| DB00176 | Fluvoxamine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | unknown | substrate | Details |
| DB00185 | Cevimeline | approved | unknown | substrate | Details |
| DB00193 | Tramadol | approved, investigational | unknown | substrate | Details |
| DB00243 | Ranolazine | approved, investigational | no | substrateinhibitor | Details |
| DB00264 | Metoprolol | approved, investigational | unknown | substrateinhibitor | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00285 | Venlafaxine | approved | unknown | substrateinhibitor | Details |
| DB00289 | Atomoxetine | approved | unknown | substrate | Details |
| DB00318 | Codeine | approved, illicit | unknown | substrate | Details |
| DB00370 | Mirtazapine | approved | unknown | substrate | Details |
| DB00373 | Timolol | approved | unknown | substrate | Details |
| DB00379 | Mexiletine | approved, investigational | unknown | substrate | Details |
| DB00433 | Prochlorperazine | approved, vet_approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | substrate | Details |
| DB00476 | Duloxetine | approved | unknown | substrateinhibitor | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00496 | Darifenacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00497 | Oxycodone | approved, illicit, investigational | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrateinhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB00521 | Carteolol | approved | unknown | substrate | Details |
| DB00557 | Hydroxyzine | approved | no | inhibitor | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00575 | Clonidine | approved | unknown | substrate | Details |
| DB00623 | Fluphenazine | approved | unknown | inhibitor | Details |
| DB00647 | Dextropropoxyphene | approved, illicit, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00656 | Trazodone | approved, investigational | unknown | substrateinhibitor | Details |
| DB00674 | Galantamine | approved | no | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrateinhibitor | Details |
| DB00679 | Thioridazine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00699 | Nicergoline | approved, investigational | unknown | substrate | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00734 | Risperidone | approved, investigational | unknown | substrateinhibitor | Details |
| DB00757 | Dolasetron | approved, investigational | unknown | substrate | Details |
| DB00805 | Minaprine | approved | unknown | substrate | Details |
| DB00843 | Donepezil | approved | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrateinhibitor | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | inhibitor | Details |
| DB00866 | Alprenolol | experimental, withdrawn | unknown | substrate | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrate | Details |
| DB00914 | Phenformin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB00934 | Maprotiline | approved, investigational | unknown | substrate | Details |
| DB00956 | Hydrocodone | approved, illicit, investigational | unknown | substrate | Details |
| DB00960 | Pindolol | approved, investigational | unknown | substrateinhibitor | Details |
| DB01012 | Cinacalcet | approved | unknown | inhibitor | Details |
| DB01035 | Procainamide | approved | unknown | substrate | Details |
| DB01036 | Tolterodine | approved, investigational | unknown | substrate | Details |
| DB01069 | Promethazine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01074 | Perhexiline | approved, investigational | unknown | substrateinhibitor | Details |
| DB01114 | Chlorpheniramine | approved | unknown | substrateinhibitor | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB01142 | Doxepin | approved, investigational | no | substrateinhibitor | Details |
| DB01151 | Desipramine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01193 | Acebutolol | approved, investigational | unknown | substrateinhibitor | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB01228 | Encainide | approved, investigational, withdrawn | unknown | substrate | Details |
| DB01233 | Metoclopramide | approved, investigational | unknown | substrateinhibitor | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01171 | Moclobemide | approved, investigational | unknown | substrateinhibitor | Details |
| DB01274 | Arformoterol | approved, investigational | unknown | substrate | Details |
| DB01410 | Ciclesonide | approved, investigational | unknown | substrate | Details |
| DB01466 | Ethylmorphine | experimental, illicit | unknown | substrate | Details |
| DB01409 | Tiotropium | approved | no | substrate | Details |
| DB01075 | Diphenhydramine | approved, investigational | unknown | substrateinhibitor | Details |
| DB04840 | Debrisoquine | approved, investigational | unknown | substrate | Details |
| DB00215 | Citalopram | approved | no | substrateinhibitor | Details |
| DB00234 | Reboxetine | approved, experimental | unknown | inhibitor | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | inhibitor | Details |
| DB00317 | Gefitinib | approved, investigational | no | substrateinhibitor | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrate | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrateinhibitor | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00458 | Imipramine | approved | unknown | substrateinhibitor | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitor | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00540 | Nortriptyline | approved | unknown | substrateinhibitor | Details |
| DB00613 | Amodiaquine | approved, investigational | unknown | inhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | inhibitor | Details |
| DB00705 | Delavirdine | approved | unknown | substrateinhibitor | Details |
| DB00726 | Trimipramine | approved | unknown | substrate | Details |
| DB00752 | Tranylcypromine | approved, investigational | unknown | inhibitor | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00933 | Mesoridazine | approved, investigational | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | substrateinhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01071 | Mequitazine | experimental | unknown | substrate | Details |
| DB01104 | Sertraline | approved | unknown | substrateinhibitor | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01115 | Nifedipine | approved | unknown | inhibitor | Details |
| DB01118 | Amiodarone | approved, investigational | no | inhibitor | Details |
| DB01131 | Proguanil | approved | no | inhibitor | Details |
| DB01149 | Nefazodone | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB01156 | Bupropion | approved | unknown | inhibitor | Details |
| DB01175 | Escitalopram | approved | no | substrateinhibitor | Details |
| DB01182 | Propafenone | approved | unknown | substrateinhibitor | Details |
| DB01191 | Dexfenfluramine | approved, illicit, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB01192 | Oxymorphone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01218 | Halofantrine | approved | unknown | inhibitor | Details |
| DB01238 | Aripiprazole | approved, investigational | no | substrate | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01551 | Dihydrocodeine | approved, illicit | unknown | substrate | Details |
| DB00377 | Palonosetron | approved, investigational | unknown | substrate | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | substrate | Details |
| DB04889 | Bicifadine | investigational | unknown | substrate | Details |
| DB01562 | 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine | experimental, illicit | unknown | inhibitor | Details |
| DB06144 | Sertindole | approved, investigational, withdrawn | unknown | substrate | Details |
| DB06148 | Mianserin | approved, investigational | unknown | substrate | Details |
| DB04905 | Tesmilifene | investigational | unknown | substrate | Details |
| DB01624 | Zuclopenthixol | approved, investigational | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrateinhibitor | Details |
| DB05271 | Rotigotine | approved | unknown | substrateinhibitor | Details |
| DB00472 | Fluoxetine | approved, vet_approved | no | substrateinhibitor | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | inhibitor | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00334 | Olanzapine | approved, investigational | no | substrateinhibitor | Details |
| DB00792 | Tripelennamine | approved, vet_approved | unknown | inhibitor | Details |
| DB00188 | Bortezomib | approved, investigational | unknown | substrate | Details |
| DB05109 | Trabectedin | approved, investigational | unknown | substrate | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | substrate | Details |
| DB04841 | Flunarizine | approved | unknown | substrate | Details |
| DB06726 | Bufuralol | experimental | unknown | substrate | Details |
| DB01472 | 4-Methoxyamphetamine | experimental, illicit | unknown | substrate | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB06727 | Sparteine | experimental, withdrawn | unknown | substrateinhibitor | Details |
| DB00283 | Clemastine | approved, investigational | unknown | inhibitor | Details |
| DB00907 | Cocaine | approved, illicit | unknown | inhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | no | substrateinhibitor | Details |
| DB00333 | Methadone | approved | no | substrateinhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB00211 | Midodrine | approved | unknown | substrate | Details |
| DB00208 | Ticlopidine | approved | unknown | substrateinhibitor | Details |
| DB00543 | Amoxapine | approved | unknown | substrateinhibitor | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB04946 | Iloperidone | approved | unknown | substrate | Details |
| DB01577 | Metamfetamine | approved, illicit, withdrawn | unknown | substrate | Details |
| DB01621 | Pipotiazine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00706 | Tamsulosin | approved, investigational | unknown | substrate | Details |
| DB04844 | Tetrabenazine | approved, investigational | unknown | substrate | Details |
| DB01601 | Lopinavir | approved | unknown | substrate | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB04855 | Dronedarone | approved | unknown | substrateinhibitor | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB06708 | Lumefantrine | approved | unknown | inhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | inhibitor | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB00238 | Nevirapine | approved | unknown | substrateinhibitor | Details |
| DB00216 | Eletriptan | approved, investigational | unknown | substrate | Details |
| DB00425 | Zolpidem | approved | unknown | substrate | Details |
| DB01628 | Etoricoxib | approved, investigational | unknown | inhibitor | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | substrate | Details |
| DB00381 | Amlodipine | approved | unknown | inhibitor | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | substrate | Details |
| DB01429 | Aprindine | experimental | unknown | substrate | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | substrate | Details |
| DB01244 | Bepridil | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00195 | Betaxolol | approved, investigational | unknown | substrate | Details |
| DB00810 | Biperiden | approved, investigational | unknown | inhibitor | Details |
| DB00297 | Bupivacaine | approved, investigational | unknown | substrate | Details |
| DB00490 | Buspirone | approved, investigational | unknown | substrate | Details |
| DB00201 | Caffeine | approved | unknown | substrate | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01093 | Dimethyl sulfoxide | approved, vet_approved | unknown | inhibitor | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00590 | Doxazosin | approved | unknown | substrate | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inhibitor | Details |
| DB00751 | Epinastine | approved, investigational | unknown | substrateinhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | inhibitor | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | substrateinhibitor | Details |
| DB01177 | Idarubicin | approved | unknown | substrate | Details |
| DB00224 | Indinavir | approved | unknown | inhibitor | Details |
| DB00598 | Labetalol | approved | unknown | substrateinhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inhibitor | Details |
| DB00528 | Lercanidipine | approved, investigational | unknown | inhibitor | Details |
| DB01206 | Lomustine | approved, investigational | unknown | inhibitor | Details |
| DB06691 | Mepyramine | approved, vet_approved | unknown | inhibitor | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | inhibitor | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB00220 | Nelfinavir | approved | no | inhibitor | Details |
| DB02701 | Nicotinamide | approved, investigational | unknown | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | substrate | Details |
| DB00627 | Niacin | approved, investigational, nutraceutical | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01096 | Oxamniquine | approved | unknown | substrateinhibitor | Details |
| DB01580 | Oxprenolol | approved | unknown | substrateinhibitor | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | inhibitor | Details |
| DB00738 | Pentamidine | approved, investigational | unknown | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB01100 | Pimozide | approved | no | inhibitor | Details |
| DB00592 | Piperazine | approved, vet_approved | unknown | substrate | Details |
| DB01087 | Primaquine | approved | unknown | inhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrate | Details |
| DB01224 | Quetiapine | approved | unknown | substrate | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB06729 | Sulfaphenazole | approved | unknown | inhibitor | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00277 | Theophylline | approved | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB01623 | Thiothixene | approved | unknown | inhibitor | Details |
| DB00209 | Trospium | approved | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB00570 | Vinblastine | approved | unknown | inhibitor | Details |
| DB00361 | Vinorelbine | approved, investigational | no | inhibitor | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB06287 | Temsirolimus | approved | unknown | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB01128 | Bicalutamide | approved | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inhibitor | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB06216 | Asenapine | approved | unknown | substrateinhibitor | Details |
| DB06589 | Pazopanib | approved | unknown | inhibitor | Details |
| DB06702 | Fesoterodine | approved | unknown | substrate | Details |
| DB06684 | Vilazodone | approved | unknown | substrate | Details |
| DB00836 | Loperamide | approved | unknown | substrate | Details |
| DB06506 | Repinotan | investigational | unknown | substrate | Details |
| DB06770 | Benzyl alcohol | approved | unknown | substrate | Details |
| DB04920 | Clevidipine | approved, investigational | unknown | substrate | Details |
| DB00633 | Dexmedetomidine | approved, vet_approved | unknown | inhibitor | Details |
| DB06370 | Indisulam | investigational | unknown | inhibitor | Details |
| DB06735 | Enclomiphene | investigational | unknown | substrate | Details |
| DB06204 | Tapentadol | approved | unknown | substrate | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrateinhibitor | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB08881 | Vemurafenib | approved | unknown | inhibitor | Details |
| DB08893 | Mirabegron | approved | no | substrateinhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrate | Details |
| DB06203 | Alogliptin | approved | unknown | substrate | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB09039 | Eliglustat | approved, investigational | no | substrateinhibitor | Details |
| DB09048 | Netupitant | approved, investigational | no | substrate | Details |
| DB09049 | Naloxegol | approved | unknown | inhibitor | Details |
| DB09076 | Umeclidinium | approved | no | substrate | Details |
| DB09065 | Cobicistat | approved | no | substrateinhibitor | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB06016 | Cariprazine | approved, investigational | no | substrateinhibitor | Details |
| DB00349 | Clobazam | approved, illicit | no | inhibitor | Details |
| DB09128 | Brexpiprazole | approved, investigational | no | substrate | Details |
| DB09291 | Rolapitant | approved, investigational | no | inhibitor | Details |
| DB06678 | Esmirtazapine | investigational | unknown | substrate | Details |
| DB06603 | Panobinostat | approved, investigational | no | inhibitor | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | inhibitor | Details |
| DB09183 | Dasabuvir | approved | no | substrate | Details |
| DB06512 | Deramciclane | investigational | unknown | inhibitor | Details |
| DB00022 | Peginterferon alfa-2b | approved | unknown | inhibitor | Details |
| DB00494 | Entacapone | approved, investigational | unknown | inhibitor | Details |
| DB04938 | Ospemifene | approved, investigational | unknown | inhibitor | Details |
| DB06820 | Sulconazole | approved | unknown | inhibitor | Details |
| DB08909 | Glycerol phenylbutyrate | approved | unknown | inhibitor | Details |
| DB00420 | Promazine | approved, vet_approved | unknown | substrate | Details |
| DB09118 | Stiripentol | approved | unknown | inhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | substrateinhibitor | Details |
| DB09555 | Dexchlorpheniramine maleate | approved | no | substrateinhibitor | Details |
| DB12161 | Deutetrabenazine | approved, investigational | no | substrate | Details |
| DB06217 | Vernakalant | approved, investigational | unknown | substrateinhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inhibitor | Details |
| DB11915 | Valbenazine | approved, investigational | no | substrate | Details |
| DB13174 | Rhein | experimental | unknown | inhibitor | Details |
| DB11994 | Diacerein | approved, investigational | unknown | inhibitor | Details |
| DB08922 | Perospirone | experimental | unknown | substrate | Details |
| DB09167 | Dosulepin | approved | unknown | substrateinhibitor | Details |
| DB11614 | Rupatadine | approved | no | substrate | Details |
| DB09238 | Manidipine | approved, investigational | unknown | inhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitor | Details |
| DB11638 | Artenimol | approved, experimental, investigational | unknown | inhibitor | Details |
| DB09195 | Lorpiprazole | approved | no | substrate | Details |
| DB09224 | Melperone | investigational | unknown | inhibitor | Details |
| DB11642 | Pitolisant | approved, investigational | unknown | substrateinhibitor | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB11130 | Opium | approved, illicit | no | substrate | Details |
| DB09053 | Ibrutinib | approved | no | substrate | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrateinhibitor | Details |
| DB14010 | 5-methoxy-N,N-dimethyltryptamine | experimental, illicit | unknown | substrate | Details |
| DB13975 | Black cohosh | experimental | no | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB13293 | Ipecac | approved, withdrawn | no | substrate | Details |
| DB04948 | Lofexidine | approved, investigational | no | substrate | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB04829 | Lysergic acid diethylamide | illicit, investigational, withdrawn | no | substrate | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | substrateinhibitor | Details |
| DB06608 | Tafenoquine | approved, investigational | no | substrate | Details |
| DB11979 | Elagolix | approved, investigational | no | substrate | Details |
| DB11785 | Anisodamine | investigational | no | substrate | Details |
| DB09204 | Arotinolol | investigational | no | substrate | Details |
| DB00335 | Atenolol | approved | no | substrate | Details |
| DB09013 | Befunolol | experimental | no | substrate | Details |
| DB01295 | Bevantolol | experimental | no | substrate | Details |
| DB08807 | Bopindolol | experimental | no | substrate | Details |
| DB12752 | Bucindolol | investigational | no | substrate | Details |
| DB08808 | Bupranolol | experimental | no | substrate | Details |
| DB04846 | Celiprolol | approved, investigational | no | substrate | Details |
| DB13508 | Cloranolol | experimental | no | substrate | Details |
| DB13757 | Epanolol | experimental | no | substrate | Details |
| DB13443 | Esatenolol | experimental | no | substrate | Details |
| DB00187 | Esmolol | approved, withdrawn | no | substrate | Details |
| DB08952 | Indenolol | withdrawn | no | substrate | Details |
| DB12212 | Landiolol | investigational | no | substrate | Details |
| DB09351 | Levobetaxolol | approved, investigational | no | substrate | Details |
| DB01210 | Levobunolol | approved | no | substrate | Details |
| DB13530 | Mepindolol | experimental | no | substrate | Details |
| DB01214 | Metipranolol | approved | no | substrate | Details |
| DB01359 | Penbutolol | approved, investigational | no | substrate | Details |
| DB01297 | Practolol | approved | no | substrate | Details |
| DB00489 | Sotalol | approved | no | substrate | Details |
| DB11770 | Talinolol | investigational | no | substrate | Details |
| DB13775 | Tertatolol | experimental | no | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB04818 | Iproniazid | withdrawn | unknown | inhibitor | Details |
| DB01267 | Paliperidone | approved | unknown | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB04911 | Oritavancin | approved, investigational | unknown | inhibitorinducer | Details |
| DB04884 | Dapoxetine | investigational | no | substrate | Details |
| DB12693 | Ritanserin | investigational | no | inhibitor | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB11963 | Dacomitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB14025 | Clinafloxacin | investigational | unknown | inhibitor | Details |
| DB01323 | St. John's Wort | approved, investigational, nutraceutical | no | inhibitor | Details |
| DB01454 | Midomafetamine | experimental, illicit, investigational | no | substrate | Details |
| DB11855 | Revefenacin | approved, investigational | no | substrate | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB01576 | Dextroamphetamine | approved, illicit | no | substrate | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | inhibitor | Details |
| DB00737 | Meclizine | approved | no | substrate | Details |
| DB01591 | Solifenacin | approved | unknown | substrate | Details |
| DB13679 | Dexchlorpheniramine | experimental, investigational | unknown | substrateinhibitor | Details |
| DB12523 | Mizolastine | approved, investigational | unknown | inhibitor | Details |
| DB01173 | Orphenadrine | approved | unknown | inhibitor | Details |
| DB09173 | Butyrfentanyl | illicit | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB04957 | Azimilide | investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | substrateinhibitor | Details |
| DB01590 | Everolimus | approved | unknown | inhibitor | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB11732 | Lasmiditan | approved, investigational | no | inhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB15091 | Upadacitinib | approved, investigational | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrate | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | inhibitor | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB01264 | Darunavir | approved | unknown | inhibitor | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | substrateinhibitor | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | inhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | substrateinhibitor | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | substrate | Details |
| DB14840 | Ripretinib | approved | unknown | substrate | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB14881 | Oliceridine | approved, investigational | unknown | substrate | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | no | substrate | Details |
| DB15982 | Berotralstat | approved | no | inhibitor | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | substrateinhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | inhibitor | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB00745 | Modafinil | approved, investigational | unknown | inducer | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | substrate | Details |
| DB05316 | Pimavanserin | approved, investigational | unknown | substrate | Details |
| DB11753 | Rifamycin | approved, investigational | unknown | inhibitor | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB15119 | Ropeginterferon alfa-2b | approved, investigational | no | inhibitor | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB16703 | Belumosudil | approved, investigational | no | substrateinhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | no | substrate | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | inhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB05087 | Ganaxolone | approved, investigational | no | substrate | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | substrateinhibitor | Details |
| DB14921 | Mavacamten | approved, investigational | no | | Details |
| DB06083 | Tapinarof | approved, investigational | no | substrate | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inhibitor | Details |
| DB15149 | Futibatinib | approved, investigational | no | substrate | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | substrate | Details |
| DB05239 | Cobimetinib | approved, investigational | no | inhibitor | Details |
| DB02709 | Resveratrol | investigational | no | inhibitor | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inhibitor | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | substrate | Details |
| DB00862 | Vardenafil | approved | unknown | inhibitor | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrate | Details |
| DB00953 | Rizatriptan | approved | no | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB12005 | Nirogacestat | approved, investigational | no | substrate | Details |
| DB16200 | Iptacopan | approved, investigational | no | substrate | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | inhibitor | Details |