| DB00184 | Nicotine | approved | unknown | substrateinhibitorinducer | Details |
| DB00228 | Enflurane | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrateinhibitor | Details |
| DB00753 | Isoflurane | approved, vet_approved | unknown | substrate | Details |
| DB00851 | Dacarbazine | approved, investigational | unknown | substrate | Details |
| DB00898 | Ethanol | approved | unknown | substrateinducer | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | substrate | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | substrateinducer | Details |
| DB01213 | Fomepizole | approved, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB01236 | Sevoflurane | approved, vet_approved | no | substrate | Details |
| DB00593 | Ethosuximide | approved | unknown | substrate | Details |
| DB00118 | Ademetionine | approved, investigational, nutraceutical | unknown | inhibitor | Details |
| DB00277 | Theophylline | approved | unknown | substrate | Details |
| DB00636 | Clofibrate | approved, investigational | unknown | inducer | Details |
| DB00780 | Phenelzine | approved | unknown | inducer | Details |
| DB00908 | Quinidine | approved, investigational | no | substrate | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB01115 | Nifedipine | approved | unknown | inhibitor | Details |
| DB01173 | Orphenadrine | approved | unknown | inhibitor | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB04977 | Plitidepsin | investigational | unknown | substrate | Details |
| DB05708 | GTS-21 | investigational | unknown | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB00468 | Quinine | approved | unknown | substrate | Details |
| DB05109 | Trabectedin | approved, investigational | unknown | substrate | Details |
| DB06728 | Aniline | experimental | unknown | substrate | Details |
| DB00822 | Disulfiram | approved | unknown | inhibitor | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB00201 | Caffeine | approved | no | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00969 | Alosetron | approved, withdrawn | unknown | inhibitor | Details |
| DB01223 | Aminophylline | approved | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | inhibitor | Details |
| DB04794 | Bifonazole | approved, investigational | unknown | inhibitor | Details |
| DB01558 | Bromazepam | approved, illicit, investigational | unknown | inhibitor | Details |
| DB01156 | Bupropion | approved | unknown | substrate | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitor | Details |
| DB01394 | Colchicine | approved | unknown | inducer | Details |
| DB01151 | Desipramine | approved, investigational | unknown | inhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01191 | Dexfenfluramine | approved, illicit, investigational, withdrawn | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | inhibitor | Details |
| DB01127 | Econazole | approved | no | inhibitor | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB01628 | Etoricoxib | approved, investigational | unknown | inhibitor | Details |
| DB00949 | Felbamate | approved | unknown | substrate | Details |
| DB00623 | Fluphenazine | approved | unknown | inhibitor | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | unknown | inhibitor | Details |
| DB09462 | Glycerin | approved, investigational | unknown | inducer | Details |
| DB00458 | Imipramine | approved | unknown | inhibitor | Details |
| DB00883 | Isosorbide dinitrate | approved, investigational | unknown | inhibitor | Details |
| DB01167 | Itraconazole | approved, investigational | no | inhibitor | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | inhibitor | Details |
| DB01011 | Metyrapone | approved, investigational | unknown | inhibitor | Details |
| DB00379 | Mexiletine | approved, investigational | unknown | substrate | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | substrate | Details |
| DB02701 | Nicotinamide | approved, investigational | unknown | substrateinhibitor | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | substrate | Details |
| DB00540 | Nortriptyline | approved | unknown | inhibitor | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrate | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | substrateinducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrateinhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01412 | Theobromine | investigational | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB00679 | Thioridazine | approved, withdrawn | unknown | inhibitor | Details |
| DB00208 | Ticlopidine | approved | unknown | inhibitor | Details |
| DB01007 | Tioconazole | approved | unknown | inhibitor | Details |
| DB00347 | Trimethadione | approved | unknown | substrate | Details |
| DB00617 | Paramethadione | approved | unknown | substrate | Details |
| DB04946 | Iloperidone | approved | unknown | substrate | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB06770 | Benzyl alcohol | approved | unknown | substrate | Details |
| DB06774 | Capsaicin | approved | unknown | substrate | Details |
| DB04920 | Clevidipine | approved, investigational | unknown | substrate | Details |
| DB00633 | Dexmedetomidine | approved, vet_approved | unknown | substrate | Details |
| DB06370 | Indisulam | investigational | unknown | inhibitor | Details |
| DB00109 | Enfuvirtide | approved, investigational | unknown | substrate | Details |
| DB00041 | Aldesleukin | approved | unknown | inhibitor | Details |
| DB04858 | Tirapazamine | investigational | unknown | substrate | Details |
| DB00428 | Streptozocin | approved, investigational | unknown | inducer | Details |
| DB06637 | Dalfampridine | approved | unknown | substrate | Details |
| DB08868 | Fingolimod | approved, investigational | unknown | substrate | Details |
| DB06201 | Rufinamide | approved | unknown | inhibitor | Details |
| DB01068 | Clonazepam | approved, illicit | unknown | inhibitor | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | inhibitor | Details |
| DB01595 | Nitrazepam | approved | unknown | inhibitor | Details |
| DB08846 | Ellagic acid | investigational | unknown | inhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inhibitor | Details |
| DB13174 | Rhein | experimental | unknown | inhibitor | Details |
| DB11994 | Diacerein | approved, investigational | unknown | inhibitor | Details |
| DB11943 | Delafloxacin | approved, investigational | unknown | inducer | Details |
| DB09120 | Zucapsaicin | approved, investigational | unknown | inhibitor | Details |
| DB13941 | Piperaquine | approved, experimental, investigational | unknown | inducer | Details |
| DB09328 | Vayarin | approved, investigational | unknown | inhibitor | Details |
| DB00486 | Nabilone | approved, investigational | no | substrateinhibitor | Details |
| DB04379 | N-Methyl-N-(Methylbenzyl)Formamide | experimental | unknown | substrate | Details |
| DB01154 | Thiamylal | approved, vet_approved | no | substrate | Details |
| DB09256 | Tegafur | approved, investigational | unknown | substrate | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB14046 | Dichlorobenzene | approved, experimental | unknown | substrate | Details |
| DB13963 | 1,2-dichlorobenzene | experimental | unknown | substrate | Details |
| DB01844 | N,N-dimethylformamide | experimental | unknown | substrate | Details |
| DB02520 | Ditiocarb | experimental | unknown | inhibitor | Details |
| DB00627 | Niacin | approved, investigational, nutraceutical | unknown | inhibitor | Details |
| DB04856 | Dexloxiglumide | investigational | unknown | substrate | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrate | Details |
| DB01104 | Sertraline | approved | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrate | Details |
| DB00794 | Primidone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00869 | Dorzolamide | approved | no | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB12466 | Favipiravir | approved, investigational | unknown | inhibitor | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB14840 | Ripretinib | approved | unknown | | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrate | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | substrate | Details |
| DB01189 | Desflurane | approved | no | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | substrate | Details |
| DB08995 | Diosmin | approved, investigational | unknown | inhibitor | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | no | substrate | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | no | substrateinhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB06016 | Cariprazine | approved, investigational | no | inhibitor | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |