | investigational | unknown | | Details |
| DB04975 | Banoxantrone | investigational | unknown | substrate | Details |
| DB06770 | Benzyl alcohol | approved | unknown | inhibitor | Details |
| DB00633 | Dexmedetomidine | approved, vet_approved | unknown | inhibitor | Details |
| DB00466 | Picrotoxin | experimental | unknown | inducer | Details |
| DB00428 | Streptozocin | approved, investigational | unknown | inducer | Details |
| DB00165 | Pyridoxine | approved, investigational, nutraceutical, vet_approved | no | inhibitor | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB08846 | Ellagic acid | investigational | unknown | inhibitorinducer | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB08931 | Riociguat | approved | no | substrate | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB08922 | Perospirone | experimental | unknown | substrate | Details |
| DB12379 | Indirubin | investigational | unknown | substrate | Details |
| DB09238 | Manidipine | approved, investigational | unknown | inhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitorinducer | Details |
| DB11155 | Triclocarban | approved | unknown | inducer | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inducer | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB00550 | Propylthiouracil | approved, investigational | no | inducer | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrate | Details |
| DB00455 | Loratadine | approved, investigational | no | substrate | Details |
| DB01591 | Solifenacin | approved | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB11511 | Difloxacin | vet_approved | unknown | substrate | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB01132 | Pioglitazone | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inhibitorinducer | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | substrate | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | no | inhibitor | Details |
| DB08995 | Diosmin | approved, investigational | unknown | inducer | Details |
| DB16165 | Finerenone | approved, investigational | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitorinducer | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrate | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrate | Details |