| DB02974 | 4-(4-Chlorophenyl)Imidazole | experimental | unknown | | Details |
| DB04664 | Cyclohexyl-pentyl-maltoside | experimental | unknown | | Details |
| DB04794 | Bifonazole | approved, investigational | unknown | | Details |
| DB00333 | Methadone | approved | unknown | substrateinducer | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrateinducer | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | substrateinducer | Details |
| DB01104 | Sertraline | approved | unknown | substrateinhibitor | Details |
| DB01156 | Bupropion | approved | unknown | substrate | Details |
| DB01181 | Ifosfamide | approved | unknown | substrate | Details |
| DB00184 | Nicotine | approved | unknown | substrate | Details |
| DB00208 | Ticlopidine | approved | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB00238 | Nevirapine | approved | unknown | substrateinducer | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB00454 | Meperidine | approved | no | substrate | Details |
| DB00503 | Ritonavir | approved, investigational | no | inhibitorinducer | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrateinducer | Details |
| DB00758 | Clopidogrel | approved | no | substrateinhibitor | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00849 | Methylphenobarbital | approved | unknown | substrate | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01043 | Memantine | approved, investigational | unknown | inhibitor | Details |
| DB01173 | Orphenadrine | approved | unknown | inhibitor | Details |
| DB00381 | Amlodipine | approved | unknown | substrateinhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | substrateinhibitor | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB04572 | Thiotepa | approved, investigational | unknown | inhibitor | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB01069 | Promethazine | approved, investigational | unknown | substrate | Details |
| DB01221 | Ketamine | approved, vet_approved | unknown | substrate | Details |
| DB01320 | Fosphenytoin | approved, investigational | unknown | inducer | Details |
| DB01151 | Desipramine | approved, investigational | unknown | inhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | no | inhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitorinducer | Details |
| DB01167 | Itraconazole | approved, investigational | no | inhibitor | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | inhibitor | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | inhibitorinducer | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | inducer | Details |
| DB01076 | Atorvastatin | approved | no | inducer | Details |
| DB06739 | Seratrodast | experimental | unknown | substrate | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB03575 | Phencyclidine | illicit | unknown | inhibitor | Details |
| DB00865 | Benzphetamine | approved, illicit | unknown | substrate | Details |
| DB08369 | 1-(biphenyl-4-ylmethyl)-1H-imidazole | experimental | unknown | | Details |
| DB06697 | Artemether | approved | unknown | substrateinducer | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | inhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB06470 | Clomethiazole | investigational | unknown | substrate | Details |
| DB01559 | Clotiazepam | approved, illicit | unknown | substrate | Details |
| DB01394 | Colchicine | approved | unknown | inhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00751 | Epinastine | approved, investigational | unknown | substrate | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00898 | Ethanol | approved | unknown | inhibitor | Details |
| DB01466 | Ethylmorphine | experimental, illicit | unknown | substrate | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | substrate | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrate | Details |
| DB00176 | Fluvoxamine | approved, investigational | unknown | inhibitor | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | substrate | Details |
| DB00458 | Imipramine | approved | unknown | substrate | Details |
| DB00753 | Isoflurane | approved, vet_approved | unknown | substrateinducer | Details |
| DB06738 | Ketobemidone | investigational | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB01601 | Lopinavir | approved | unknown | inhibitor | Details |
| DB00772 | Malathion | approved, investigational | unknown | substrate | Details |
| DB04817 | Metamizole | approved, investigational, withdrawn | unknown | inducer | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB06710 | Methyltestosterone | approved | unknown | substrate | Details |
| DB00379 | Mexiletine | approved, investigational | unknown | substrate | Details |
| DB06148 | Mianserin | approved, investigational | unknown | substrate | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00745 | Modafinil | approved, investigational | unknown | inhibitorinducer | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | inducer | Details |
| DB01115 | Nifedipine | approved | unknown | inducer | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | inhibitor | Details |
| DB01074 | Perhexiline | approved, investigational | unknown | substrate | Details |
| DB04930 | Permethrin | approved, investigational | unknown | substrateinducer | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB00296 | Ropivacaine | approved | no | substrate | Details |
| DB00778 | Roxithromycin | approved, investigational, withdrawn | no | inhibitor | Details |
| DB01236 | Sevoflurane | approved, vet_approved | unknown | substrate | Details |
| DB06729 | Sulfaphenazole | approved | unknown | inhibitor | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | inducer | Details |
| DB00231 | Temazepam | approved, investigational | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB00193 | Tramadol | approved, investigational | unknown | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inducer | Details |
| DB00661 | Verapamil | approved | unknown | substrateactivator | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | inducer | Details |
| DB06413 | Armodafinil | approved, investigational | unknown | inducer | Details |
| DB00836 | Loperamide | approved | unknown | substrate | Details |
| DB04975 | Banoxantrone | investigational | unknown | substrate | Details |
| DB00435 | Nitric Oxide | approved | unknown | inhibitor | Details |
| DB00515 | Cisplatin | approved | unknown | inhibitor | Details |
| DB06209 | Prasugrel | approved | no | substrate | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB08899 | Enzalutamide | approved | no | inhibitor | Details |
| DB04938 | Ospemifene | approved, investigational | unknown | substrate | Details |
| DB09074 | Olaparib | approved | unknown | inducer | Details |
| DB09054 | Idelalisib | approved | no | inducer | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09280 | Lumacaftor | approved | no | inducer | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | inhibitor | Details |
| DB05219 | Crisaborole | approved, investigational | no | inhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inducer | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrate | Details |
| DB05541 | Brivaracetam | approved, investigational | no | substrate | Details |
| DB09238 | Manidipine | approved, investigational | unknown | inhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB12070 | Letermovir | approved, investigational | no | inducer | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13941 | Piperaquine | approved, experimental, investigational | unknown | inhibitor | Details |
| DB11642 | Pitolisant | approved, investigational | unknown | inducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inducer | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrate | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB13132 | Artemisinin | investigational | no | substrateinducer | Details |
| DB00582 | Voriconazole | approved | unknown | inhibitor | Details |
| DB14568 | Ivosidenib | approved, investigational | unknown | inducer | Details |
| DB00615 | Rifabutin | approved, investigational | no | inducer | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitorinducer | Details |
| DB01201 | Rifapentine | approved, investigational | no | inducer | Details |
| DB08883 | Perampanel | approved | unknown | substrateinducer | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB01095 | Fluvastatin | approved | unknown | inducer | Details |
| DB08912 | Dabrafenib | approved, investigational | no | inhibitorinducer | Details |
| DB08881 | Vemurafenib | approved | unknown | inducer | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | inducer | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | inhibitor | Details |
| DB11823 | Esketamine | approved, investigational | unknown | substrateinducer | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitorinducer | Details |
| DB00956 | Hydrocodone | approved, illicit, investigational | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | inhibitor | Details |
| DB04856 | Dexloxiglumide | investigational | unknown | substrate | Details |
| DB12808 | Trifarotene | approved, investigational | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB15035 | Zanubrutinib | approved, investigational | no | inducer | Details |
| DB14975 | Voxelotor | approved, investigational | unknown | substrate | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inducer | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB01222 | Budesonide | approved | unknown | inducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | inducer | Details |
| DB11951 | Lemborexant | approved, investigational | unknown | inducer | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | substrate | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB11932 | Abametapir | approved, investigational | unknown | inhibitor | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB11853 | Relugolix | approved, investigational | unknown | | Details |
| DB11632 | Opicapone | approved, investigational | no | inhibitor | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB00476 | Duloxetine | approved | unknown | inhibitor | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | substrate | Details |
| DB08822 | Azilsartan medoxomil | approved, investigational | no | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | inducer | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB08816 | Ticagrelor | approved | unknown | inducer | Details |
| DB15569 | Sotorasib | approved, investigational | unknown | inducer | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB15011 | Avacopan | approved, investigational | no | inducer | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitor | Details |
| DB14973 | Abrocitinib | approved, investigational | no | substrate | Details |
| DB16236 | Mitapivat | approved, investigational | no | inducer | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitorinducer | Details |
| DB05087 | Ganaxolone | approved, investigational | no | substrate | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB14921 | Mavacamten | approved, investigational | no | inducer | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | inhibitor | Details |
| DB12020 | Tecovirimat | approved, investigational | no | inducer | Details |
| DB09118 | Stiripentol | approved | unknown | inhibitorinducer | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | unknown | inhibitor | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inducer | Details |
| DB09499 | Thiosulfuric acid | approved, investigational | unknown | inducer | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | substrate | Details |
| DB02709 | Resveratrol | investigational | no | inhibitor | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | substrate | Details |
| DB16267 | Olutasidenib | approved, investigational | unknown | inducer | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inhibitorinducer | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | inducer | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB01194 | Brinzolamide | approved | unknown | substrate | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | inducer | Details |
| DB05467 | Palovarotene | approved, investigational | no | inducer | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | inhibitor | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitorinducer | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inducer | Details |
| DB12005 | Nirogacestat | approved, investigational | no | inducer | Details |
| DB06636 | Isavuconazonium | approved, investigational | unknown | inducer | Details |