| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00224 | Indinavir | approved | unknown | substrateinhibitor | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB00468 | Quinine | approved | unknown | substrate | Details |
| DB00541 | Vincristine | approved, investigational | no | substrate | Details |
| DB00661 | Verapamil | approved | unknown | substrateinhibitor | Details |
| DB00683 | Midazolam | approved, illicit | unknown | substrate | Details |
| DB00694 | Daunorubicin | approved | unknown | inducer | Details |
| DB00758 | Clopidogrel | approved | no | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | substrate | Details |
| DB00864 | Tacrolimus | approved, investigational | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | no | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB13179 | Troleandomycin | approved | unknown | inhibitor | Details |
| DB04856 | Dexloxiglumide | investigational | unknown | substrate | Details |
| DB04957 | Azimilide | investigational | unknown | substrate | Details |
| DB06267 | Udenafil | approved, investigational | unknown | substrate | Details |
| DB06287 | Temsirolimus | approved | unknown | substrateinhibitor | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | substrate | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrate | Details |
| DB01181 | Ifosfamide | approved | unknown | substrate | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00540 | Nortriptyline | approved | unknown | substrate | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB00220 | Nelfinavir | approved | no | substrateinhibitor | Details |
| DB00238 | Nevirapine | approved | unknown | substrate | Details |
| DB06652 | Vicriviroc | investigational | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | substrate | Details |
| DB01211 | Clarithromycin | approved | unknown | substrateinhibitor | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | substrate | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00897 | Triazolam | approved, investigational | unknown | substrate | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | substrate | Details |
| DB01114 | Chlorpheniramine | approved | unknown | substrate | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | substrate | Details |
| DB00381 | Amlodipine | approved | unknown | substrateinhibitor | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrateinhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | substrate | Details |
| DB00528 | Lercanidipine | approved, investigational | unknown | substrate | Details |
| DB00401 | Nisoldipine | approved | unknown | substrate | Details |
| DB01054 | Nitrendipine | approved, investigational | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB01238 | Aripiprazole | approved, investigational | no | substrate | Details |
| DB00490 | Buspirone | approved, investigational | unknown | substrate | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00700 | Eplerenone | approved | unknown | substrate | Details |
| DB01216 | Finasteride | approved | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrate | Details |
| DB01100 | Pimozide | approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB01224 | Quetiapine | approved | unknown | substrate | Details |
| DB00938 | Salmeterol | approved | unknown | substrate | Details |
| DB00877 | Sirolimus | approved, investigational | no | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrate | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB00656 | Trazodone | approved, investigational | unknown | substrate | Details |
| DB00962 | Zaleplon | approved, illicit, investigational | unknown | substrate | Details |
| DB01167 | Itraconazole | approved, investigational | no | inhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00446 | Chloramphenicol | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00705 | Delavirdine | approved | unknown | inhibitor | Details |
| DB06730 | Gestodene | investigational | unknown | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB06731 | Seproxetine | investigational | unknown | inhibitor | Details |
| DB00582 | Voriconazole | approved | unknown | substrateinhibitor | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB06772 | Cabazitaxel | approved | unknown | substrate | Details |
| DB06697 | Artemether | approved | unknown | substrate | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | substrate | Details |
| DB00278 | Argatroban | approved, investigational | unknown | substrate | Details |
| DB00394 | Beclomethasone dipropionate | approved, investigational | unknown | inducer | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrateinducer | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | no | substrate | Details |
| DB00822 | Disulfiram | approved | unknown | substrate | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB01218 | Halofantrine | approved | unknown | substrate | Details |
| DB01103 | Quinacrine | investigational | no | substrate | Details |
| DB00745 | Modafinil | approved, investigational | no | substrateinducer | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | inhibitor | Details |
| DB00776 | Oxcarbazepine | approved | no | inhibitorinducer | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | substrate | Details |
| DB00497 | Oxycodone | approved, illicit, investigational | unknown | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB01174 | Phenobarbital | approved, investigational | no | inducer | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | no | substrate | Details |
| DB00206 | Reserpine | approved, investigational, withdrawn | unknown | inducer | Details |
| DB00444 | Teniposide | approved | no | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00862 | Vardenafil | approved | unknown | substrate | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB00588 | Fluticasone propionate | approved | unknown | substrateinhibitor | Details |
| DB00738 | Pentamidine | approved, investigational | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | no | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrate | Details |
| DB01259 | Lapatinib | approved, investigational | unknown | substrate | Details |
| DB04946 | Iloperidone | approved | unknown | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB06335 | Saxagliptin | approved | unknown | substrate | Details |
| DB06413 | Armodafinil | approved, investigational | unknown | inducer | Details |
| DB00575 | Clonidine | approved | unknown | substrate | Details |
| DB06419 | Cethromycin | investigational | unknown | substrate | Details |
| DB08873 | Boceprevir | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB06228 | Rivaroxaban | approved | unknown | substrate | Details |
| DB08883 | Perampanel | approved | no | substrate | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB06626 | Axitinib | approved, investigational | no | substrate | Details |
| DB08899 | Enzalutamide | approved | no | substrateinducer | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrate | Details |
| DB05773 | Trastuzumab emtansine | approved, investigational | unknown | substrate | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrate | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrate | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB09053 | Ibrutinib | approved | unknown | substrate | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | substrate | Details |
| DB06403 | Ambrisentan | approved, investigational | no | substrate | Details |
| DB06789 | Hydroxyprogesterone caproate | approved, investigational | unknown | substrate | Details |
| DB09297 | Paritaprevir | approved, investigational | no | substrate | Details |
| DB12161 | Deutetrabenazine | approved, investigational | no | substrate | Details |
| DB11915 | Valbenazine | approved, investigational | no | substrate | Details |
| DB08820 | Ivacaftor | approved | no | substrateinhibitor | Details |
| DB09054 | Idelalisib | approved | no | substrateinhibitor | Details |
| DB09065 | Cobicistat | approved | no | substrate | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inducer | Details |
| DB11574 | Elbasvir | approved | unknown | substrate | Details |
| DB12483 | Copanlisib | approved, investigational | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB09231 | Benidipine | experimental | no | substrate | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | substrateinducer | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB14011 | Nabiximols | investigational | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inducer | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | substrate | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | substrate | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | substrate | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | substrate | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | substrate | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | substrate | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | substrate | Details |
| DB01222 | Budesonide | approved | no | inducer | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB11703 | Acalabrutinib | approved, investigational | unknown | inhibitor | Details |
| DB01267 | Paliperidone | approved | unknown | substrate | Details |
| DB11737 | Icotinib | experimental, investigational | unknown | substrateinducer | Details |
| DB00909 | Zonisamide | approved, investigational | no | substrate | Details |
| DB09256 | Tegafur | approved, investigational | unknown | substrate | Details |
| DB12301 | Doravirine | approved, investigational | unknown | substrate | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrate | Details |
| DB09074 | Olaparib | approved | unknown | substrateinhibitor | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrate | Details |
| DB13867 | Fluticasone | approved, experimental | unknown | substrateinhibitorinducer | Details |
| DB08906 | Fluticasone furoate | approved | no | substrateinhibitorinducer | Details |
| DB01126 | Dutasteride | approved, investigational | no | substrate | Details |
| DB00905 | Bimatoprost | approved, investigational | unknown | substrate | Details |
| DB00916 | Metronidazole | approved | unknown | substrate | Details |
| DB00288 | Amcinonide | approved | unknown | inducer | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB11750 | Clobetasol | approved, experimental, investigational | unknown | inducer | Details |
| DB01013 | Clobetasol propionate | approved | unknown | inducer | Details |
| DB14652 | Clocortolone acetate | experimental | unknown | inducer | Details |
| DB13843 | Cloprednol | experimental | unknown | inducer | Details |
| DB14681 | Cortisone | experimental | unknown | inducer | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | inducer | Details |
| DB13003 | Cortivazol | investigational | unknown | inducer | Details |
| DB11921 | Deflazacort | approved, investigational | unknown | inducer | Details |
| DB11487 | Dexamethasone isonicotinate | vet_approved | unknown | inducer | Details |
| DB09095 | Difluocortolone | approved, investigational, withdrawn | unknown | inducer | Details |
| DB01047 | Fluocinonide | approved, investigational | unknown | inducer | Details |
| DB08971 | Fluocortolone | approved, withdrawn | unknown | inducer | Details |
| DB00324 | Fluorometholone | approved, investigational | unknown | inducer | Details |
| DB08970 | Fluprednidene | experimental | unknown | inducer | Details |
| DB14634 | Fluprednidene acetate | experimental | unknown | inducer | Details |
| DB13728 | Halometasone | experimental | unknown | inducer | Details |
| DB00253 | Medrysone | approved | unknown | inducer | Details |
| DB14659 | Melengestrol acetate | experimental | unknown | inducer | Details |
| DB09383 | Meprednisone | approved, investigational | unknown | inducer | Details |
| DB14644 | Methylprednisolone hemisuccinate | approved | unknown | inducer | Details |
| DB00764 | Mometasone | experimental | unknown | inducer | Details |
| DB14512 | Mometasone furoate | approved, investigational, vet_approved | no | inducer | Details |
| DB01384 | Paramethasone | experimental | unknown | inducer | Details |
| DB14633 | Prednisolone hemisuccinate | experimental | unknown | inducer | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB14646 | Prednisone acetate | approved, experimental, investigational | unknown | inducer | Details |
| DB13208 | Prednylidene | experimental | unknown | inducer | Details |
| DB00896 | Rimexolone | approved | unknown | inducer | Details |
| DB00620 | Triamcinolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00196 | Fluconazole | approved, investigational | unknown | inhibitor | Details |
| DB02520 | Ditiocarb | experimental | unknown | inhibitor | Details |
| DB00367 | Levonorgestrel | approved, investigational | unknown | substrate | Details |
| DB01016 | Glyburide | approved | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB11761 | Tenapanor | approved, investigational | unknown | substrate | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB04855 | Dronedarone | approved | unknown | substrateinhibitor | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrate | Details |
| DB15444 | Elexacaftor | approved, investigational | no | substrate | Details |
| DB00557 | Hydroxyzine | approved | no | substrate | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrateinhibitor | Details |
| DB11951 | Lemborexant | approved, investigational | unknown | substrate | Details |
| DB01115 | Nifedipine | approved | unknown | substrate | Details |
| DB01190 | Clindamycin | approved, vet_approved | unknown | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB15822 | Pralsetinib | approved, investigational | no | inhibitorinducer | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrateinhibitor | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inhibitorinducer | Details |
| DB14984 | Casimersen | approved, investigational | no | inhibitor | Details |
| DB12016 | Ponesimod | approved, investigational | unknown | substrate | Details |
| DB05316 | Pimavanserin | approved, investigational | unknown | substrate | Details |
| DB08816 | Ticagrelor | approved | unknown | substrateactivator | Details |
| DB16222 | Loncastuximab tesirine | approved, investigational | unknown | substrate | Details |
| DB12543 | Samidorphan | approved, investigational | no | substrate | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB16390 | Mobocertinib | approved, investigational | unknown | substrate | Details |
| DB12834 | Secnidazole | approved | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB06230 | Nalmefene | approved, investigational, withdrawn | no | substrate | Details |
| DB05087 | Ganaxolone | approved, investigational | no | substrate | Details |
| DB06016 | Cariprazine | approved, investigational | no | inducer | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | inhibitor | Details |
| DB14921 | Mavacamten | approved, investigational | no | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | substrate | Details |
| DB05239 | Cobimetinib | approved, investigational | no | | Details |
| DB12240 | Polatuzumab vedotin | approved, investigational | no | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inducer | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB09065 | Cobicistat | approved | yes | inhibitor | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrate | Details |
| DB12874 | Quizartinib | approved, investigational | no | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |
| DB01072 | Atazanavir | approved, investigational | unknown | inhibitor | Details |
| DB15114 | Vamorolone | approved, investigational | no | substrate | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inhibitor | Details |
| DB11679 | Fruquintinib | approved, investigational | no | substrate | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | substrate | Details |
| DB00648 | Mitotane | approved | unknown | inducer | Details |