| DB04665 | Coumarin | experimental | unknown | | Details |
| DB00184 | Nicotine | approved | unknown | substrateinhibitor | Details |
| DB01006 | Letrozole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrate | Details |
| DB00553 | Methoxsalen | approved | unknown | inhibitor | Details |
| DB00752 | Tranylcypromine | approved, investigational | unknown | inhibitor | Details |
| DB01011 | Metyrapone | approved, investigational | unknown | inhibitor | Details |
| DB01085 | Pilocarpine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | substrate | Details |
| DB04977 | Plitidepsin | investigational | unknown | substrate | Details |
| DB01115 | Nifedipine | approved | unknown | substrate | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01181 | Ifosfamide | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB00238 | Nevirapine | approved | unknown | substrate | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | substrate | Details |
| DB04841 | Flunarizine | approved | unknown | substrate | Details |
| DB00471 | Montelukast | approved | unknown | substrate | Details |
| DB07609 | N,N-DIMETHYL(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE | experimental | unknown | | Details |
| DB07617 | N-METHYL(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE | experimental | unknown | | Details |
| DB07621 | (5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE | experimental | unknown | | Details |
| DB07623 | 4,4'-DIPYRIDYL DISULFIDE | experimental | unknown | | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | unknown | inhibitor | Details |
| DB00972 | Azelastine | approved | unknown | substrateinhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB06470 | Clomethiazole | investigational | unknown | substrate | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitor | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00216 | Eletriptan | approved, investigational | unknown | inducer | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | substrate | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB01213 | Fomepizole | approved, vet_approved | unknown | inhibitor | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB01043 | Memantine | approved, investigational | unknown | inhibitor | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | inhibitor | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB06739 | Seratrodast | experimental | unknown | inhibitor | Details |
| DB01236 | Sevoflurane | approved, vet_approved | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB01274 | Arformoterol | approved, investigational | unknown | substrate | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | inhibitor | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | unknown | inducer | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09256 | Tegafur | approved, investigational | no | substrate | Details |
| DB09327 | Tegafur-uracil | approved, investigational | no | substrate | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrate | Details |
| DB09274 | Artesunate | approved, investigational | unknown | substrate | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | inhibitor | Details |
| DB00916 | Metronidazole | approved | unknown | substrate | Details |
| DB05676 | Apremilast | approved, investigational | unknown | substrate | Details |
| DB01039 | Fenofibrate | approved | unknown | inhibitor | Details |
| DB00717 | Norethisterone | approved | unknown | substrate | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inducer | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrate | Details |
| DB01222 | Budesonide | approved | unknown | inducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | inducer | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrate | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrate | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB15119 | Ropeginterferon alfa-2b | approved, investigational | no | inhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB12816 | Terpinen-4-ol | investigational | no | substrate | Details |
| DB06374 | Elacestrant | approved, investigational | unknown | substrate | Details |
| DB01194 | Brinzolamide | approved | no | substrate | Details |