| DB00188 | Bortezomib | approved, investigational | no | substrateinhibitor | Details |
| DB00213 | Pantoprazole | approved | unknown | substrateinhibitor | Details |
| DB00215 | Citalopram | approved | no | substrateinhibitor | Details |
| DB00220 | Nelfinavir | approved | no | substrateinducer | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB00273 | Topiramate | approved | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB00395 | Carisoprodol | approved | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00420 | Promazine | approved, vet_approved | unknown | substrate | Details |
| DB00444 | Teniposide | approved | unknown | substrate | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00546 | Adinazolam | experimental | unknown | substrate | Details |
| DB00582 | Voriconazole | approved | unknown | substrateinhibitor | Details |
| DB00665 | Nilutamide | approved, investigational | unknown | substrateinhibitor | Details |
| DB00679 | Thioridazine | approved, withdrawn | unknown | substrate | Details |
| DB00736 | Esomeprazole | approved, investigational | no | substrateinhibitor | Details |
| DB00738 | Pentamidine | approved, investigational | unknown | substrate | Details |
| DB00794 | Primidone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00849 | Methylphenobarbital | approved | unknown | substrate | Details |
| DB00949 | Felbamate | approved | unknown | inhibitor | Details |
| DB01018 | Guanfacine | approved, investigational | unknown | substrate | Details |
| DB01104 | Sertraline | approved | unknown | substrateinhibitor | Details |
| DB01124 | Tolbutamide | approved, investigational | unknown | substrate | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB01131 | Proguanil | approved | unknown | substrate | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB01171 | Moclobemide | approved, investigational | unknown | substrateinhibitor | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | substrateinducer | Details |
| DB01274 | Arformoterol | approved, investigational | unknown | substrate | Details |
| DB01320 | Fosphenytoin | approved, investigational | unknown | substrate | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | substrate | Details |
| DB00176 | Fluvoxamine | approved, investigational | no | inhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00208 | Ticlopidine | approved | unknown | substrateinhibitor | Details |
| DB00321 | Amitriptyline | approved | unknown | substrateinhibitor | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrate | Details |
| DB00455 | Loratadine | approved, investigational | no | substrateinhibitor | Details |
| DB00458 | Imipramine | approved | unknown | substrateinhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | no | inducer | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | inhibitor | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | inducer | Details |
| DB00745 | Modafinil | approved, investigational | unknown | inhibitor | Details |
| DB00752 | Tranylcypromine | approved, investigational | unknown | inhibitor | Details |
| DB00776 | Oxcarbazepine | approved | unknown | inhibitor | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrateinhibitor | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB06442 | Avasimibe | investigational | unknown | inhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | substrate | Details |
| DB01076 | Atorvastatin | approved | no | inhibitor | Details |
| DB01095 | Fluvastatin | approved | unknown | inhibitor | Details |
| DB00196 | Fluconazole | approved, investigational | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitor | Details |
| DB01142 | Doxepin | approved, investigational | no | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB05109 | Trabectedin | approved, investigational | unknown | substrate | Details |
| DB01418 | Acenocoumarol | approved, investigational | unknown | substrate | Details |
| DB00682 | Warfarin | approved | unknown | substrateinhibitor | Details |
| DB00540 | Nortriptyline | approved | unknown | substrate | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00972 | Azelastine | approved | unknown | substrateinhibitor | Details |
| DB01075 | Diphenhydramine | approved, investigational | unknown | substrate | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00446 | Chloramphenicol | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00758 | Clopidogrel | approved | no | substrate | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrate | Details |
| DB01355 | Hexobarbital | experimental | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB01175 | Escitalopram | approved | no | substrate | Details |
| DB06414 | Etravirine | approved | unknown | substrateinhibitor | Details |
| DB01181 | Ifosfamide | approved | unknown | substrate | Details |
| DB05246 | Methsuximide | approved | unknown | substrateinhibitor | Details |
| DB00726 | Trimipramine | approved | unknown | substrate | Details |
| DB00357 | Aminoglutethimide | approved, investigational | unknown | inducer | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | inhibitorinducer | Details |
| DB01601 | Lopinavir | approved | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB06413 | Armodafinil | approved, investigational | unknown | inhibitor | Details |
| DB00705 | Delavirdine | approved | unknown | inhibitor | Details |
| DB01241 | Gemfibrozil | approved | unknown | inhibitor | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB06268 | Sitaxentan | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB00216 | Eletriptan | approved, investigational | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrateinhibitor | Details |
| DB00425 | Zolpidem | approved | unknown | substrate | Details |
| DB01036 | Tolterodine | approved, investigational | unknown | substrate | Details |
| DB01283 | Lumiracoxib | approved, investigational | unknown | substrate | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrateinhibitor | Details |
| DB00672 | Chlorpropamide | approved, investigational | unknown | substrate | Details |
| DB01120 | Gliclazide | approved | unknown | substrate | Details |
| DB01016 | Glyburide | approved | unknown | substrate | Details |
| DB06739 | Seratrodast | experimental | unknown | substrate | Details |
| DB06697 | Artemether | approved | unknown | substrateinducer | Details |
| DB00945 | Acetylsalicylic acid | approved, vet_approved | unknown | inducer | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | substrateinhibitor | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | inhibitor | Details |
| DB00673 | Aprepitant | approved, investigational | unknown | substrateinhibitor | Details |
| DB00289 | Atomoxetine | approved | unknown | substrate | Details |
| DB01558 | Bromazepam | approved, illicit, investigational | unknown | substrate | Details |
| DB00297 | Bupivacaine | approved, investigational | unknown | substrate | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | inhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB06470 | Clomethiazole | investigational | unknown | substrate | Details |
| DB01559 | Clotiazepam | approved, illicit | unknown | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB01093 | Dimethyl sulfoxide | approved, vet_approved | unknown | inhibitor | Details |
| DB00590 | Doxazosin | approved | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00898 | Ethanol | approved | unknown | inhibitor | Details |
| DB01628 | Etoricoxib | approved, investigational | unknown | inhibitor | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB06738 | Ketobemidone | investigational | unknown | substrate | Details |
| DB00678 | Losartan | approved | unknown | inhibitor | Details |
| DB01043 | Memantine | approved, investigational | unknown | inhibitor | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | substrate | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | inhibitor | Details |
| DB00717 | Norethisterone | approved | unknown | substrateinducer | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | inhibitor | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | substrate | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | no | substrate | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | inducer | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01589 | Quazepam | approved, illicit | no | substrate | Details |
| DB01224 | Quetiapine | approved | unknown | substrate | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB00373 | Timolol | approved | unknown | substrate | Details |
| DB01007 | Tioconazole | approved | unknown | inhibitor | Details |
| DB00347 | Trimethadione | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | inhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | substrateinhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | inhibitor | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00980 | Ramelteon | approved, investigational | unknown | substrate | Details |
| DB01128 | Bicalutamide | approved | unknown | inhibitor | Details |
| DB01259 | Lapatinib | approved, investigational | unknown | substrate | Details |
| DB01621 | Pipotiazine | approved, investigational | unknown | substrate | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB04920 | Clevidipine | approved, investigational | unknown | inhibitor | Details |
| DB00109 | Enfuvirtide | approved, investigational | unknown | substrate | Details |
| DB00239 | Oxiconazole | approved | unknown | substrate | Details |
| DB06204 | Tapentadol | approved | unknown | substrate | Details |
| DB06209 | Prasugrel | approved | no | substrate | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB08864 | Rilpivirine | approved | unknown | substrateinhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB06626 | Axitinib | approved, investigational | no | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | inhibitor | Details |
| DB08899 | Enzalutamide | approved | no | inducer | Details |
| DB08895 | Tofacitinib | approved, investigational | no | substrate | Details |
| DB04938 | Ospemifene | approved, investigational | unknown | substrate | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | inhibitor | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB08932 | Macitentan | approved | no | substrate | Details |
| DB08933 | Luliconazole | approved | no | inhibitor | Details |
| DB09049 | Naloxegol | approved | unknown | inhibitor | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | | Details |
| DB09054 | Idelalisib | approved | no | inhibitor | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09280 | Lumacaftor | approved | no | inducer | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB09119 | Eslicarbazepine acetate | approved | no | inhibitor | Details |
| DB06789 | Hydroxyprogesterone caproate | approved, investigational | unknown | inducer | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB09118 | Stiripentol | approved | unknown | substrateinhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inhibitorinducer | Details |
| DB05541 | Brivaracetam | approved, investigational | no | substrate | Details |
| DB05351 | Dexlansoprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB09120 | Zucapsaicin | approved, investigational | unknown | inhibitor | Details |
| DB09198 | Lobeglitazone | experimental | no | inhibitor | Details |
| DB09167 | Dosulepin | approved | unknown | inhibitor | Details |
| DB09166 | Etizolam | experimental | unknown | substrate | Details |
| DB11614 | Rupatadine | approved | no | substrate | Details |
| DB12319 | Benzbromarone | investigational, withdrawn | unknown | inhibitor | Details |
| DB09238 | Manidipine | approved, investigational | unknown | inhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | inducer | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB11638 | Artenimol | approved, experimental, investigational | unknown | inhibitor | Details |
| DB13941 | Piperaquine | approved, experimental, investigational | unknown | substrateinhibitor | Details |
| DB11901 | Apalutamide | approved, investigational | no | inducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrate | Details |
| DB14011 | Nabiximols | investigational | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB11632 | Opicapone | approved, investigational | no | inducer | Details |
| DB13746 | Bioallethrin | approved, experimental | no | substrate | Details |
| DB04948 | Lofexidine | approved, investigational | no | substrate | Details |
| DB00598 | Labetalol | approved | unknown | substrate | Details |
| DB11967 | Binimetinib | approved, investigational | no | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | substrate | Details |
| DB12474 | Lynestrenol | approved, investigational | no | substrateinhibitor | Details |
| DB00615 | Rifabutin | approved, investigational | no | inducer | Details |
| DB01201 | Rifapentine | approved, investigational | no | inducer | Details |
| DB01220 | Rifaximin | approved, investigational | no | inducer | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB01483 | Barbital | illicit | no | substrateinducer | Details |
| DB00418 | Secobarbital | approved, vet_approved | no | inducer | Details |
| DB00599 | Thiopental | approved, vet_approved | no | substrate | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB14055 | (S)-Warfarin | experimental, investigational | unknown | substrate | Details |
| DB04911 | Oritavancin | approved, investigational | unknown | inhibitor | Details |
| DB06218 | Lacosamide | approved | unknown | substrate | Details |
| DB13762 | Dexrabeprazole | experimental | unknown | substrate | Details |
| DB12319 | Benzbromarone | investigational, withdrawn | unknown | inhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB00518 | Albendazole | approved, vet_approved | no | substrate | Details |
| DB14025 | Clinafloxacin | investigational | unknown | inhibitor | Details |
| DB06731 | Seproxetine | investigational | unknown | inhibitor | Details |
| DB14575 | Eslicarbazepine | approved | unknown | inhibitor | Details |
| DB01323 | St. John's Wort | approved, investigational, nutraceutical | no | substrateinducer | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrate | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB11823 | Esketamine | approved, investigational | unknown | substrate | Details |
| DB06684 | Vilazodone | approved | unknown | substrate | Details |
| DB12015 | Alpelisib | approved, investigational | unknown | inhibitor | Details |
| DB00977 | Ethinylestradiol | approved | unknown | inhibitor | Details |
| DB06730 | Gestodene | investigational | unknown | inhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrate | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | substrate | Details |
| DB00956 | Hydrocodone | approved, illicit, investigational | unknown | substrate | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | substrate | Details |
| DB08502 | Capravirine | investigational | unknown | substrate | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB01039 | Fenofibrate | approved | unknown | inhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB14975 | Voxelotor | approved, investigational | unknown | substrate | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inducer | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrateinhibitor | Details |
| DB01222 | Budesonide | approved | unknown | inducer | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | inducer | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | inhibitor | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB01006 | Letrozole | approved, investigational | unknown | inhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | inducer | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | substrateinhibitor | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | inducer | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB14881 | Oliceridine | approved, investigational | unknown | substrate | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB15093 | Somapacitan | approved, investigational | unknown | inhibitor | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrateinhibitor | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | substrateinhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB00935 | Oxymetazoline | approved, investigational | no | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB00476 | Duloxetine | approved | unknown | inhibitor | Details |
| DB00052 | Somatotropin | approved, investigational | unknown | inhibitor | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB14984 | Casimersen | approved, investigational | no | inhibitor | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | substrate | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB05271 | Rotigotine | approved | no | inhibitor | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | substrate | Details |
| DB12543 | Samidorphan | approved, investigational | no | substrate | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB16703 | Belumosudil | approved, investigational | no | inhibitor | Details |
| DB15463 | Belzutifan | approved, investigational | no | substrate | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB16220 | Lonapegsomatropin | approved, investigational | unknown | inhibitor | Details |
| DB16349 | Vicagrel | investigational | unknown | substrate | Details |
| DB12597 | Asciminib | approved, investigational | no | inhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB14973 | Abrocitinib | approved, investigational | no | substrate | Details |
| DB05467 | Palovarotene | approved, investigational | no | substrate | Details |
| DB16236 | Mitapivat | approved, investigational | no | inducer | Details |
| DB12834 | Secnidazole | approved | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | no | substrateinhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | substrate | Details |
| DB11697 | Pacritinib | approved, investigational | no | inhibitor | Details |
| DB05087 | Ganaxolone | approved, investigational | no | substrate | Details |
| DB06016 | Cariprazine | approved, investigational | no | inhibitor | Details |
| DB14921 | Mavacamten | approved, investigational | no | substrateinducer | Details |
| DB12020 | Tecovirimat | approved, investigational | no | inhibitor | Details |
| DB06083 | Tapinarof | approved, investigational | no | substrate | Details |
| DB00285 | Venlafaxine | approved | no | substrate | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inhibitor | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | substrateinhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | substrate | Details |
| DB02709 | Resveratrol | investigational | no | inhibitor | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inhibitorinducer | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | inducer | Details |
| DB00381 | Amlodipine | approved | no | inhibitor | Details |
| DB00862 | Vardenafil | approved | unknown | inhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB15669 | Fezolinetant | approved, investigational | no | substrate | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | substrate | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB14766 | Etrasimod | approved | no | substrate | Details |
| DB16826 | Repotrectinib | approved, investigational | no | inducer | Details |
| DB11679 | Fruquintinib | approved, investigational | no | substrate | Details |
| DB12005 | Nirogacestat | approved, investigational | unknown | substrateinducer | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | inhibitor | Details |