| DB00176 | Fluvoxamine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00188 | Bortezomib | approved, investigational | no | substrateinhibitor | Details |
| DB00201 | Caffeine | approved | unknown | substrateinhibitor | Details |
| DB00261 | Anagrelide | approved | unknown | substrateinhibitor | Details |
| DB00268 | Ropinirole | approved, investigational | unknown | substrate | Details |
| DB00277 | Theophylline | approved | unknown | substrate | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrateinhibitor | Details |
| DB00296 | Ropivacaine | approved | no | substrate | Details |
| DB00315 | Zolmitriptan | approved, investigational | no | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00334 | Olanzapine | approved, investigational | no | substrate | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00370 | Mirtazapine | approved | unknown | substrate | Details |
| DB00379 | Mexiletine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00382 | Tacrine | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00458 | Imipramine | approved | unknown | substrateinhibitor | Details |
| DB00476 | Duloxetine | approved | unknown | substrateinhibitor | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB00502 | Haloperidol | approved | unknown | substrate | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB00540 | Nortriptyline | approved | unknown | substrate | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB00655 | Estrone | approved | unknown | substrate | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB00682 | Warfarin | approved | unknown | substrate | Details |
| DB00697 | Tizanidine | approved, investigational | unknown | substrate | Details |
| DB00740 | Riluzole | approved, investigational | unknown | substrate | Details |
| DB00744 | Zileuton | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00851 | Dacarbazine | approved, investigational | unknown | substrate | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | substrate | Details |
| DB00978 | Lomefloxacin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00980 | Ramelteon | approved, investigational | unknown | substrate | Details |
| DB00998 | Frovatriptan | approved, investigational | unknown | substrate | Details |
| DB01002 | Levobupivacaine | approved, investigational | unknown | substrate | Details |
| DB01012 | Cinacalcet | approved | unknown | substrate | Details |
| DB01094 | Hesperetin | experimental | unknown | substrate | Details |
| DB01097 | Leflunomide | approved, investigational | unknown | substrate | Details |
| DB01100 | Pimozide | approved | unknown | substrate | Details |
| DB01165 | Ofloxacin | approved | unknown | inhibitor | Details |
| DB01182 | Propafenone | approved | unknown | substrateinhibitor | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | no | substrate | Details |
| DB00969 | Alosetron | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB01367 | Rasagiline | approved | unknown | substrate | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrate | Details |
| DB00467 | Enoxacin | approved, investigational | unknown | inhibitor | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00487 | Pefloxacin | approved | unknown | inhibitor | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00532 | Mephenytoin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00533 | Rofecoxib | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00730 | Thiabendazole | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00908 | Quinidine | approved, investigational | unknown | inhibitor | Details |
| DB00972 | Azelastine | approved | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB01059 | Norfloxacin | approved | unknown | inhibitor | Details |
| DB01418 | Acenocoumarol | approved, investigational | unknown | substrate | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB00377 | Palonosetron | approved, investigational | unknown | substrate | Details |
| DB05708 | GTS-21 | investigational | unknown | substrate | Details |
| DB06442 | Avasimibe | investigational | unknown | inhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | substrate | Details |
| DB01115 | Nifedipine | approved | unknown | substrateinhibitor | Details |
| DB00619 | Imatinib | approved | no | substrate | Details |
| DB00468 | Quinine | approved | unknown | substrate | Details |
| DB01142 | Doxepin | approved, investigational | no | substrate | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | inhibitorinducer | Details |
| DB00425 | Zolpidem | approved | unknown | substrate | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | inhibitor | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | substrate | Details |
| DB04841 | Flunarizine | approved | unknown | substrate | Details |
| DB00788 | Naproxen | approved, vet_approved | unknown | substrate | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB00553 | Methoxsalen | approved | unknown | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB00745 | Modafinil | approved, investigational | unknown | inducer | Details |
| DB00607 | Nafcillin | approved, investigational | unknown | inducer | Details |
| DB06732 | beta-Naphthoflavone | experimental | unknown | inducer | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01223 | Aminophylline | approved | unknown | substrate | Details |
| DB06216 | Asenapine | approved | unknown | substrate | Details |
| DB00195 | Betaxolol | approved, investigational | unknown | substrate | Details |
| DB04574 | Estrone sulfate | approved | unknown | substrate | Details |
| DB00629 | Guanabenz | approved, investigational | unknown | substrate | Details |
| DB01623 | Thiothixene | approved | unknown | substrate | Details |
| DB00831 | Trifluoperazine | approved, investigational | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | no | inducer | Details |
| DB01241 | Gemfibrozil | approved | unknown | inhibitor | Details |
| DB00752 | Tranylcypromine | approved, investigational | unknown | inhibitor | Details |
| DB01087 | Primaquine | approved | unknown | substrateinducer | Details |
| DB00758 | Clopidogrel | approved | no | substrate | Details |
| DB00420 | Promazine | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB01628 | Etoricoxib | approved, investigational | unknown | substrate | Details |
| DB01645 | Genistein | investigational | unknown | substrateinhibitor | Details |
| DB07453 | alpha-Naphthoflavone | experimental | unknown | | Details |
| DB02709 | Resveratrol | investigational | no | substrateinhibitorinducer | Details |
| DB00518 | Albendazole | approved, vet_approved | unknown | inducer | Details |
| DB01558 | Bromazepam | approved, illicit, investigational | unknown | substrate | Details |
| DB00215 | Citalopram | approved | no | inhibitor | Details |
| DB01151 | Desipramine | approved, investigational | unknown | product of | Details |
| DB01191 | Dexfenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | substrateinhibitor | Details |
| DB00898 | Ethanol | approved | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB00400 | Griseofulvin | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01283 | Lumiracoxib | approved, investigational | unknown | substrate | Details |
| DB00772 | Malathion | approved, investigational | unknown | substrate | Details |
| DB00934 | Maprotiline | approved, investigational | unknown | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitorinducer | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB06148 | Mianserin | approved, investigational | unknown | substrate | Details |
| DB00184 | Nicotine | approved | unknown | substrateinducer | Details |
| DB00806 | Pentoxifylline | approved, investigational | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrate | Details |
| DB00388 | Phenylephrine | approved | unknown | inducer | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | no | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inhibitorinducer | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inducer | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | inhibitor | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01405 | Temafloxacin | withdrawn | unknown | substrateinhibitor | Details |
| DB01412 | Theobromine | investigational | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB00208 | Ticlopidine | approved | unknown | inhibitor | Details |
| DB06264 | Tolperisone | investigational | unknown | substrate | Details |
| DB00384 | Triamterene | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | inhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | inhibitor | Details |
| DB01303 | Oxtriphylline | approved | unknown | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrate | Details |
| DB00418 | Secobarbital | approved, vet_approved | unknown | inducer | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrate | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrate | Details |
| DB06210 | Eltrombopag | approved | unknown | substrate | Details |
| DB06413 | Armodafinil | approved, investigational | unknown | inducer | Details |
| DB00575 | Clonidine | approved | unknown | substrate | Details |
| DB06594 | Agomelatine | approved, investigational | unknown | substrate | Details |
| DB06510 | Muraglitazar | investigational | unknown | substrate | Details |
| DB06770 | Benzyl alcohol | approved | unknown | substrate | Details |
| DB06774 | Capsaicin | approved | unknown | substrateinducer | Details |
| DB00633 | Dexmedetomidine | approved, vet_approved | unknown | inhibitor | Details |
| DB06235 | Vadimezan | investigational | unknown | substrate | Details |
| DB00461 | Nabumetone | approved | unknown | substrate | Details |
| DB06803 | Niclosamide | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00435 | Nitric Oxide | approved | unknown | inhibitor | Details |
| DB06820 | Sulconazole | approved | unknown | inhibitor | Details |
| DB00428 | Streptozocin | approved, investigational | unknown | inducer | Details |
| DB06589 | Pazopanib | approved | unknown | substrate | Details |
| DB08867 | Ulipristal | approved | no | substrate | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB08881 | Vemurafenib | approved | unknown | inhibitor | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB06626 | Axitinib | approved, investigational | no | substrate | Details |
| DB08910 | Pomalidomide | approved | unknown | substrate | Details |
| DB06290 | Simeprevir | approved | no | inhibitor | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | | Details |
| DB05812 | Abiraterone | approved | unknown | inhibitor | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB09330 | Osimertinib | approved | no | inducer | Details |
| DB06769 | Bendamustine | approved, investigational | no | substrate | Details |
| DB00105 | Interferon alfa-2b | approved | unknown | inhibitor | Details |
| DB05990 | Obeticholic acid | approved | unknown | inhibitordownregulator | Details |
| DB01173 | Orphenadrine | approved | unknown | inhibitor | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00008 | Peginterferon alfa-2a | approved, investigational | unknown | inhibitor | Details |
| DB00022 | Peginterferon alfa-2b | approved | unknown | inhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB11737 | Icotinib | experimental, investigational | unknown | substrate | Details |
| DB12161 | Deutetrabenazine | approved, investigational | no | substrate | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inhibitorinducer | Details |
| DB05015 | Belinostat | approved, investigational | unknown | inducer | Details |
| DB13174 | Rhein | experimental | unknown | inhibitor | Details |
| DB11994 | Diacerein | approved, investigational | unknown | inhibitor | Details |
| DB09120 | Zucapsaicin | approved, investigational | unknown | inhibitor | Details |
| DB09118 | Stiripentol | approved | unknown | substrateinhibitorinducer | Details |
| DB09198 | Lobeglitazone | experimental | no | inhibitor | Details |
| DB09167 | Dosulepin | approved | unknown | inhibitor | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB09225 | Zotepine | approved, investigational, withdrawn | no | substrate | Details |
| DB11642 | Pitolisant | approved, investigational | unknown | inducer | Details |
| DB13975 | Black cohosh | experimental | no | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitorinducer | Details |
| DB11198 | Peppermint oil | approved, investigational | unknown | inhibitor | Details |
| DB04948 | Lofexidine | approved, investigational | no | substrate | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB00238 | Nevirapine | approved | unknown | inhibitor | Details |
| DB11967 | Binimetinib | approved, investigational | no | substrate | Details |
| DB06654 | Safinamide | approved, investigational | unknown | inhibitor | Details |
| DB08883 | Perampanel | approved | unknown | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | unknown | inhibitor | Details |
| DB05928 | Dovitinib | investigational | unknown | inducer | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB14132 | 8-chlorotheophylline | experimental | no | substrate | Details |
| DB01320 | Fosphenytoin | approved, investigational | unknown | inducer | Details |
| DB00993 | Azathioprine | approved | no | substrate | Details |
| DB14029 | Furafylline | experimental | no | inhibitor | Details |
| DB04076 | Hypoxanthine | experimental | no | substrate | Details |
| DB12406 | Lisofylline | investigational | no | substrate | Details |
| DB02134 | Xanthine | experimental | no | substrate | Details |
| DB06771 | Besifloxacin | approved | no | inhibitor | Details |
| DB00827 | Cinoxacin | approved, investigational, withdrawn | no | inhibitor | Details |
| DB11511 | Difloxacin | vet_approved | no | inhibitor | Details |
| DB06160 | Garenoxacin | investigational | no | inhibitor | Details |
| DB01044 | Gatifloxacin | approved, investigational, withdrawn | no | inhibitor | Details |
| DB01155 | Gemifloxacin | approved, investigational | no | inhibitor | Details |
| DB00218 | Moxifloxacin | approved, investigational | no | inhibitor | Details |
| DB06600 | Nemonoxacin | investigational | no | inhibitor | Details |
| DB11443 | Orbifloxacin | vet_approved | no | inhibitor | Details |
| DB11774 | Pazufloxacin | investigational | no | inhibitor | Details |
| DB13823 | Pipemidic acid | experimental | no | inhibitor | Details |
| DB11892 | Prulifloxacin | investigational | no | inhibitor | Details |
| DB00817 | Rosoxacin | approved, investigational | no | inhibitor | Details |
| DB13772 | Rufloxacin | experimental | no | inhibitor | Details |
| DB11491 | Sarafloxacin | vet_approved, withdrawn | no | inhibitor | Details |
| DB13261 | Sitafloxacin | experimental, investigational | no | inhibitor | Details |
| DB01208 | Sparfloxacin | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB05488 | Technetium Tc-99m ciprofloxacin | investigational | no | inhibitor | Details |
| DB00685 | Trovafloxacin | approved, investigational, withdrawn | no | inhibitor | Details |
| DB01667 | 8-azaguanine | experimental | no | substrate | Details |
| DB04356 | 9-Deazaguanine | experimental | no | substrate | Details |
| DB02489 | 9-Methylguanine | experimental | no | substrate | Details |
| DB13573 | Acefylline | experimental | no | substrate | Details |
| DB13203 | Bamifylline | experimental | no | substrate | Details |
| DB14018 | Bromotheophylline | approved | no | substrate | Details |
| DB13812 | Bufylline | experimental | no | substrate | Details |
| DB09273 | Doxofylline | experimental | no | substrate | Details |
| DB13592 | Etamiphylline | experimental | no | substrate | Details |
| DB01482 | Fenethylline | experimental | no | substrate | Details |
| DB13634 | Pentifylline | experimental | no | substrate | Details |
| DB06479 | Propentofylline | investigational | unknown | substrate | Details |
| DB13449 | Proxyphylline | experimental | no | substrate | Details |
| DB09256 | Tegafur | approved, investigational | unknown | substrate | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB00280 | Disopyramide | approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | inducer | Details |
| DB09290 | Ramosetron | investigational | unknown | substrate | Details |
| DB09071 | Tasimelteon | approved, investigational | unknown | substrate | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | substrateinhibitor | Details |
| DB12945 | Dihydralazine | approved, experimental | unknown | substrateinhibitor | Details |
| DB11450 | Pimobendan | vet_approved | unknown | substrate | Details |
| DB08880 | Teriflunomide | approved | unknown | inducer | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | inhibitor | Details |
| DB08972 | Flumequine | withdrawn | unknown | inhibitor | Details |
| DB14025 | Clinafloxacin | investigational | unknown | inhibitor | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitor | Details |
| DB01056 | Tocainide | approved | no | substrateinhibitor | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | inhibitor | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00455 | Loratadine | approved, investigational | unknown | substrate | Details |
| DB05676 | Apremilast | approved, investigational | unknown | substrate | Details |
| DB11404 | Enrofloxacin | vet_approved | unknown | inhibitor | Details |
| DB00779 | Nalidixic acid | approved, investigational | unknown | inhibitor | Details |
| DB05396 | Albinterferon Alfa-2B | investigational | unknown | inhibitor | Details |
| DB12814 | Cepeginterferon alfa-2B | investigational | unknown | inhibitor | Details |
| DB15119 | Ropeginterferon alfa-2b | approved, investigational | no | inhibitor | Details |
| DB09122 | Peginterferon beta-1a | approved | unknown | downregulator | Details |
| DB00033 | Interferon gamma-1b | approved, investigational | unknown | inhibitor | Details |
| DB00068 | Interferon beta-1b | approved | unknown | inhibitor | Details |
| DB00060 | Interferon beta-1a | approved, investigational | unknown | inhibitor | Details |
| DB00069 | Interferon alfacon-1 | approved, investigational | unknown | inhibitor | Details |
| DB00018 | Interferon alfa-n3 | approved, investigational | unknown | inhibitor | Details |
| DB00011 | Interferon alfa-n1 | approved, investigational | unknown | inhibitor | Details |
| DB15131 | Interferon alfa-2c | investigational | unknown | inhibitor | Details |
| DB00034 | Interferon alfa-2a | approved, investigational | unknown | inhibitor | Details |
| DB05258 | Interferon alfa | investigational | unknown | inhibitor | Details |
| DB14999 | Human interferon beta | approved, investigational | unknown | downregulator | Details |
| DB01306 | Insulin aspart | approved | unknown | inducer | Details |
| DB09456 | Insulin beef | approved | unknown | inducer | Details |
| DB09564 | Insulin degludec | approved | no | inducer | Details |
| DB01307 | Insulin detemir | approved | no | inducer | Details |
| DB00047 | Insulin glargine | approved | unknown | inducer | Details |
| DB01309 | Insulin glulisine | approved | unknown | inducer | Details |
| DB00030 | Insulin human | approved, investigational | unknown | inducer | Details |
| DB00046 | Insulin lispro | approved | unknown | inducer | Details |
| DB11567 | Insulin peglispro | investigational | unknown | inducer | Details |
| DB00071 | Insulin pork | approved | unknown | inducer | Details |
| DB05115 | NN344 | investigational | unknown | inducer | Details |
| DB11568 | Insulin tregopil | investigational | unknown | inducer | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB01233 | Metoclopramide | approved, investigational | unknown | substrate | Details |
| DB04889 | Bicifadine | investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | inhibitor | Details |
| DB01195 | Flecainide | approved, withdrawn | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | inhibitor | Details |
| DB01072 | Atazanavir | approved, investigational | unknown | inhibitor | Details |
| DB15444 | Elexacaftor | approved, investigational | no | inhibitor | Details |
| DB00717 | Norethisterone | approved | unknown | substrate | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | inducer | Details |
| DB00794 | Primidone | approved, vet_approved | unknown | inducer | Details |
| DB00927 | Famotidine | approved | no | inhibitor | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB01601 | Lopinavir | approved | unknown | substrateinhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | inhibitor | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | inhibitor | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | inhibitor | Details |
| DB11932 | Abametapir | approved, investigational | no | substrateinhibitor | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB15093 | Somapacitan | approved, investigational | unknown | inducer | Details |
| DB15822 | Pralsetinib | approved, investigational | no | substrate | Details |
| DB06448 | Lonafarnib | approved, investigational | no | substrate | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | inhibitor | Details |
| DB08912 | Dabrafenib | approved, investigational | no | inhibitor | Details |
| DB11632 | Opicapone | approved, investigational | no | inhibitor | Details |
| DB00784 | Mefenamic acid | approved | unknown | substrateinhibitor | Details |
| DB00052 | Somatotropin | approved, investigational | unknown | inducer | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB15442 | Trilaciclib | approved, investigational | unknown | inducer | Details |
| DB14989 | Umbralisib | approved, investigational, withdrawn | unknown | substrate | Details |
| DB04854 | Febuxostat | approved | no | substrate | Details |
| DB01086 | Benzocaine | approved, investigational | unknown | substrate | Details |
| DB11564 | Insulin argine | experimental | unknown | inducer | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | no | inhibitor | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB12151 | Brincidofovir | approved, investigational | no | inhibitor | Details |
| DB16703 | Belumosudil | approved, investigational | no | inhibitor | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB16220 | Lonapegsomatropin | approved, investigational | unknown | inducer | Details |
| DB15011 | Avacopan | approved, investigational | no | inducer | Details |
| DB06234 | Maribavir | approved, investigational | no | substrate | Details |
| DB04216 | Quercetin | experimental, investigational | no | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | inducer | Details |
| DB16236 | Mitapivat | approved, investigational | no | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00470 | Dronabinol | approved, illicit | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | inhibitor | Details |
| DB11697 | Pacritinib | approved, investigational | no | inhibitorinducer | Details |
| DB06016 | Cariprazine | approved, investigational | no | inhibitor | Details |
| DB06083 | Tapinarof | approved, investigational | no | substrate | Details |
| DB01656 | Roflumilast | approved | no | substrate | Details |
| DB16650 | Deucravacitinib | approved, investigational | unknown | substrate | Details |
| DB11793 | Niraparib | approved, investigational | no | inducer | Details |
| DB16267 | Olutasidenib | approved, investigational | no | substrateinducer | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | inhibitor | Details |
| DB00349 | Clobazam | approved, illicit | no | substrate | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrateinhibitor | Details |
| DB11712 | Tezacaftor | approved, investigational | no | inhibitor | Details |
| DB15669 | Fezolinetant | approved, investigational | no | substrate | Details |
| DB14924 | Ritlecitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | inhibitor | Details |